ATE305008T1 - Gonadotropin freisetzenden hormon rezeptor antagonisten und ihre verwandten verwendungen - Google Patents
Gonadotropin freisetzenden hormon rezeptor antagonisten und ihre verwandten verwendungenInfo
- Publication number
- ATE305008T1 ATE305008T1 AT00973591T AT00973591T ATE305008T1 AT E305008 T1 ATE305008 T1 AT E305008T1 AT 00973591 T AT00973591 T AT 00973591T AT 00973591 T AT00973591 T AT 00973591T AT E305008 T1 ATE305008 T1 AT E305008T1
- Authority
- AT
- Austria
- Prior art keywords
- receptor antagonists
- releasing hormone
- hormone receptor
- gonadotropin releasing
- related uses
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Dermatology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41876899A | 1999-10-15 | 1999-10-15 | |
| PCT/US2000/028677 WO2001029044A1 (en) | 1999-10-15 | 2000-10-16 | Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE305008T1 true ATE305008T1 (de) | 2005-10-15 |
Family
ID=23659500
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00973591T ATE305008T1 (de) | 1999-10-15 | 2000-10-16 | Gonadotropin freisetzenden hormon rezeptor antagonisten und ihre verwandten verwendungen |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP1220857B1 (enExample) |
| JP (1) | JP2003512379A (enExample) |
| KR (1) | KR20020045609A (enExample) |
| AT (1) | ATE305008T1 (enExample) |
| AU (1) | AU769855B2 (enExample) |
| CA (1) | CA2386942A1 (enExample) |
| DE (1) | DE60022769T2 (enExample) |
| ES (1) | ES2249302T3 (enExample) |
| HK (1) | HK1047437B (enExample) |
| MX (1) | MXPA02003614A (enExample) |
| WO (1) | WO2001029044A1 (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1255738T3 (da) | 2000-01-25 | 2012-06-25 | Neurocrine Biosciences Inc | Gonadotropin-frigivende hormonreceptor-antagonister og fremgangsmåder relateret dertil |
| WO2002102401A1 (en) | 2001-04-30 | 2002-12-27 | Zentaris Gmbh | Treatment of dementia and neurodegenerative diseases with intermediate doses of lhrh antagonists |
| MXPA04000985A (es) * | 2001-08-02 | 2005-02-17 | Neurocrine Biosciences Inc | Piridin-4-onas sustituidas y su uso como antagonistas del receptor de hormona de liberacion de gonadotropina. |
| US6750350B2 (en) | 2001-08-02 | 2004-06-15 | Neurocrine Biosciences, Inc. | Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
| US6740656B2 (en) | 2001-08-02 | 2004-05-25 | Neurocrine Biosciences, Inc. | Gonadotropin-releasing hormone receptor antagonists and methods relating thereto |
| JP2005500352A (ja) | 2001-08-02 | 2005-01-06 | ニューロクライン バイオサイエンシーズ， インコーポレイテッド | ゴナドトロピン放出ホルモンレセプター（ＧｎＲＨ）アンタゴニストとしての１，２，４−トリアジン−３，５−ジオン |
| AU2002324586B2 (en) | 2001-08-02 | 2008-04-24 | Neurocrine Biosciences, Inc. | 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists |
| AU2003202115A1 (en) | 2002-02-12 | 2003-09-04 | Pfizer Inc. | Non-peptide compounds affecting the action of gonadotropin-releasing hormone (gnrh) |
| CA2489252A1 (en) | 2002-06-13 | 2003-12-24 | Pfizer Inc. | Non-peptide gnrh agents, pharmaceutical compositions and methods for their use |
| ATE557007T1 (de) | 2003-07-07 | 2012-05-15 | Neurocrine Biosciences Inc | Arylpyrimidine geeignet zur behandlung von sexualhormonbedingten zuständen wie endometriose, prostatakrebs und dergleichen |
| WO2005007165A1 (en) | 2003-07-07 | 2005-01-27 | Neurocrine Biosciences, Inc. | Pyrimidine-2, 4-dione derivatives as gonadotropin-releasing hormone receptor antagonists |
| DE602004020638D1 (de) | 2003-07-07 | 2009-05-28 | Neurocrine Biosciences Inc | Pyrimidin-2,4-dion-derivate als gonadotropin freisetzende hormon-rezeptor-antagonisten |
| CL2008000986A1 (es) | 2007-04-06 | 2008-10-17 | Neurocrine Biosciences Inc | COMPUESTO DERIVADO DE HETEROCICLOS DE NITROGENO, AGONISTAS DEL RECEPTOR GnRH; COMPOSICION FARMACEUTICA QUE COMPRENDE A DICHO COMPUESTO; Y USO PARA TRATAR UNA AFECCION RELACIONADA CON LAS HORMONAS SEXUALES, ENDOMETRIOSIS, DISMENORREA, ENFERMEDAD DE OV |
| AR065948A1 (es) | 2007-04-06 | 2009-07-15 | Neurocrine Biosciences Inc | Antagonistas del receptor de la hormona liberadora de gonadotropina y procedimientos relacionados con los mismos |
| NZ586271A (en) | 2007-12-13 | 2012-08-31 | Vertex Pharma | Fused pyrimidinone derivatives as modulators of cystic fibrosis transmembrane conductance regulator |
| CN101987865B (zh) * | 2009-07-29 | 2014-07-30 | 中国人民解放军军事医学科学院毒物药物研究所 | 含有乙内酰脲结构的促黄体生成素释放激素拮抗剂 |
| TW201130854A (en) | 2009-12-22 | 2011-09-16 | Bayer Schering Pharma Ag | Pyridinone derivatives and pharmaceutical compositions thereof |
| WO2012175514A1 (en) | 2011-06-21 | 2012-12-27 | Bayer Intellectual Property Gmbh | Pyridinone derivatives and pharmaceutical compositions thereof |
| CA2865547C (en) * | 2012-02-28 | 2020-03-10 | Sk Chemicals Co., Ltd. | Gonadotropin releasing hormone receptor antagonists, method for the preparation thereof and pharmaceutical composition comprising the same |
| JPWO2014133112A1 (ja) * | 2013-03-01 | 2017-02-02 | 国立大学法人 東京大学 | オートタキシン阻害活性を有する８−置換イミダゾピリミジノン誘導体 |
| KR101973074B1 (ko) * | 2018-11-30 | 2019-04-26 | 주식회사 티움바이오 | 퓨로피리미딘 화합물의 염 및 결정형, 및 이를 포함하는 약학적 조성물 |
| PH12022551282A1 (en) | 2019-11-25 | 2023-11-29 | Amgen Inc | Heterocyclic compounds as delta-5 desaturase inhibitors and methods of use |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU1687199A (en) * | 1997-12-26 | 1999-07-19 | Takeda Chemical Industries Ltd. | Nitrogen-containing heterocyclic compounds, their production and use |
| US6081508A (en) * | 1998-02-25 | 2000-06-27 | Indus River Networks, Inc. | Remote computer communication |
| WO1999051232A1 (en) * | 1998-04-02 | 1999-10-14 | Merck & Co., Inc. | Antagonists of gonadotropin releasing hormone |
-
2000
- 2000-10-16 CA CA002386942A patent/CA2386942A1/en not_active Abandoned
- 2000-10-16 ES ES00973591T patent/ES2249302T3/es not_active Expired - Lifetime
- 2000-10-16 EP EP00973591A patent/EP1220857B1/en not_active Expired - Lifetime
- 2000-10-16 DE DE60022769T patent/DE60022769T2/de not_active Expired - Fee Related
- 2000-10-16 KR KR1020027004773A patent/KR20020045609A/ko not_active Withdrawn
- 2000-10-16 AU AU12089/01A patent/AU769855B2/en not_active Ceased
- 2000-10-16 WO PCT/US2000/028677 patent/WO2001029044A1/en not_active Ceased
- 2000-10-16 JP JP2001531842A patent/JP2003512379A/ja active Pending
- 2000-10-16 AT AT00973591T patent/ATE305008T1/de not_active IP Right Cessation
- 2000-10-16 MX MXPA02003614A patent/MXPA02003614A/es active IP Right Grant
- 2000-10-16 HK HK02109095.3A patent/HK1047437B/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| HK1047437B (en) | 2005-12-16 |
| KR20020045609A (ko) | 2002-06-19 |
| AU769855B2 (en) | 2004-02-05 |
| ES2249302T3 (es) | 2006-04-01 |
| EP1220857B1 (en) | 2005-09-21 |
| HK1047437A1 (en) | 2003-02-21 |
| EP1220857A1 (en) | 2002-07-10 |
| DE60022769D1 (de) | 2006-02-02 |
| MXPA02003614A (es) | 2002-10-23 |
| CA2386942A1 (en) | 2001-04-26 |
| DE60022769T2 (de) | 2006-07-06 |
| JP2003512379A (ja) | 2003-04-02 |
| WO2001029044A1 (en) | 2001-04-26 |
| AU1208901A (en) | 2001-04-30 |
Similar Documents
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| ATE305008T1 (de) | Gonadotropin freisetzenden hormon rezeptor antagonisten und ihre verwandten verwendungen | |
| ATE548357T1 (de) | Gonadotropin freisetzende hormon rezeptor antagonisten und ihre verwandten verfahren | |
| IL172833A0 (en) | Pyrimidine-2,4-dione derivatives and pharmaceutical compositions containing the same | |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |