ATE22087T1 - N-acyl peptiden, verfahren zu deren herstellung und deren pharmazeutische zusammensetzungen. - Google Patents

N-acyl peptiden, verfahren zu deren herstellung und deren pharmazeutische zusammensetzungen.

Info

Publication number
ATE22087T1
ATE22087T1 AT82306928T AT82306928T ATE22087T1 AT E22087 T1 ATE22087 T1 AT E22087T1 AT 82306928 T AT82306928 T AT 82306928T AT 82306928 T AT82306928 T AT 82306928T AT E22087 T1 ATE22087 T1 AT E22087T1
Authority
AT
Austria
Prior art keywords
alkyl
carboxy
hydrogen
amino
processes
Prior art date
Application number
AT82306928T
Other languages
English (en)
Inventor
Kazuyoshi Umehara
Keizo Yoshida
Hirokazu Tanaka
Itsuo Uchida
Masanobu Kohsaka
Hiroshi Imanaka
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Application granted granted Critical
Publication of ATE22087T1 publication Critical patent/ATE22087T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06052—Val-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT82306928T 1982-01-05 1982-12-23 N-acyl peptiden, verfahren zu deren herstellung und deren pharmazeutische zusammensetzungen. ATE22087T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB8200212 1982-01-05
GB8215910 1982-06-01
EP82306928A EP0085255B1 (de) 1982-01-05 1982-12-23 N-Acyl Peptiden, Verfahren zu deren Herstellung und deren pharmazeutische Zusammensetzungen

Publications (1)

Publication Number Publication Date
ATE22087T1 true ATE22087T1 (de) 1986-09-15

Family

ID=26281659

Family Applications (1)

Application Number Title Priority Date Filing Date
AT82306928T ATE22087T1 (de) 1982-01-05 1982-12-23 N-acyl peptiden, verfahren zu deren herstellung und deren pharmazeutische zusammensetzungen.

Country Status (11)

Country Link
US (1) US4643990A (de)
EP (1) EP0085255B1 (de)
KR (1) KR840003235A (de)
AT (1) ATE22087T1 (de)
AU (1) AU9173582A (de)
DE (1) DE3273256D1 (de)
DK (1) DK579682A (de)
ES (1) ES518771A0 (de)
FI (1) FI824453L (de)
GR (1) GR77060B (de)
NO (1) NO830011L (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU560285B2 (en) * 1982-07-19 1987-04-02 Imperial Chemical Industries Plc Heterocyclyl carbonyl sulphonamides
EP0136879A3 (de) * 1983-09-30 1987-01-07 Yamanouchi Pharmaceutical Co., Ltd. Fettsäure-Derivate und Verfahren zu deren Herstellung
DE3423582A1 (de) * 1984-06-27 1986-01-09 Bayer Ag, 5090 Leverkusen Substituierte 5-acylamino-1-phenylpyrazole
DE3700173A1 (de) * 1987-01-05 1988-07-14 Hoechst Ag Verfahren zur herstellung von lipophilen aminosaeurederivaten sowie lipophile aminosaeurederivate
FR2611205B1 (fr) * 1987-02-20 1990-03-02 Serbio Dipeptides, procede de preparation et utilisation dans le dosage de proteases
US5464825A (en) * 1991-03-14 1995-11-07 Cornell Research Foundation, Inc. Raising glutathione equivalent levels using N-acyl glutathione monoesters
EP0697882A4 (de) * 1993-05-03 1999-04-07 Cornell Res Foundation Inc Verwendung von glutathion-diestern
US5627210A (en) * 1995-02-06 1997-05-06 Chiron Corporation Branched combinatorial libraries
WO2001035982A1 (fr) * 1999-11-12 2001-05-25 Fujimoto Brothers Co., Ltd. Compositions medicinales anti-inflammatoires
WO2005053727A2 (en) * 2003-11-29 2005-06-16 Sangstat Medical Corporation Pharmaceutical compositions for bioactive peptide agents

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL279057A (de) * 1900-01-01
NL109134C (de) * 1900-01-01
FR2907E (fr) * 1903-03-09 1904-07-12 Brunet Loiseau Freres Soc Interrupteur-vibreur pour bobine d'induction, en vue de l'allumage des moteurs
FR4629E (fr) * 1904-04-21 1905-09-02 Jean Victorin Poplawski Générateur de vapeur à mèche
FR7648E (fr) * 1906-02-26 1907-09-17 Georges Clesse Dispositif de changement de vitesse et de renversement de marche pour voitures automobiles
NL299197A (de) * 1957-07-11
JPS4211925Y1 (de) * 1966-02-09 1967-07-05
DE1593858A1 (de) * 1967-03-02 1970-10-29 Hoechst Ag Verfahren zur Herstellung tyrosinhaltiger Peptide und deren Derivaten
JPS468685Y1 (de) * 1967-08-02 1971-03-27
JPS46164Y1 (de) * 1967-09-05 1971-01-07
US3893992A (en) * 1970-11-19 1975-07-08 Rohm & Haas N-acylated peptides of amino aromatic sulfonic acids and their derivatives
FR2340983A1 (fr) * 1976-02-10 1977-09-09 Ugine Kuhlmann Activateurs pour percomposes
LU78804A1 (de) * 1977-12-30 1979-07-20 Byk Gulden Lomberg Chem Fab N-substituierte w-aminoalkanoyl-w-aminoalkansaeuren,ihre verwendung und verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
US4205069A (en) * 1978-09-29 1980-05-27 American Home Products Corporation Dipeptide narcotic antagonists
EP0011283B1 (de) * 1978-11-14 1982-07-28 Fujisawa Pharmaceutical Co., Ltd. Lactyl-tetrapeptid, Verfahren zu seiner Herstellung und dieses enthaltende pharmazeutische Zusammensetzungen
US4311640A (en) * 1978-11-14 1982-01-19 Fujisawa Pharmaceutical Co., Ltd. Peptide, process for preparation thereof and use thereof
FR2460288A1 (fr) * 1979-06-29 1981-01-23 Rhone Poulenc Ind Nouveaux dipeptides, leur preparation et les medicaments qui les contiennent
US4436726A (en) * 1980-12-15 1984-03-13 Fujisawa Pharmaceutical Co., Ltd. N-Acylpeptide compound, processes for the preparation thereof and the pharmaceutical compositions

Also Published As

Publication number Publication date
EP0085255A2 (de) 1983-08-10
ES8500892A1 (es) 1984-03-01
AU9173582A (en) 1983-07-14
US4643990A (en) 1987-02-17
ES518771A0 (es) 1984-03-01
DK579682A (da) 1983-07-06
FI824453L (fi) 1983-07-06
FI824453A0 (fi) 1982-12-27
NO830011L (no) 1983-07-06
EP0085255A3 (en) 1984-08-01
EP0085255B1 (de) 1986-09-10
DE3273256D1 (en) 1986-10-16
GR77060B (de) 1984-09-05
KR840003235A (ko) 1984-08-20

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