ATE442145T1 - Pharmazeutische zusammensetzung mit einem benzodiazepin-derivat und einem hemmer des rsv- fusionsproteins - Google Patents
Pharmazeutische zusammensetzung mit einem benzodiazepin-derivat und einem hemmer des rsv- fusionsproteinsInfo
- Publication number
- ATE442145T1 ATE442145T1 AT05728747T AT05728747T ATE442145T1 AT E442145 T1 ATE442145 T1 AT E442145T1 AT 05728747 T AT05728747 T AT 05728747T AT 05728747 T AT05728747 T AT 05728747T AT E442145 T1 ATE442145 T1 AT E442145T1
- Authority
- AT
- Austria
- Prior art keywords
- pharmaceutical composition
- fusion protein
- composition containing
- benzodiazepine derivative
- protein inhibitor
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0406279.0A GB0406279D0 (en) | 2004-03-19 | 2004-03-19 | Therapeutic compounds |
PCT/GB2005/001029 WO2005089771A1 (en) | 2004-03-19 | 2005-03-18 | Pharmaceutical composition comprising a benzodiazepine derivative and a inhibitor of the rsv fusion protein |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE442145T1 true ATE442145T1 (de) | 2009-09-15 |
Family
ID=32118066
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT05728747T ATE442145T1 (de) | 2004-03-19 | 2005-03-18 | Pharmazeutische zusammensetzung mit einem benzodiazepin-derivat und einem hemmer des rsv- fusionsproteins |
Country Status (17)
Country | Link |
---|---|
US (1) | US20070185096A1 (de) |
EP (1) | EP1727551B1 (de) |
JP (1) | JP2007529491A (de) |
KR (1) | KR20070009630A (de) |
CN (1) | CN100496499C (de) |
AT (1) | ATE442145T1 (de) |
AU (1) | AU2005224159B2 (de) |
BR (1) | BRPI0507652A (de) |
CA (1) | CA2557931A1 (de) |
DE (1) | DE602005016532D1 (de) |
DK (1) | DK1727551T3 (de) |
ES (1) | ES2331479T3 (de) |
GB (1) | GB0406279D0 (de) |
PL (1) | PL1727551T3 (de) |
PT (1) | PT1727551E (de) |
RU (1) | RU2006136881A (de) |
WO (1) | WO2005089771A1 (de) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0406282D0 (en) * | 2004-03-19 | 2004-04-21 | Arrow Therapeutics Ltd | Therapeutic compounds |
MX2009002019A (es) | 2006-08-24 | 2009-03-09 | Novartis Ag | Derivados de 2-(pirazin-2-il)-tiazol y 2-(1h-pirazol-3-il)-tiazol asi como compuestos relacionados como inhibidores de la estearoil-coa-desaturasa (scd) para el tratamiento de trastornos metabolicos, cardiovasculares, y otros. |
EP2066664A1 (de) | 2006-09-22 | 2009-06-10 | Novartis AG | Organische heterozyklische verbindungen |
BRPI0720452A2 (pt) | 2006-12-20 | 2014-01-14 | Novartis Ag | Compostos orgânicos |
BRPI0912539A2 (pt) * | 2008-05-05 | 2015-10-13 | Amgen Inc | composto, composição farmacêutica , método para tratar uma doença, e, uso do composto. |
US9556236B1 (en) | 2012-11-29 | 2017-01-31 | University Of South Florida | Compositions and methods for treating respiratory syncytial virus infection |
AU2016297024B2 (en) | 2015-07-22 | 2021-03-04 | Enanta Pharmaceuticals, Inc. | Benzodiazepine derivatives as RSV inhibitors |
EP3402799B1 (de) | 2016-01-15 | 2022-05-04 | Enanta Pharmaceuticals, Inc. | Heterocyclische verbindungen als rsv-inhibitoren |
GB201613942D0 (en) | 2016-08-15 | 2016-09-28 | Univ Of Durham The | An antimicrobial compound |
WO2018129287A1 (en) | 2017-01-06 | 2018-07-12 | Enanta Pharmaceuticals, Inc. | Heteroaryldiazepine derivatives as rsv inhibitors |
EP3582784B1 (de) * | 2017-02-16 | 2022-06-08 | Enanta Pharmaceuticals, Inc. | Verfahren zur herstellung von benzodiazepinderivaten |
WO2018226801A1 (en) | 2017-06-07 | 2018-12-13 | Enanta Pharmaceuticals, Inc. | Aryldiazepine derivatives as rsv inhibitors |
US11091501B2 (en) | 2017-06-30 | 2021-08-17 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as RSV inhibitors |
WO2019006291A1 (en) | 2017-06-30 | 2019-01-03 | Enanta Pharmaceuticals, Inc. | HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS |
WO2019046364A1 (en) * | 2017-08-29 | 2019-03-07 | Emory University | INHIBITORS OF SYNCYTIAL RESPIRATORY VIRUS (RSV) REPLICATION AND USES THEREOF |
MX2020004084A (es) | 2017-09-29 | 2020-07-29 | Enanta Pharm Inc | Agentes farmaceuticos como inhibidores del rsv para utilizar en combinacion. |
CN111343990B (zh) | 2017-11-13 | 2023-08-04 | 英安塔制药有限公司 | 苯并二氮杂䓬-2-酮和苯并氮杂䓬-2-酮衍生物的拆分方法 |
WO2019094920A1 (en) | 2017-11-13 | 2019-05-16 | Enanta Pharmaceuticals, Inc. | Azepin-2-one derivatives as rsv inhibitors |
US10975094B2 (en) | 2018-04-11 | 2021-04-13 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as RSV inhibitors |
WO2020190935A1 (en) | 2019-03-18 | 2020-09-24 | Enanta Pharmaceuticals, Inc. | Benzodiazepine derivatives as rsv inhibitors |
WO2020210246A1 (en) | 2019-04-09 | 2020-10-15 | Enanta Pharmaceuticals, Inc, | Heterocyclic compounds as rsv inhibitors |
GB201911944D0 (en) | 2019-08-20 | 2019-10-02 | Reviral Ltd | Pharmaceutical compounds |
CA3153297A1 (en) | 2019-10-04 | 2021-04-08 | Adam SZYMANIAK | Antiviral heterocyclic compounds |
US11505558B1 (en) | 2019-10-04 | 2022-11-22 | Enanta Pharmaceuticals, Inc. | Antiviral heterocyclic compounds |
GB201915273D0 (en) * | 2019-10-22 | 2019-12-04 | Reviral Ltd | Pharmaceutical compounds |
UY39032A (es) | 2020-01-24 | 2021-07-30 | Enanta Pharm Inc | Compuestos heterocíclicos como agentes antivirales |
US11534439B2 (en) | 2020-07-07 | 2022-12-27 | Enanta Pharmaceuticals, Inc. | Dihydroquinoxaline and dihydropyridopyrazine derivatives as RSV inhibitors |
WO2022086840A1 (en) | 2020-10-19 | 2022-04-28 | Enanta Pharmaceuticals, Inc. | Heterocyclic compounds as anti-viral agents |
BR112023016970A2 (pt) | 2021-02-26 | 2023-10-10 | Enanta Pharm Inc | Compostos heterocíclicos antivirais |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4324794A (en) * | 1980-08-26 | 1982-04-13 | Research Triangle Institute | Inhibition of respiratory syncytial virus-induced cell fusion by amidino compounds |
US4820834A (en) * | 1984-06-26 | 1989-04-11 | Merck & Co., Inc. | Benzodiazepine analogs |
EP0491218A1 (de) * | 1990-12-17 | 1992-06-24 | F. Hoffmann-La Roche Ag | Benzodiazepinone |
US6489338B2 (en) * | 2000-06-13 | 2002-12-03 | Bristol-Myers Squibb Company | Imidazopyridine and imidazopyrimidine antiviral agents |
US6919331B2 (en) * | 2001-12-10 | 2005-07-19 | Bristol-Myers Squibb Company | Substituted 2-methyl-benzimidazole respiratory syncytial virus antiviral agents |
EP1461036A4 (de) * | 2001-12-10 | 2005-11-16 | Bristol Myers Squibb Co | Bis-hydrochlorid-monohydratsalz des rsv-fusionshemmers |
BR0314595A (pt) * | 2002-09-20 | 2005-08-09 | Arrow Therapeutics Ltd | Uso de um derivado de benzodiazepina ou um sal farmaceuticamente aceitável deste, inalador ou nebulisador, produto, usos de um produto e de um composto ou sal farmaceuticamente aceitável deste, derivado de benzodiazepina, composto, e, composição farmacêutica |
GB0406282D0 (en) * | 2004-03-19 | 2004-04-21 | Arrow Therapeutics Ltd | Therapeutic compounds |
-
2004
- 2004-03-19 GB GBGB0406279.0A patent/GB0406279D0/en not_active Ceased
-
2005
- 2005-03-18 BR BRPI0507652-8A patent/BRPI0507652A/pt not_active IP Right Cessation
- 2005-03-18 CN CNB2005800089207A patent/CN100496499C/zh not_active Expired - Fee Related
- 2005-03-18 AU AU2005224159A patent/AU2005224159B2/en not_active Ceased
- 2005-03-18 PT PT05728747T patent/PT1727551E/pt unknown
- 2005-03-18 PL PL05728747T patent/PL1727551T3/pl unknown
- 2005-03-18 EP EP05728747A patent/EP1727551B1/de not_active Not-in-force
- 2005-03-18 WO PCT/GB2005/001029 patent/WO2005089771A1/en active Application Filing
- 2005-03-18 DE DE602005016532T patent/DE602005016532D1/de not_active Expired - Fee Related
- 2005-03-18 ES ES05728747T patent/ES2331479T3/es active Active
- 2005-03-18 KR KR1020067021651A patent/KR20070009630A/ko not_active Application Discontinuation
- 2005-03-18 DK DK05728747T patent/DK1727551T3/da active
- 2005-03-18 US US10/593,382 patent/US20070185096A1/en not_active Abandoned
- 2005-03-18 JP JP2007503412A patent/JP2007529491A/ja not_active Withdrawn
- 2005-03-18 CA CA002557931A patent/CA2557931A1/en not_active Abandoned
- 2005-03-18 RU RU2006136881/15A patent/RU2006136881A/ru not_active Application Discontinuation
- 2005-03-18 AT AT05728747T patent/ATE442145T1/de not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
WO2005089771A1 (en) | 2005-09-29 |
ES2331479T3 (es) | 2010-01-05 |
DE602005016532D1 (de) | 2009-10-22 |
AU2005224159A1 (en) | 2005-09-29 |
PL1727551T3 (pl) | 2010-02-26 |
PT1727551E (pt) | 2009-10-08 |
GB0406279D0 (en) | 2004-04-21 |
AU2005224159B2 (en) | 2009-05-21 |
EP1727551B1 (de) | 2009-09-09 |
US20070185096A1 (en) | 2007-08-09 |
KR20070009630A (ko) | 2007-01-18 |
CA2557931A1 (en) | 2005-09-29 |
DK1727551T3 (da) | 2009-12-14 |
CN100496499C (zh) | 2009-06-10 |
BRPI0507652A (pt) | 2007-07-10 |
JP2007529491A (ja) | 2007-10-25 |
EP1727551A1 (de) | 2006-12-06 |
RU2006136881A (ru) | 2008-04-27 |
CN1933841A (zh) | 2007-03-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE442145T1 (de) | Pharmazeutische zusammensetzung mit einem benzodiazepin-derivat und einem hemmer des rsv- fusionsproteins | |
ATE437643T1 (de) | Pharmazeutische zusammensetzung mit einem benzodiazepin-derivat und einem hemmer des rsv- fusionsproteins | |
WO2006128184A3 (en) | Pyrimidine or triazine fused bicyclic metalloprotease inhibitors | |
AU2003264038A1 (en) | Combination pharmaceutical agents as inhibitors of hcv replication | |
WO2007139856A3 (en) | Heterobicyclic metalloprotease inhibitors | |
ECSP055701A (es) | Nuevos derivados de pirimidinamida y el uso de los mismos | |
PE20061373A1 (es) | Composicion farmaceutica que contiene 'n-(2-cloro-6-metilfenil)-2-[[6-[4-(2-hidroxietil)-1-piperazinil]-2-metil-4-pirimidinil]amino]-5-tiazolcarboxamida | |
CR8102A (es) | Derivados de pirazolo- quinazolina, procedimiento para preparacion y su uso como inhibidores de quinasa | |
DE60332433D1 (de) | Azolylaminoazine als proteinkinasehemmer | |
DE60332604D1 (de) | Azolylaminoazine als proteinkinasehemmer | |
MXPA05002871A (es) | Derivados de benzodiazaepina y composiciones farmaceuticas que los contienen. | |
MXPA02005844A (es) | Inhibidores de cinasas de proteina. | |
MY143466A (en) | Inhibitors of tyrosine kinases | |
BR0316350A (pt) | Diaminotriazóis úteis como inibidores de proteìna cinases | |
GEP20084367B (en) | Diazepinoindole derivatives as kinase inhibitors | |
UY28897A1 (es) | Ácido 2-((2-(2-metilaminopirimidin-4-il)-1h-indol-5-carbonil)amino)-3-(fenilpiridin-2-ilamino)propiónico sustancialmente puro como inhibidor de la cinasa ikb | |
IL179206A0 (en) | Pyrrolylpyrimidine derivatives and pharmaceutical compositions containing the same | |
WO2007011878A3 (en) | Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists | |
MXPA05007609A (es) | Antagonista de un receptor sensible al calcio. | |
MXPA05010521A (es) | Inhibidores de cinasa de amida de bifenilcarboxilica p38. | |
EA200801614A1 (ru) | Фармацевтическая композиция, содержащая монтелукаст | |
WO2004016741A3 (en) | Prenylation inhibitors containing dimethyl-cyclobutane and methods of their synthesis and use | |
AR056517A1 (es) | Composiciones y metodos farmaceuticos utilizando temozolomida y un inhibidor de la proteina quinasa | |
DE60134735D1 (de) | Neue neurokinin-antagonisten zum gebrauch als arzneimittel | |
EA200601592A1 (ru) | Фармацевтическая композиция, содержащая ингибитор pde4 или pde3/4 и антагонист гистаминового рецептора |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification |
Ref document number: 1727551 Country of ref document: EP |
|
REN | Ceased due to non-payment of the annual fee |