ATE214705T1 - Nichtalkalische reinigung von aminophosphonsäuren - Google Patents

Nichtalkalische reinigung von aminophosphonsäuren

Info

Publication number
ATE214705T1
ATE214705T1 AT94929152T AT94929152T ATE214705T1 AT E214705 T1 ATE214705 T1 AT E214705T1 AT 94929152 T AT94929152 T AT 94929152T AT 94929152 T AT94929152 T AT 94929152T AT E214705 T1 ATE214705 T1 AT E214705T1
Authority
AT
Austria
Prior art keywords
aminophosphonic acids
alkaline purification
purification
aminophosphonic
acids
Prior art date
Application number
AT94929152T
Other languages
English (en)
Inventor
Benjamin A Belinka Jr
Daniel J Coughlin
Original Assignee
Cytogen Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cytogen Corp filed Critical Cytogen Corp
Application granted granted Critical
Publication of ATE214705T1 publication Critical patent/ATE214705T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6524Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having four or more nitrogen atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/025Purification; Separation; Stabilisation; Desodorisation of organo-phosphorus compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3808Acyclic saturated acids which can have further substituents on alkyl
    • C07F9/3817Acids containing the structure (RX)2P(=X)-alk-N...P (X = O, S, Se)

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Detergent Compositions (AREA)
AT94929152T 1993-11-04 1994-09-15 Nichtalkalische reinigung von aminophosphonsäuren ATE214705T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/145,591 US5495042A (en) 1993-11-04 1993-11-04 Non-alkaline purification of aminophosphonic acids
PCT/US1994/010106 WO1995012586A1 (en) 1993-11-04 1994-09-15 Non-alkaline purification of aminophosphonic acids

Publications (1)

Publication Number Publication Date
ATE214705T1 true ATE214705T1 (de) 2002-04-15

Family

ID=22513770

Family Applications (1)

Application Number Title Priority Date Filing Date
AT94929152T ATE214705T1 (de) 1993-11-04 1994-09-15 Nichtalkalische reinigung von aminophosphonsäuren

Country Status (10)

Country Link
US (1) US5495042A (de)
EP (1) EP0724576B1 (de)
JP (1) JP2894839B2 (de)
AT (1) ATE214705T1 (de)
AU (1) AU7831794A (de)
BR (1) BR9407990A (de)
CA (1) CA2175221C (de)
DE (1) DE69430206T2 (de)
PH (1) PH31639A (de)
WO (1) WO1995012586A1 (de)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6011021A (en) * 1996-06-17 2000-01-04 Guilford Pharmaceuticals Inc. Methods of cancer treatment using naaladase inhibitors
US5795877A (en) * 1996-12-31 1998-08-18 Guilford Pharmaceuticals Inc. Inhibitors of NAALADase enzyme activity
US6025345A (en) * 1996-06-17 2000-02-15 Guilford Pharmaceuticals Inc. Inhibitors of NAALADase enzyme activity
US6054444A (en) 1997-04-24 2000-04-25 Guilford Pharmaceuticals Inc. Phosphonic acid derivatives
US6071965A (en) * 1996-06-17 2000-06-06 Guilford Pharmaceuticals Inc. Phosphinic alkanoic acid derivatives
HUP9903421A3 (en) 1996-06-17 2001-08-28 Guilford Pharmaceuticals Inc B Use of phosphonic and phosphinic acid derivatives for producing pharmaceutical compositions having naaladase inhibitor activity
US6384022B1 (en) 1996-06-17 2002-05-07 Guilford Pharmaceuticals Inc. Prodrugs of NAALAdase inhibitors
US6017903A (en) 1996-09-27 2000-01-25 Guilford Pharmaceuticals Inc. Pharmaceutical compositions and methods of treating a glutamate abnormality and effecting a neuronal activity in an animal using NAALADase inhibitors
US5863536A (en) * 1996-12-31 1999-01-26 Guilford Pharmaceuticals Inc. Phosphoramidate derivatives
US6025344A (en) * 1996-06-17 2000-02-15 Guilford Pharmaceuticals Inc. Certain dioic acid derivatives useful as NAALADase inhibitors
US6046180A (en) * 1996-06-17 2000-04-04 Guilford Pharmaceuticals Inc. NAALADase inhibitors
US5824662A (en) * 1996-09-27 1998-10-20 Guilford Pharmaceuticals Inc. Treatment of global and focal ischemia using naaladase inhibitors
US5817708A (en) * 1996-07-19 1998-10-06 The B. F. Goodrich Company Low volatile organic solvent based adhesive
US5962521A (en) 1997-04-04 1999-10-05 Guilford Pharmaceuticals Inc. Hydroxamic acid derivatives
KR20000036227A (ko) 1996-09-27 2000-06-26 토마스 씨. 서 날라다아제조성물, 글루탐산염 이상 치료법 및 동물내의 뉴우런활성법
US5981209A (en) * 1997-12-04 1999-11-09 Guilford Pharmaceuticals Inc. Use of NAALADase activity to identify prostate cancer and benign prostatic hyperplasia
US6028216A (en) * 1997-12-31 2000-02-22 Guilford Pharmaceuticals Inc. Asymmetric syntheses and intermediates for preparing enantiomer-enriched hydroxyphosphinyl derivatives
US6265609B1 (en) 1998-07-06 2001-07-24 Guilford Pharmaceuticals Inc. Thio-substituted pentanedioic acid derivatives
US6395718B1 (en) 1998-07-06 2002-05-28 Guilford Pharmaceuticals Inc. Pharmaceutical compositions and methods of inhibiting angiogenesis using naaladase inhibitors
CA2337797C (en) 1998-07-06 2009-04-14 Guilford Pharmaceuticals Inc. Naaladase inhibitors useful as pharmaceutical compounds and compositions
US6313159B1 (en) 1999-08-20 2001-11-06 Guilford Pharmaceuticals Inc. Metabotropic glutamate receptor ligand derivatives as naaladase inhibitors
JP5581832B2 (ja) * 2010-06-11 2014-09-03 三菱瓦斯化学株式会社 高純度アミノメチレンホスホン酸の製造方法
CN106661062A (zh) * 2014-06-02 2017-05-10 奇默和施瓦茨莫斯多夫有限及两合公司 用于制备结晶dtpmp的方法
DE102014210378B4 (de) 2014-06-02 2018-10-04 Zschimmer & Schwarz Mohsdorf GmbH &Co.KG. Verfahren zur Herstellung hochreiner Aminoalkylenphosphonsäuren

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1230121A (de) * 1967-01-27 1971-04-28
BE764270A (fr) * 1970-03-20 1971-08-02 Benckiser Gmbh Joh A Acide niril-tris-(methylenephosphonique) et son procede de preparation
DE2132511C3 (de) * 1971-06-30 1974-06-27 Joh. A. Benckiser Gmbh, 6700 Ludwigshafen Verfahren zur Herstellung von Aminomethylenphosphonsäuren
US3959361A (en) * 1970-03-20 1976-05-25 Joh. A. Benckiser Gmbh Process of producing amino methylene phosphonic acids
DE2017974A1 (de) * 1970-04-15 1971-11-04 Joh. A. Benckiser Gmbh Chemische Fabrik, 6700 Ludwigshafen Verfahren zur Herstellung von Aminoalkylenphosphonsäuren
DE2021148A1 (de) * 1970-04-30 1971-11-11 Benckiser Gmbh Joh A Verfahren und Anlage zur kontinuierlichen Herstellung von Aminoalkylenphosphonsaeuren
US4012440A (en) * 1970-11-18 1977-03-15 Petrolite Corporation Methylene phosphonates of oxyalkylated polyalkylene polyamines and uses therefor
US4035412A (en) * 1971-05-28 1977-07-12 Petrolite Corporation Methylene phosphonates of poly-diepoxidized polyalkylene polyamines
GB1436843A (en) * 1972-07-21 1976-05-26 Ici Ltd Preparation of n-phosphonomethyl-glycine
DE2741504C3 (de) * 1977-09-15 1981-11-19 Joh. A. Benckiser Gmbh, 6700 Ludwigshafen Verfahren zur Herstellung von Aminoalkylenphosphonsäuren
HU177486B (en) * 1978-04-11 1981-10-28 Nitrokemia Ipartelepek Process for preparing phosphonic acid derivatives
FR2473488A1 (fr) * 1980-01-14 1981-07-17 Oxysynthese Procede cyclique de production de peroxyde d'hydrogene
JPS5775990A (en) * 1980-10-27 1982-05-12 Mitsubishi Gas Chem Co Inc Preparation of n,n,n',n'-tetra(phosphonomethyl) diaminoalkane
EP0225409A1 (de) * 1985-12-02 1987-06-16 The Dow Chemical Company Organoaminophosphonische Säurekomplexe für die Behandlung von Kalktumoren
US4937333A (en) * 1989-08-04 1990-06-26 The Dow Chemical Company Method for purifying aminomethylenephosphonic acids for pharmaceutical use
US5159108A (en) * 1990-09-18 1992-10-27 Merck & Co., Inc. Process for preparing an antihypercalcemic agent
TW263511B (de) * 1990-10-10 1995-11-21 Hoechst Ag

Also Published As

Publication number Publication date
JP2894839B2 (ja) 1999-05-24
PH31639A (en) 1999-01-12
EP0724576A1 (de) 1996-08-07
US5495042A (en) 1996-02-27
CA2175221C (en) 2000-01-18
DE69430206T2 (de) 2002-10-10
JPH09504545A (ja) 1997-05-06
WO1995012586A1 (en) 1995-05-11
BR9407990A (pt) 1996-12-03
CA2175221A1 (en) 1995-05-11
DE69430206D1 (de) 2002-04-25
EP0724576A4 (de) 1997-02-12
AU7831794A (en) 1995-05-23
EP0724576B1 (de) 2002-03-20

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