ATE517896T1 - P38-kinase-inhibitoren - Google Patents

P38-kinase-inhibitoren

Info

Publication number
ATE517896T1
ATE517896T1 AT05702029T AT05702029T ATE517896T1 AT E517896 T1 ATE517896 T1 AT E517896T1 AT 05702029 T AT05702029 T AT 05702029T AT 05702029 T AT05702029 T AT 05702029T AT E517896 T1 ATE517896 T1 AT E517896T1
Authority
AT
Austria
Prior art keywords
kinase inhibitors
kinase
activity
mediated
inhibitors
Prior art date
Application number
AT05702029T
Other languages
German (de)
English (en)
Inventor
Michael David Barker
Julie Nicole Hamblin
Katherine Louise Jones
Vipulkumar Kantibhai Patel
Stephen Swanson
Ann Louise Walker
Original Assignee
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Llc filed Critical Glaxosmithkline Llc
Application granted granted Critical
Publication of ATE517896T1 publication Critical patent/ATE517896T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P11/00—Drugs for disorders of the respiratory system
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
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    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
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AT05702029T 2004-01-30 2005-01-27 P38-kinase-inhibitoren ATE517896T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0402137.4A GB0402137D0 (en) 2004-01-30 2004-01-30 Novel compounds
PCT/GB2005/000274 WO2005073232A1 (en) 2004-01-30 2005-01-27 P38 kinase inhibitors

Publications (1)

Publication Number Publication Date
ATE517896T1 true ATE517896T1 (de) 2011-08-15

Family

ID=31971797

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05702029T ATE517896T1 (de) 2004-01-30 2005-01-27 P38-kinase-inhibitoren

Country Status (6)

Country Link
US (1) US20070161673A1 (https=)
EP (1) EP1709046B1 (https=)
JP (1) JP2007519694A (https=)
AT (1) ATE517896T1 (https=)
GB (1) GB0402137D0 (https=)
WO (1) WO2005073232A1 (https=)

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GB0402137D0 (en) 2004-03-03
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EP1709046A1 (en) 2006-10-11
US20070161673A1 (en) 2007-07-12

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