ATE236924T1 - 8-substituierte b-nor-6-thiaequilin verbindungen als selektiven östrogenrezeptormodulatoren - Google Patents
8-substituierte b-nor-6-thiaequilin verbindungen als selektiven östrogenrezeptormodulatorenInfo
- Publication number
- ATE236924T1 ATE236924T1 AT97305932T AT97305932T ATE236924T1 AT E236924 T1 ATE236924 T1 AT E236924T1 AT 97305932 T AT97305932 T AT 97305932T AT 97305932 T AT97305932 T AT 97305932T AT E236924 T1 ATE236924 T1 AT E236924T1
- Authority
- AT
- Austria
- Prior art keywords
- receptor modulators
- estrogen receptor
- substituted
- compounds
- thiaequiline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
- C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
- C07J73/006—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by sulfur as hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2336696P | 1996-08-06 | 1996-08-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE236924T1 true ATE236924T1 (de) | 2003-04-15 |
Family
ID=21814667
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT97305932T ATE236924T1 (de) | 1996-08-06 | 1997-08-05 | 8-substituierte b-nor-6-thiaequilin verbindungen als selektiven östrogenrezeptormodulatoren |
Country Status (7)
Country | Link |
---|---|
US (1) | US6218425B1 (de) |
EP (1) | EP0823437B1 (de) |
JP (1) | JPH1067778A (de) |
AT (1) | ATE236924T1 (de) |
CA (1) | CA2212204A1 (de) |
DE (1) | DE69720620T2 (de) |
ES (1) | ES2196264T3 (de) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE524170T1 (de) * | 2000-02-14 | 2011-09-15 | Merck Sharp & Dohme | Östrogenrezeptor modulatoren |
US20050107350A1 (en) * | 2003-08-22 | 2005-05-19 | Pharmacia Corporation | Method for the treatment or prevention of bone disorders with a cyclooxygenase-2 inhibitor alone and in combination with a bone disorder treatment agent and compositions therewith |
CA2861066C (en) * | 2012-01-12 | 2024-01-02 | Yale University | Compounds and methods for the enhanced degradation of targeted proteins and other polypeptides by an e3 ubiquitin ligase |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US1444277A (en) * | 1922-02-20 | 1923-02-06 | Firm Kalle & Company Ag | Manufacture of dyestuffs |
US2480746A (en) * | 1947-04-22 | 1949-08-30 | Du Pont | 8, 9-benzthiophanthrone |
US3417100A (en) * | 1966-04-29 | 1968-12-17 | Lab For Organic Chemistry Univ | 8,(9)-dehydro-6-thiaestrone-3-methyl ether |
US3586710A (en) * | 1968-11-12 | 1971-06-22 | American Cyanamid Co | Estrogenic b-nor steroids |
US5679694A (en) * | 1992-07-20 | 1997-10-21 | The Wellcome Foundation Ltd. | Tetracyclic compounds, intermediates for their preparation and their use as antitumor agents |
US5834488A (en) * | 1997-09-19 | 1998-11-10 | Eli Lilly And Company | Dihydrobenzo B! indeno 2, 1-D! thiophene compounds, intermediates, processes, compositions and methods |
-
1997
- 1997-07-29 US US08/902,485 patent/US6218425B1/en not_active Expired - Fee Related
- 1997-08-01 CA CA002212204A patent/CA2212204A1/en not_active Abandoned
- 1997-08-05 EP EP97305932A patent/EP0823437B1/de not_active Expired - Lifetime
- 1997-08-05 ES ES97305932T patent/ES2196264T3/es not_active Expired - Lifetime
- 1997-08-05 DE DE69720620T patent/DE69720620T2/de not_active Expired - Fee Related
- 1997-08-05 AT AT97305932T patent/ATE236924T1/de not_active IP Right Cessation
- 1997-08-06 JP JP9211700A patent/JPH1067778A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
JPH1067778A (ja) | 1998-03-10 |
DE69720620D1 (de) | 2003-05-15 |
EP0823437A2 (de) | 1998-02-11 |
CA2212204A1 (en) | 1998-02-06 |
ES2196264T3 (es) | 2003-12-16 |
DE69720620T2 (de) | 2004-03-25 |
EP0823437A3 (de) | 1999-04-28 |
EP0823437B1 (de) | 2003-04-09 |
US6218425B1 (en) | 2001-04-17 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE69935335D1 (de) | Pyrazole als modulatoren des östrogenrezeptors | |
IL129968A0 (en) | use of cntf receptor activators for the treatment of obesity | |
AU5467699A (en) | Substituted isoxazole as estrogen receptor modulators | |
IL112638A0 (en) | 3 alfa-hydroxylated pregnane and androstane derivatives and pharmaceutical compositions containing the same | |
ATE248157T1 (de) | Verbindungen und verfahren zur modulation von estrogen rezeptoren | |
ATE265510T1 (de) | Umweltunschädliche vereisungsschutzmittel und enteisungsmittel | |
BR9802005A (pt) | Derivado de pirazola tricìclico | |
TR200003377T2 (tr) | Estrojenler ile bütünleşik 2-fenil-1-[4-(2-aminoetoksi)benzil]-indol | |
GR980300076T1 (en) | Estrogen receptor | |
ATE236924T1 (de) | 8-substituierte b-nor-6-thiaequilin verbindungen als selektiven östrogenrezeptormodulatoren | |
EP0874625A4 (de) | Indanderivate für antipsychotische mittel | |
EA200300474A1 (ru) | Модуляторы рецепторов эстрогена | |
DE69902684D1 (de) | Estrogenische estra-1,3,5(10)-trien verbindungen mit verschiedenen wirkungen auf estrogenrezeptor alpha und beta mit einer unverzweigten kohlenwasserstoffkette von 5-9 kohlenstoffatomen in position 11 | |
ECSP045113A (es) | Benzopiranos sustituidos como agonistas selectivos del receptor estrogenico beta | |
PL316899A1 (en) | Thickener system for building material mixes | |
MX9702252A (es) | Nuevos androstanos para inducir efectos hipotalamicos. | |
NO994903L (no) | Behandling eller profylakse av prostatakreft og benign prostatahyperplasi med selektive östrogenreseptormodulatorer | |
Barrero et al. | Synthesis of monoterpenic analogues of puupehenone and puupehedione | |
TWI265923B (en) | Process for the preparation of 3-acylated indoles | |
PT943772E (pt) | Estrutura de montagem de portas deslizantes | |
EP1196428A4 (de) | Durch 11-beta-aryl-17,17-spirothiolan substituierte steroide | |
ATE339415T1 (de) | Benzocarbazol und indenoindole derivate als östrogene agentien | |
AU1959697A (en) | Benzothiophenes, and formulations and methods, using same | |
GB469198A (en) | Improvements in the distribution of road dressing material | |
SE8900443D0 (sv) | Anordning vid foerdelningsbrunnar |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |