AU2001269698A1 - Heterocycle carboxamides as antiviral agents - Google Patents
Heterocycle carboxamides as antiviral agentsInfo
- Publication number
- AU2001269698A1 AU2001269698A1 AU2001269698A AU6969801A AU2001269698A1 AU 2001269698 A1 AU2001269698 A1 AU 2001269698A1 AU 2001269698 A AU2001269698 A AU 2001269698A AU 6969801 A AU6969801 A AU 6969801A AU 2001269698 A1 AU2001269698 A1 AU 2001269698A1
- Authority
- AU
- Australia
- Prior art keywords
- antiviral agents
- carboxamides
- heterocycle
- heterocycle carboxamides
- antiviral
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- -1 Heterocycle carboxamides Chemical class 0.000 title 1
- 239000003443 antiviral agent Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
- C07D217/14—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US21755600P | 2000-07-12 | 2000-07-12 | |
US60/217,556 | 2000-07-12 | ||
PCT/US2001/016492 WO2002004443A2 (fr) | 2000-07-12 | 2001-06-25 | Carboxamides heterocycliques utilises comme agents antiviraux |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001269698A1 true AU2001269698A1 (en) | 2002-01-21 |
Family
ID=22811560
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001269698A Abandoned AU2001269698A1 (en) | 2000-07-12 | 2001-06-25 | Heterocycle carboxamides as antiviral agents |
AU2001269697A Abandoned AU2001269697A1 (en) | 2000-07-12 | 2001-06-25 | Heterocycle carboxamides as antiviral agents |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001269697A Abandoned AU2001269697A1 (en) | 2000-07-12 | 2001-06-25 | Heterocycle carboxamides as antiviral agents |
Country Status (7)
Country | Link |
---|---|
US (2) | US6730682B2 (fr) |
EP (2) | EP1363907A2 (fr) |
JP (2) | JP2004502758A (fr) |
AR (2) | AR030244A1 (fr) |
AU (2) | AU2001269698A1 (fr) |
PE (2) | PE20020143A1 (fr) |
WO (2) | WO2002004422A2 (fr) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CZ20031028A3 (cs) | 2000-10-12 | 2003-08-13 | Merck & Co., Inc. | Aza- a polyazanaftalenylkarboxamidy |
DE60128936T2 (de) | 2000-10-12 | 2008-04-10 | Merck & Co, Inc. | Aza- und polyaza-naphthalenylcarbonsäureamide als hiv-integrase-hemmer |
WO2002055079A2 (fr) | 2000-10-12 | 2002-07-18 | Merck & Co Inc | Aza- et polyaza-naphthalenyl carboxamides convenant comme inhibiteurs de l'integrase du vih |
EP2033952B1 (fr) | 2001-03-01 | 2012-08-29 | Shionogi&Co., Ltd. | Composés d'hétéroaryle contenant de l'azote exerçant un effet inhibiteur sur l'intégrase du VIH |
AR036256A1 (es) | 2001-08-17 | 2004-08-25 | Merck & Co Inc | Sal sodica de un inhibidor de integrasa del vih, procesos para su preparacion, composiciones farmaceuticas que lo contienen y su uso para la manufactura de un medicamento |
ES2291642T3 (es) | 2002-01-17 | 2008-03-01 | MERCK & CO., INC. | Hidroxinaftiridinoncarboxamidas utiles como inhibidores de la integrasa de vih. |
JP4494020B2 (ja) | 2002-03-15 | 2010-06-30 | メルク・シャープ・エンド・ドーム・コーポレイション | Hivインテグラーゼ阻害剤として有用なn−(置換ベンジル)−8−ヒドロキシ−1,6−ナフチリジン−7−カルボキサミド |
BRPI0306214B1 (pt) * | 2002-11-20 | 2017-08-08 | Japan Tobacco Inc. | 4-oxoquinoline compound and use of this as a hiv integrase inhibitor |
DE10319612A1 (de) | 2003-05-02 | 2004-11-18 | Bayer Healthcare Ag | Substituierte Dihydrochinazoline |
DE10320780A1 (de) * | 2003-05-09 | 2005-01-20 | Bayer Healthcare Ag | Heterocyclyl-substituierte Dihydrochinazoline |
WO2004106334A2 (fr) * | 2003-05-28 | 2004-12-09 | Pfizer Products Inc. | Procede de preparation de 1,5-naphtyridine-3-carboxyamides par amidation directe d'esters |
DE10352499A1 (de) * | 2003-11-11 | 2005-06-09 | Bayer Healthcare Ag | Substituierte Dihydrochinazoline II |
DE102004022672A1 (de) * | 2004-05-07 | 2005-11-24 | Bayer Healthcare Ag | Substituierte Azachinazoline |
WO2005113509A1 (fr) * | 2004-05-20 | 2005-12-01 | Japan Tobacco Inc. | Nouveau composé 4-oxoquinoline et utilisation de celui-ci comme inhibiteur d'intégrase de vih |
GB0428475D0 (en) * | 2004-12-30 | 2005-02-02 | 4 Aza Bioscience Nv | Pyrido(3,2-D)pyrimidine derivatives and pharmaceutical compositions useful as medicines for the treatment of autoimmune disorders |
CN101166730A (zh) | 2005-03-01 | 2008-04-23 | 惠氏公司 | 噌啉化合物及其作为肝x受体调节剂的用途 |
DE102005027517A1 (de) * | 2005-06-15 | 2006-12-21 | Bayer Healthcare Ag | Verfahren zur Herstellung von Dihydrochinazolinen |
AU2006261607A1 (en) * | 2005-06-24 | 2006-12-28 | Gilead Sciences, Inc. | Pyrido(3,2-d)pyrimidines and pharmaceutical compositions useful for treating hepatitis C. |
IN2014CN00613A (fr) * | 2006-03-06 | 2015-08-21 | Japan Tobacco Inc | |
US8338435B2 (en) * | 2006-07-20 | 2012-12-25 | Gilead Sciences, Inc. | Substituted pyrido(3,2-D) pyrimidines and pharmaceutical compositions for treating viral infections |
US8143394B2 (en) * | 2006-12-26 | 2012-03-27 | Gilead Sciences, Inc. | Pyrido(3,2-d)pyrimidines useful for treating viral infections |
TW200840584A (en) * | 2006-12-26 | 2008-10-16 | Gilead Sciences Inc | Pyrido(3,2-d)pyrimidines useful for treating viral infections |
US8637531B2 (en) * | 2006-12-26 | 2014-01-28 | Gilead Sciences, Inc. | Pyrido(3,2-d)pyridmidines useful for treating viral infections |
US8536187B2 (en) * | 2008-07-03 | 2013-09-17 | Gilead Sciences, Inc. | 2,4,6-trisubstituted pyrido(3,2-d)pyrimidines useful for treating viral infections |
EP3317277B1 (fr) | 2015-07-01 | 2021-01-20 | Crinetics Pharmaceuticals, Inc. | Modulateurs de la somatostatine et leurs utilisations |
WO2017058242A1 (fr) * | 2015-10-02 | 2017-04-06 | United Technologies Corporation | Cellule électronique de puissance universelle pour production distribuée |
US11028068B2 (en) | 2017-07-25 | 2021-06-08 | Crinetics Pharmaceuticals, Inc. | Somatostatin modulators and uses thereof |
CN112890578A (zh) | 2017-08-09 | 2021-06-04 | 沙克忍者运营有限责任公司 | 烹饪系统 |
KR20230170813A (ko) | 2018-09-12 | 2023-12-19 | 노파르티스 아게 | 항바이러스 피리도피라진디온 화합물 |
US11667613B2 (en) | 2019-09-26 | 2023-06-06 | Novartis Ag | Antiviral pyrazolopyridinone compounds |
US20230077499A1 (en) * | 2019-12-20 | 2023-03-16 | Merck Sharp & Dohme Llc | Amido-substituted heterocyclic compounds and methods of use thereof for the treatment of herpes viruses |
CA3235718A1 (fr) | 2021-10-28 | 2023-05-04 | Insilico Medicine Ip Limited | Inhibiteurs de la proteine contenant un domaine prolyl hydroxylase (phd) et leurs utilisations |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0733729A (ja) | 1993-07-26 | 1995-02-03 | Kirin Brewery Co Ltd | N−シアノ−n′−置換−アリールカルボキシイミダミド化合物の製造法 |
JPH08301849A (ja) | 1995-05-01 | 1996-11-19 | Takeda Chem Ind Ltd | ヘテロ環化合物およびその製造法 |
ATE239477T1 (de) | 1995-08-02 | 2003-05-15 | Darwin Discovery Ltd | Chinolone und deren therapeutische verwendung |
CA2225555A1 (fr) | 1995-08-02 | 1997-02-13 | Chiroscience Limited | Quinolones et leur utilisation therapeutique |
US5945431A (en) | 1996-03-15 | 1999-08-31 | Biochem Therapeutics Incorporated | Cytomegalovirus inhibiting compounds |
GB9605437D0 (en) | 1996-03-15 | 1996-05-15 | Iaf Biochem Int | Cytomegalovirus inhibiting compounds |
AU4172197A (en) | 1996-09-10 | 1998-04-02 | Pharmacia & Upjohn Company | 8-hydroxy-7-substituted quinolines as anti-viral agents |
US5932618A (en) | 1996-11-04 | 1999-08-03 | Signal Pharmaceuticals, Inc. | Anti-viral agents and methods relating to the use thereof |
WO1999010347A1 (fr) | 1997-08-25 | 1999-03-04 | Neurogen Corporation | 4-oxo-naphtyridine-3-carboxamides substitues comme ligands de recepteur de gaba du cerveau |
NZ505362A (en) | 1997-12-22 | 2004-12-24 | Upjohn Co | 4-hydroxyquinoline-3-carboxamides and -hydrazides useful as antiviral agents |
US6248739B1 (en) | 1999-01-08 | 2001-06-19 | Pharmacia & Upjohn Company | Quinolinecarboxamides as antiviral agents |
JP2000256323A (ja) | 1999-01-08 | 2000-09-19 | Japan Tobacco Inc | 2−オキソキノリン化合物及びその医薬用途 |
US6248736B1 (en) | 1999-01-08 | 2001-06-19 | Pharmacia & Upjohn Company | 4-oxo-1,4-dihydro-3-quinolinecarboxamides as antiviral agents |
DK1159279T3 (da) | 1999-03-09 | 2003-02-17 | Upjohn Co | 4-Oxo-4,7-dihydro-thieno[2,3-b]pyridin-5-carboxamider som antivirale midler |
-
2001
- 2001-06-22 US US09/887,620 patent/US6730682B2/en not_active Expired - Fee Related
- 2001-06-25 EP EP01948225A patent/EP1363907A2/fr not_active Withdrawn
- 2001-06-25 JP JP2002509289A patent/JP2004502758A/ja active Pending
- 2001-06-25 AU AU2001269698A patent/AU2001269698A1/en not_active Abandoned
- 2001-06-25 AU AU2001269697A patent/AU2001269697A1/en not_active Abandoned
- 2001-06-25 EP EP01948224A patent/EP1299360A2/fr not_active Withdrawn
- 2001-06-25 WO PCT/US2001/016491 patent/WO2002004422A2/fr not_active Application Discontinuation
- 2001-06-25 JP JP2002509308A patent/JP2004502769A/ja active Pending
- 2001-06-25 WO PCT/US2001/016492 patent/WO2002004443A2/fr not_active Application Discontinuation
- 2001-07-05 AR ARP010103210A patent/AR030244A1/es not_active Application Discontinuation
- 2001-07-05 AR ARP010103209A patent/AR030243A1/es not_active Application Discontinuation
- 2001-07-06 PE PE2001000673A patent/PE20020143A1/es not_active Application Discontinuation
- 2001-07-09 PE PE2001000676A patent/PE20020256A1/es not_active Application Discontinuation
-
2004
- 2004-03-29 US US10/812,229 patent/US20040180910A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
WO2002004443A2 (fr) | 2002-01-17 |
PE20020143A1 (es) | 2002-02-15 |
US20040180910A1 (en) | 2004-09-16 |
EP1299360A2 (fr) | 2003-04-09 |
WO2002004422A2 (fr) | 2002-01-17 |
WO2002004443A3 (fr) | 2003-09-12 |
EP1363907A2 (fr) | 2003-11-26 |
AR030244A1 (es) | 2003-08-13 |
JP2004502758A (ja) | 2004-01-29 |
JP2004502769A (ja) | 2004-01-29 |
AU2001269697A1 (en) | 2002-01-21 |
AR030243A1 (es) | 2003-08-13 |
US20020019397A1 (en) | 2002-02-14 |
PE20020256A1 (es) | 2002-03-23 |
US6730682B2 (en) | 2004-05-04 |
WO2002004422A3 (fr) | 2002-06-20 |
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