AU2001284188A1 - Thiazolidine derivatives and its use as antifungal agent - Google Patents

Thiazolidine derivatives and its use as antifungal agent

Info

Publication number
AU2001284188A1
AU2001284188A1 AU2001284188A AU8418801A AU2001284188A1 AU 2001284188 A1 AU2001284188 A1 AU 2001284188A1 AU 2001284188 A AU2001284188 A AU 2001284188A AU 8418801 A AU8418801 A AU 8418801A AU 2001284188 A1 AU2001284188 A1 AU 2001284188A1
Authority
AU
Australia
Prior art keywords
antifungal agent
thiazolidine derivatives
nr3r4
thiazolidine
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001284188A
Other languages
English (en)
Inventor
Judi Charlotte Neuss
Michael Glen Orchard
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Oxford Glycosciences (UK) Ltd
Original Assignee
Oxford Glycosciences (UK) Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oxford Glycosciences (UK) Ltd filed Critical Oxford Glycosciences (UK) Ltd
Publication of AU2001284188A1 publication Critical patent/AU2001284188A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU2001284188A 2000-08-31 2001-08-30 Thiazolidine derivatives and its use as antifungal agent Abandoned AU2001284188A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0021419.7A GB0021419D0 (en) 2000-08-31 2000-08-31 Compounds
GB0021419 2000-08-31
PCT/GB2001/003860 WO2002022612A1 (en) 2000-08-31 2001-08-30 Thiazolidine derivatives and its use as antifungal agent

Publications (1)

Publication Number Publication Date
AU2001284188A1 true AU2001284188A1 (en) 2002-03-26

Family

ID=9898614

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001284188A Abandoned AU2001284188A1 (en) 2000-08-31 2001-08-30 Thiazolidine derivatives and its use as antifungal agent

Country Status (9)

Country Link
US (1) US6740670B2 (enExample)
EP (1) EP1313731B1 (enExample)
JP (1) JP2004509121A (enExample)
AT (1) ATE482954T1 (enExample)
AU (1) AU2001284188A1 (enExample)
DE (1) DE60143165D1 (enExample)
ES (1) ES2353685T3 (enExample)
GB (1) GB0021419D0 (enExample)
WO (1) WO2002022612A1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ544820A (en) * 2003-08-11 2009-02-28 Hoffmann La Roche Piperazine with or-substituted phenyl group and their use as GlyT1 inhibitors
KR101166342B1 (ko) 2004-03-15 2012-07-18 얀센 파마슈티카 엔.브이. 아편계 약물 수용체 조절자로서의 신규의 화합물
PL1828154T3 (pl) 2004-12-09 2009-10-30 Hoffmann La Roche Pochodne fenylopiperazynometanonu
MX2007006896A (es) 2004-12-15 2007-06-26 Hoffmann La Roche Fenil-metanonas bi- y triciclicas sustituidas como inhibidores del transportador 1 de glicina (glyt-1) para el tratamiento de la enfermedad de alzheimer.
US7485637B2 (en) 2005-01-04 2009-02-03 Hoffmann-La Roche Inc. Benzoyl-tetrahydropiperidine derivatives
ATE472327T1 (de) 2005-01-07 2010-07-15 Hoffmann La Roche Ä4-(heteroaryl)piperazin-1-ylü-(2,5-substituier e phenyl)methanon-derivate als glycin-transporter 1 (glyt-1) hemmer zur behandlung von neurologischen und neuropsychiatrischen erkrankungen
DE602006007682D1 (de) 2005-01-18 2009-08-20 Hoffmann La Roche 2,5-disubstituierte phenylmethanonderivative als glycintransporter-1-inhibitoren (glyt-1) zur behandlung von neurologischen und neuropsychiatrischen störungen
BRPI0607241A2 (pt) 2005-01-26 2009-08-25 Hoffmann La Roche derivados de fenil metanona e o uso dos mesmos como inibidores do transportador de glicina 1
WO2006082001A1 (en) 2005-02-07 2006-08-10 F.Hoffmann-La Roche Ag Heterocyclic substituted phenyl methanones as inhibitors of the glycine transporter 1
ATE536347T1 (de) 2008-05-20 2011-12-15 Merck Sharp & Dohme Effiziente herstellung heterologer proteine unter verwendung von mannosyltransferaseinhibitoren
US10059723B2 (en) 2011-02-28 2018-08-28 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
US8957066B2 (en) 2011-02-28 2015-02-17 Biomarin Pharmaceutical Inc. Histone deacetylase inhibitors
RU2662153C1 (ru) * 2017-04-20 2018-07-24 Общество С Ограниченной Ответственностью "Дермавитал Групп" Гибридные эфиры на основе производных тиазолидин-2,4-диона и азолов (1н-1,3-имидазола и 1н-1,3,4-триазола) и их применение
RU2690161C1 (ru) * 2018-06-28 2019-05-31 Общество С Ограниченной Ответственностью "Дермавитал Групп" 3,5-Замещенные производные тиазолидин-2,4-диона, обладающие противомикробной активностью
RU2703997C1 (ru) * 2018-12-13 2019-10-23 Общество с ограниченной ответственностью "Л-Био" Гибридные амиды на основе триазола и тиазолидина, обладающие антимикробной активностью
US11292776B2 (en) 2019-12-12 2022-04-05 University Of Sharjah Small molecule inhibitors of fungal hyphae and biofilm formation

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US47109A (en) * 1865-04-04 Improvement in governors
FR1604530A (enExample) * 1967-06-06 1971-11-29
JPS5740478A (en) * 1980-08-22 1982-03-06 Ono Pharmaceut Co Ltd Rhodanine derivative, its preparation and aldose reductase inhibitor containing rhodanine derivative
DE4318550A1 (de) * 1993-06-04 1994-12-08 Boehringer Mannheim Gmbh Aryliden-4-oxo-2-thioxo-3- thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE19835316A1 (de) * 1998-08-05 2000-02-10 Bosch Gmbh Robert Gesteuerte Gleichrichterbrücke mit Überspannungsschutz
AU6330799A (en) * 1998-09-30 2000-04-17 Roche Diagnostics Gmbh Rhodanine carboxylic acid derivatives for the treatment and prevention of metabolic bone disorders

Also Published As

Publication number Publication date
EP1313731B1 (en) 2010-09-29
ES2353685T3 (es) 2011-03-04
GB0021419D0 (en) 2000-10-18
US20030216453A1 (en) 2003-11-20
EP1313731A1 (en) 2003-05-28
DE60143165D1 (de) 2010-11-11
WO2002022612A1 (en) 2002-03-21
WO2002022612A8 (en) 2002-05-23
US6740670B2 (en) 2004-05-25
JP2004509121A (ja) 2004-03-25
ATE482954T1 (de) 2010-10-15

Similar Documents

Publication Publication Date Title
WO2002022612A8 (en) Thiazolidine derivatives and its use as antifungal agent
BR0208365A (pt) Derivados de 2-amino-propanol
AU2001284190A1 (en) Benzylidene thiazolidinediones and their use as antimycotic agents
DK109487A (da) Fungicid paa basis af et cyanopyrrolderivat
PT1078923E (pt) Processo para a preparacao de derivados de benzotiofeno
AU6055894A (en) Benzofuranyl- and -thiophenyl-alkanecarboxyclic acid derivatives
DE69010139D1 (de) Haarkräftigungsmittel.
WO2004063330A3 (en) (2-carboxamido) (3-amino) thiophene compounds
PT96664A (pt) Processo para a preparacao de derivados neuroprotectores de 3-piperidino-4-hidroxicromano
CA2194885A1 (en) Substituted benzamidines, their preparation and their use as pharmaceutical compounds
DE60221508D1 (de) Aminosäurederivate als hiv-protease-inhibitoren
ATE248187T1 (de) Echinocandin-kohlenhydrate-komplexe
WO2003030886A3 (en) Allylamides useful in the treatment of alzheimer's disease
AU1058492A (en) Improvements in or relating to organic compounds
AU8062487A (en) New substituted cephalosporin sulfones as anti-inflammatory and antidegenerative agents
AU9678501A (en) Pharmaceutical solutions of modafinil compounds
SI0843967T1 (en) Use of Beta-aminopropionic acid derivatives as fungicides
SE9904765D0 (sv) Pharmaceutically-useful compounds
CA2121123A1 (en) Anti-seborrhoeic formulation
AU5801286A (en) Spiro-imidazolidines as aldose reductase inhibitors
ATE250610T1 (de) Kaliumkanal-blockierende mittel
ATE317263T1 (de) Diphosphonat derivate von therapeutisch wirksamen stoffen
AU3565700A (en) Antibacterial agents
EP1207166A3 (en) Process for the preparation of 6.alpha.-fluoro,9,11.beta.-epoxy-steroids
CA2434408A1 (en) Process for the preparation of heterocyclic indene analogs