ATE452641T1 - Orale pharmazeutische zusammensetzung enthaltend 15-hydroxytestosteron und seine derivate - Google Patents
Orale pharmazeutische zusammensetzung enthaltend 15-hydroxytestosteron und seine derivateInfo
- Publication number
- ATE452641T1 ATE452641T1 AT03794351T AT03794351T ATE452641T1 AT E452641 T1 ATE452641 T1 AT E452641T1 AT 03794351 T AT03794351 T AT 03794351T AT 03794351 T AT03794351 T AT 03794351T AT E452641 T1 ATE452641 T1 AT E452641T1
- Authority
- AT
- Austria
- Prior art keywords
- hydroxytestosterone
- hydroxytestosterones
- androsten
- dihydroxy
- derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP02078643 | 2002-09-05 | ||
PCT/NL2003/000621 WO2004022065A1 (en) | 2002-09-05 | 2003-09-05 | Pharmaceutical application of 15- or 16- substituted testosterone analogues |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE452641T1 true ATE452641T1 (de) | 2010-01-15 |
Family
ID=31970390
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT03794351T ATE452641T1 (de) | 2002-09-05 | 2003-09-05 | Orale pharmazeutische zusammensetzung enthaltend 15-hydroxytestosteron und seine derivate |
Country Status (9)
Country | Link |
---|---|
US (1) | US7943602B2 (de) |
EP (1) | EP1551415B1 (de) |
CN (2) | CN101785775B (de) |
AT (1) | ATE452641T1 (de) |
AU (1) | AU2003263663A1 (de) |
CA (1) | CA2497838C (de) |
DE (1) | DE60330695D1 (de) |
ES (1) | ES2338782T3 (de) |
WO (1) | WO2004022065A1 (de) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY142989A (en) | 2004-03-10 | 2011-02-14 | Bayer Schering Pharma Ag | Stabilised supersaturated solids of lipophilic drugs |
DE602005014227D1 (de) * | 2004-03-10 | 2009-06-10 | Bayer Schering Pharma Ag | Zusammensetzungen aus drospirenon in molekularer dispersion |
US7401307B2 (en) * | 2004-11-03 | 2008-07-15 | International Business Machines Corporation | Slack sensitivity to parameter variation based timing analysis |
US9375437B2 (en) * | 2010-06-18 | 2016-06-28 | Lipocine Inc. | Progesterone containing oral dosage forms and kits |
US8951996B2 (en) | 2011-07-28 | 2015-02-10 | Lipocine Inc. | 17-hydroxyprogesterone ester-containing oral compositions and related methods |
US9301920B2 (en) | 2012-06-18 | 2016-04-05 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
BR112014012444B1 (pt) | 2011-11-23 | 2021-12-14 | Therapeuticsmd, Inc | Composição farmacêutica compreendendo estradiol solubilizado, progesterona e um agente de solubilização, bem como usos desta para tratar um sintoma relacionado à menopausa em uma mulher |
US20130338122A1 (en) | 2012-06-18 | 2013-12-19 | Therapeuticsmd, Inc. | Transdermal hormone replacement therapies |
US20150196640A1 (en) | 2012-06-18 | 2015-07-16 | Therapeuticsmd, Inc. | Progesterone formulations having a desirable pk profile |
US10806740B2 (en) | 2012-06-18 | 2020-10-20 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
US10806697B2 (en) | 2012-12-21 | 2020-10-20 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US9352047B2 (en) * | 2012-11-14 | 2016-05-31 | Abon Pharmaceuticals, Llc | Oral transmucosal drug delivery system |
US11246875B2 (en) | 2012-12-21 | 2022-02-15 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US11266661B2 (en) | 2012-12-21 | 2022-03-08 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10471072B2 (en) | 2012-12-21 | 2019-11-12 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10537581B2 (en) | 2012-12-21 | 2020-01-21 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10568891B2 (en) | 2012-12-21 | 2020-02-25 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US9180091B2 (en) | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
JP2017516768A (ja) | 2014-05-22 | 2017-06-22 | セラピューティックスエムディー インコーポレーテッドTherapeuticsmd, Inc. | 天然の併用ホルモン補充療法剤及び療法 |
BR112017027688A2 (pt) | 2015-06-22 | 2018-09-04 | Lipocine Inc | Composições orais que contêm éster de 17- hidroxiprogesterona e métodos relacionados |
US10328087B2 (en) | 2015-07-23 | 2019-06-25 | Therapeuticsmd, Inc. | Formulations for solubilizing hormones |
US10286077B2 (en) | 2016-04-01 | 2019-05-14 | Therapeuticsmd, Inc. | Steroid hormone compositions in medium chain oils |
EP3435977A4 (de) | 2016-04-01 | 2019-10-16 | Therapeuticsmd, Inc. | Pharmazeutische steroidhormonzusammensetzung |
US11633405B2 (en) | 2020-02-07 | 2023-04-25 | Therapeuticsmd, Inc. | Steroid hormone pharmaceutical formulations |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2793216A (en) * | 1954-08-17 | 1957-05-21 | Upjohn Co | 15-oxy-androstenes and 15-oxy-19-norandrostenes |
GB774064A (en) * | 1954-08-17 | 1957-05-01 | Upjohn Co | Steroids |
FR2035786A1 (en) * | 1969-03-28 | 1970-12-24 | Squibb & Sons Inc | A-d-glucosides of steroids contng 16a-and 17-oh gps |
US6117446A (en) * | 1999-01-26 | 2000-09-12 | Place; Virgil A. | Drug dosage unit for buccal administration of steroidal active agents |
EP1187618A1 (de) * | 1999-06-04 | 2002-03-20 | The General Hospital Corporation | PHARMAZEUTISCHE FORMüLIERUNGEN ZUR BEHANDLUNG VON FRAUEN IN DER POSTMENOPAUSE UND PERIMENOPAUSE UND DEREN ANWENDUNG |
CA2670236C (en) | 1999-09-30 | 2012-06-05 | Hollis-Eden Pharmaceuticals, Inc. | Therapeutic treatment of androgen receptor driven conditions |
-
2003
- 2003-09-05 DE DE60330695T patent/DE60330695D1/de not_active Expired - Lifetime
- 2003-09-05 WO PCT/NL2003/000621 patent/WO2004022065A1/en not_active Application Discontinuation
- 2003-09-05 AU AU2003263663A patent/AU2003263663A1/en not_active Abandoned
- 2003-09-05 EP EP03794351A patent/EP1551415B1/de not_active Expired - Lifetime
- 2003-09-05 US US10/526,730 patent/US7943602B2/en not_active Expired - Fee Related
- 2003-09-05 ES ES03794351T patent/ES2338782T3/es not_active Expired - Lifetime
- 2003-09-05 CN CN200910221753.4A patent/CN101785775B/zh not_active Expired - Fee Related
- 2003-09-05 CA CA2497838A patent/CA2497838C/en not_active Expired - Fee Related
- 2003-09-05 CN CN038248905A patent/CN1694710B/zh not_active Expired - Fee Related
- 2003-09-05 AT AT03794351T patent/ATE452641T1/de not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CN1694710A (zh) | 2005-11-09 |
CA2497838C (en) | 2012-07-17 |
WO2004022065A1 (en) | 2004-03-18 |
US7943602B2 (en) | 2011-05-17 |
AU2003263663A1 (en) | 2004-03-29 |
CA2497838A1 (en) | 2004-03-18 |
EP1551415B1 (de) | 2009-12-23 |
CN1694710B (zh) | 2012-09-05 |
EP1551415A1 (de) | 2005-07-13 |
ES2338782T3 (es) | 2010-05-12 |
DE60330695D1 (de) | 2010-02-04 |
CN101785775B (zh) | 2015-03-25 |
US20060122158A1 (en) | 2006-06-08 |
CN101785775A (zh) | 2010-07-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |