ATE510837T1 - Caspase inhibitoren und deren verwendung - Google Patents

Caspase inhibitoren und deren verwendung

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Publication number
ATE510837T1
ATE510837T1 AT01970836T AT01970836T ATE510837T1 AT E510837 T1 ATE510837 T1 AT E510837T1 AT 01970836 T AT01970836 T AT 01970836T AT 01970836 T AT01970836 T AT 01970836T AT E510837 T1 ATE510837 T1 AT E510837T1
Authority
AT
Austria
Prior art keywords
group
optionally substituted
ring
hydrogen
caspase inhibitors
Prior art date
Application number
AT01970836T
Other languages
German (de)
English (en)
Inventor
Jean-Damien Charrier
Ronald Knegtel
Michael Mortimore
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Application granted granted Critical
Publication of ATE510837T1 publication Critical patent/ATE510837T1/de

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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AT01970836T 2000-09-13 2001-09-12 Caspase inhibitoren und deren verwendung ATE510837T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23257300P 2000-09-13 2000-09-13
PCT/US2001/028450 WO2002022611A2 (en) 2000-09-13 2001-09-12 Caspase inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
ATE510837T1 true ATE510837T1 (de) 2011-06-15

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Family Applications (1)

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AT01970836T ATE510837T1 (de) 2000-09-13 2001-09-12 Caspase inhibitoren und deren verwendung

Country Status (8)

Country Link
US (1) US6800619B2 (OSRAM)
EP (1) EP1317454B1 (OSRAM)
JP (2) JP2004509120A (OSRAM)
AT (1) ATE510837T1 (OSRAM)
AU (1) AU2001290795A1 (OSRAM)
CA (1) CA2418720A1 (OSRAM)
PE (1) PE20020500A1 (OSRAM)
WO (1) WO2002022611A2 (OSRAM)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020058636A1 (en) * 1994-09-21 2002-05-16 Geoffrey P. Symonds Ribozymes targeting the retroviral packaging sequence expression constructs and recombinant retroviruses containing such constructs
PE20011350A1 (es) 2000-05-19 2002-01-15 Vertex Pharma PROFARMACO DE UN INHIBIDOR DE ENZIMA CONVERTIDORA DE INTERLEUCINA-1ß (ICE)
EP1317454B1 (en) * 2000-09-13 2011-05-25 Vertex Pharmaceuticals Incorporated Caspase inhibitors and uses thereof
FR2815541B1 (fr) * 2000-10-24 2008-02-29 Lipha Utilisation d'inhibiteurs de l'apoptose des pericytes pour le traitement et/ou la prevention de la retinopathie diabetique
EP1381602A1 (en) * 2001-04-19 2004-01-21 Vertex Pharmaceuticals Incorporated Heterocyclyldicarbamides as caspase inhibitors
EP1392289A2 (en) * 2001-05-23 2004-03-03 Vertex Pharmaceuticals Incorporated Caspase inhibitors and uses thereof
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