ATE203897T1 - Konservierungsmittelhaltige ophtalmisch anzuwendende arzneizusammensetzungen enthaltend quaternäre polymerammoniumverbindungen - Google Patents

Konservierungsmittelhaltige ophtalmisch anzuwendende arzneizusammensetzungen enthaltend quaternäre polymerammoniumverbindungen

Info

Publication number
ATE203897T1
ATE203897T1 AT95939996T AT95939996T ATE203897T1 AT E203897 T1 ATE203897 T1 AT E203897T1 AT 95939996 T AT95939996 T AT 95939996T AT 95939996 T AT95939996 T AT 95939996T AT E203897 T1 ATE203897 T1 AT E203897T1
Authority
AT
Austria
Prior art keywords
ammonium compounds
preservatively
medicinal compositions
compositions containing
quaternary polymer
Prior art date
Application number
AT95939996T
Other languages
English (en)
Inventor
Suketu Dipakbhai Desai
Diane S Nelms
Original Assignee
Alcon Lab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alcon Lab Inc filed Critical Alcon Lab Inc
Application granted granted Critical
Publication of ATE203897T1 publication Critical patent/ATE203897T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT95939996T 1994-11-16 1995-11-16 Konservierungsmittelhaltige ophtalmisch anzuwendende arzneizusammensetzungen enthaltend quaternäre polymerammoniumverbindungen ATE203897T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/340,763 US5603929A (en) 1994-11-16 1994-11-16 Preserved ophthalmic drug compositions containing polymeric quaternary ammonium compounds
PCT/US1995/014910 WO1996014829A1 (en) 1994-11-16 1995-11-16 Preserved ophthalmic drug compositions containing polymeric quaternary ammonium compounds

Publications (1)

Publication Number Publication Date
ATE203897T1 true ATE203897T1 (de) 2001-08-15

Family

ID=23334841

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95939996T ATE203897T1 (de) 1994-11-16 1995-11-16 Konservierungsmittelhaltige ophtalmisch anzuwendende arzneizusammensetzungen enthaltend quaternäre polymerammoniumverbindungen

Country Status (12)

Country Link
US (2) US5603929A (de)
EP (1) EP0739197B1 (de)
JP (1) JP2954356B2 (de)
AT (1) ATE203897T1 (de)
AU (1) AU686917B2 (de)
CA (1) CA2180554C (de)
DE (1) DE69522094T2 (de)
DK (1) DK0739197T3 (de)
ES (1) ES2160722T3 (de)
GR (1) GR3036622T3 (de)
PT (1) PT739197E (de)
WO (1) WO1996014829A1 (de)

Families Citing this family (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5505953A (en) * 1992-05-06 1996-04-09 Alcon Laboratories, Inc. Use of borate-polyol complexes in ophthalmic compositions
US5683993A (en) * 1995-06-22 1997-11-04 Ciba Vision Corporation Compositions and methods for stabilizing polymers
JP2000505486A (ja) * 1996-02-14 2000-05-09 アルコン ラボラトリーズ,インコーポレイテッド ポリマー第4級アンモニウム化合物と、眼科用抗微生物剤としてのその使用
EP0877600B1 (de) * 1996-08-09 2003-10-22 Alcon Manufacturing Ltd. Konservierungssysteme fur cyclodextrine enthaltende arzneimittel
ATE326983T1 (de) 1996-12-13 2006-06-15 Alcon Lab Inc Aminoalkohole enthaltende ophthalmische zusammensetzungen
ATE391492T1 (de) * 1997-07-29 2008-04-15 Alcon Lab Inc Ophthalmische zusammensetzungen enthaltend galaktomannanpolymere und borat
JP4064625B2 (ja) 1997-11-26 2008-03-19 アドバンスト メディカル オプティクス, インコーポレーテッド コンタクトレンズ洗浄組成物
US6063745A (en) * 1997-11-26 2000-05-16 Allergan Mutli-purpose contact lens care compositions
JPH11249087A (ja) * 1997-12-18 1999-09-17 Tome:Kk コンタクトレンズ用液剤
JP2006111636A (ja) * 1997-12-26 2006-04-27 Astellas Pharma Inc 徐放性医薬組成物
US7678836B2 (en) * 1999-11-04 2010-03-16 Fxs Ventures, Llc Method for rendering a contact lens wettable
CA2395866C (en) 2000-01-25 2009-10-13 Alcon, Inc. Ophthalmic anti-allergy compositions suitable for use with contact lenses
AR035509A1 (es) * 2000-12-21 2004-06-02 Alcon Inc Solucion de lagrimas artificiales mejorada que contiene una combinacion de tres emolientes y el uso de dicha solucion para la fabricacion de un medicamento
US7923469B2 (en) 2001-04-30 2011-04-12 Allergen, Inc. Compositions including vitamin-based surfactants and methods for using same
JP4286480B2 (ja) * 2001-09-17 2009-07-01 株式会社メニコン 殺菌液
EP1586316B1 (de) 2003-01-21 2008-04-30 Senju Pharmaceutical Co., Ltd. Wässrige flüssige zubereitung mit 2-amino-3-(4-bromobenzoyl)phenylessigsäure
CA2505836C (en) * 2004-05-06 2013-08-27 Alcon Inc. Topical brimonidine tartrate formulations that lack chlorine dioxide
US20060073184A1 (en) * 2004-09-29 2006-04-06 Bausch & Lomb Inc. Viscoelastic composition, methods of use and packaging device with anti-oxidant
CN1993118B (zh) 2004-11-05 2010-06-16 千寿制药株式会社 促进眼内渗透性的水性滴眼剂
JP5108234B2 (ja) * 2005-02-07 2012-12-26 日本特殊陶業株式会社 マイクロヒータ及びセンサ
US7947010B2 (en) 2005-07-08 2011-05-24 Depuy Products, Inc. Composition and system for wound decontamination
US20100130580A1 (en) * 2006-01-25 2010-05-27 Aciex Therapeutics, Inc. Formulations and Methods for Treating Dry Eye
CA2621616A1 (en) * 2007-02-19 2008-08-19 Alcon Research, Ltd. Topical gatifloxacin formulations
US7705112B2 (en) 2007-04-17 2010-04-27 Abbott Medical Optics Inc. Polyquaternium-1 synthesis methods
MX2009012645A (es) * 2007-05-24 2010-03-08 Aciex Therapeutics Inc Formulaciones y metodos para tratar el ojo seco.
AU2008310956B2 (en) 2007-10-08 2014-08-07 Aurinia Pharmaceuticals Inc. Ophthalmic compositions comprising calcineurin inhibitors or mTOR inhibitors
BRPI0908502A2 (pt) * 2008-02-21 2017-05-23 Ista Pharmaceuticals aines oftálmicos como adjuvantes
US9192571B2 (en) 2008-03-03 2015-11-24 Allergan, Inc. Ketorolac tromethamine compositions for treating or preventing ocular pain
RU2431469C1 (ru) * 2008-03-03 2011-10-20 Аллерган, Инк. Композиции кеторолака трометамина для лечения или профилактики глазной боли
BRPI0909738A2 (pt) 2008-03-17 2015-10-06 Alcon Res Ltd composições farmacêuticas aquosas contendo complexos de boratopoliol
TWI544927B (zh) 2008-03-17 2016-08-11 愛爾康研究有限公司 具有低濃度的表面活性劑以促進治療劑之生物可利用性的藥學組成物
TWI454289B (zh) * 2008-04-03 2014-10-01 Alcon Res Ltd 使用順式二醇的聚合物於抑制陽離子殺生物劑被吸收進入水凝膠生物材質中之用途
TW201038295A (en) * 2009-04-17 2010-11-01 Alcon Res Ltd Aqueous ophthalmic compositions containing anionic therapeutic agents
MX338355B (es) 2009-06-09 2016-04-13 Aurinia Pharmaceuticals Inc Sistemas de suministro de farmaco topico para uso oftalmico.
TWI489997B (zh) 2009-06-19 2015-07-01 Alcon Res Ltd 含有硼酸-多元醇錯合物之水性藥學組成物
WO2012099142A1 (ja) 2011-01-18 2012-07-26 千寿製薬株式会社 保存効力を有するブロムフェナク水性液剤組成物
JP6128572B2 (ja) * 2012-11-19 2017-05-17 ボシュ・アンド・ロム・インコーポレイテッドBausch & Lomb Incorporated 2−アミノ−3−(4−ブロモベンゾイル)フェニル酢酸を含有する水性液体組成物
US20160143869A1 (en) 2013-06-19 2016-05-26 Sentiss Research Center Stable bromfenac solution
BR112016003692B1 (pt) 2013-08-20 2022-02-08 3M Innovative Properties Company Complexo poliéter boro-silano
WO2015087267A2 (en) 2013-12-12 2015-06-18 Sentiss Pharma Private Limited Stable bromfenac ophthalmic solution
US10632202B2 (en) 2016-03-04 2020-04-28 Johnson & Johnson Consumer Inc. Preservative containing compositions
US20190224275A1 (en) 2017-05-12 2019-07-25 Aurinia Pharmaceuticals Inc. Protocol for treatment of lupus nephritis
US20230159202A1 (en) * 2021-11-23 2023-05-25 Bausch + Lomb Ireland Limited Method for making a preservative-free packaged ophthalmic device product

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3931319A (en) * 1974-10-29 1976-01-06 Millmaster Onyx Corporation Capped polymers
US4027020A (en) * 1974-10-29 1977-05-31 Millmaster Onyx Corporation Randomly terminated capped polymers
US4136173A (en) * 1977-01-31 1979-01-23 American Home Products Corp. Mixed xanthan gum and locust beam gum therapeutic compositions
US4136178A (en) * 1977-01-31 1979-01-23 American Home Products Corp. Locust bean gum therapeutic compositions
US4136177A (en) * 1977-01-31 1979-01-23 American Home Products Corp. Xanthan gum therapeutic compositions
FR2508440B1 (fr) * 1981-06-25 1985-11-08 Saint Gobain Isover Procede de preparation d'alcools orthohydroxybenzyliques
US4407791A (en) * 1981-09-28 1983-10-04 Alcon Laboratories, Inc. Ophthalmic solutions
US4525346A (en) * 1981-09-28 1985-06-25 Alcon Laboratories, Inc. Aqueous antimicrobial ophthalmic solutions
US4836986A (en) * 1984-09-28 1989-06-06 Bausch & Lomb Incorporated Disinfecting and preserving systems and methods of use
FR2588189B1 (fr) * 1985-10-03 1988-12-02 Merck Sharp & Dohme Composition pharmaceutique de type a transition de phase liquide-gel
US4822819A (en) * 1986-11-07 1989-04-18 Alcon Laboratories, Inc. Use of trimoprostil and derivatives in glaucoma therapy
US4822820A (en) * 1986-11-24 1989-04-18 Alcon Laboratories, Inc. Use of tri-methyl PG-F2 a and derivatives in glaucoma therapy
ZA886757B (en) * 1987-09-11 1990-05-30 Syntex Inc Preservative system for ophthalmics formulations
US5110493A (en) * 1987-09-11 1992-05-05 Syntex (U.S.A.) Inc. Ophthalmic NSAID formulations containing a quaternary ammonium preservative and a nonionic surfactant
US5188826A (en) * 1988-02-08 1993-02-23 Insite Vision Incorporated Topical ophthalmic suspensions
IE63392B1 (en) * 1988-02-08 1995-04-19 Insite Vision Inc Ophthalmic suspensions
US5149693A (en) * 1988-03-09 1992-09-22 Alcon Laboratories, Inc. Combination of tobramycin and fluorometholone for topical ophthalmic use
US5149694A (en) * 1988-03-09 1992-09-22 Alcon Laboratories, Inc. Combination of tobramycin and dexamethasone for topical ophthalmic use
US5173507A (en) * 1988-07-18 1992-12-22 Alcon Laboratories, Inc. Prostaglandin combinations in glaucoma therapy
US4960799A (en) * 1988-09-13 1990-10-02 Ciba-Geigy Corporation Stabilized aqueous solutions of pharmaceutically acceptable salts of ortho-(2,6-dichlorophenyl)-aminophenylacetic acid for opthalmic use
US5037647A (en) * 1988-09-15 1991-08-06 Alcon Laboratories, Inc. Aqueous antimicrobial opthalmic solutions comprised of quaternary ammonium compound, citric acid, citrate and sodium chloride
US5145643A (en) * 1990-01-05 1992-09-08 Allergan, Inc. Nonoxidative ophthalmic compositions and methods for preserving and using same
ATE300936T1 (de) * 1992-05-06 2005-08-15 Alcon Lab Inc Anwendung von boral-polyol-komplexen für ophthalmische arzneizusammensetzungen
US5300287A (en) * 1992-11-04 1994-04-05 Alcon Laboratories, Inc. Polymeric antimicrobials and their use in pharmaceutical compositions
WO1994015597A1 (en) * 1993-01-11 1994-07-21 Allergan, Inc. Ophthalmic compositions comprising benzyllauryldimethylammonium chloride

Also Published As

Publication number Publication date
CA2180554C (en) 2001-08-21
JP2954356B2 (ja) 1999-09-27
DK0739197T3 (da) 2001-10-29
AU686917B2 (en) 1998-02-12
DE69522094D1 (de) 2001-09-13
AU4162296A (en) 1996-06-06
HK1012556A1 (en) 1999-08-06
PT739197E (pt) 2001-12-28
EP0739197A1 (de) 1996-10-30
GR3036622T3 (en) 2001-12-31
DE69522094T2 (de) 2001-11-22
US5603929A (en) 1997-02-18
EP0739197B1 (de) 2001-08-08
CA2180554A1 (en) 1996-05-23
US5653972A (en) 1997-08-05
ES2160722T3 (es) 2001-11-16
JPH09503791A (ja) 1997-04-15
WO1996014829A1 (en) 1996-05-23

Similar Documents

Publication Publication Date Title
ATE203897T1 (de) Konservierungsmittelhaltige ophtalmisch anzuwendende arzneizusammensetzungen enthaltend quaternäre polymerammoniumverbindungen
DK0479005T3 (da) Farmaceutisk præparat i form af en gel i dispenseremballage
FI941969L (fi) Shampookoostumuksia, jotka sisältävät hoitavina aineina silikonia, kationista polymeeriä ja öljymäistä nestettä
ATE263579T1 (de) Abgabe von polyethylene glycol-molekül- konjugaten aus abbaubarem hydrogel
FI971033A0 (fi) Metoder foer infoerande av material i huden, samt daerfoer anvaenda kompositioner
MX9705954A (es) Formulaciones y metodos para reducir irritacion de la piel.
FI960892L (fi) Polymeerimatriisit ja niiden käyttö farmaseuttisissa koostumuksissa
NO971889D0 (no) Forbindelser og sammensetninger for levering av aktive midler
IT235830Y1 (it) "raccordo luer-lock con cappuccio di protezione per linee medicali diinfusione-trasfusione."
DK0684958T3 (da) Polymerer indeholdende guanidinogrupper til anvendelse i terapi
DE59407457D1 (de) Blockierung der anlagerung von keimen an menschliche zellen
ATE243196T1 (de) Piperidine und pyrrolidine
PT731714E (pt) Utilizacao de compostos quaternarios de amonio polimericos contendo oxido de polietileno em composicoes farmaceuticas
ATE223204T1 (de) Liposomenzusammensetzung
DE69619052D1 (de) Feste, wasserfreie, pharmazeutische Zubereitungen für vaginale Verwendung
RU95101375A (ru) Производные n-(3-аминопропил)-n-фенил-5,6,7,8-тетрагидронафталин-2-карбоксамида, их получение и применение в терапии
DE69119810D1 (de) Pyrogensorbentmittel
FI944770L (fi) Neurotensiiniin vaikuttavia substituoituja 1-naftyylipyratsoli-3-karboksiamideja, niiden valmistus ja niitä sisältäviä farmaseuttisia koostumuksia
NO953995D0 (no) Ionenolymere som anthelmintica i dyr
IT1274241B (it) Complessi agente terapeutico/matrice polimerica dotati di migliorate caratteristiche di sapore e composizioni farmaceutiche che li contengono
PT996462E (pt) Preparados de combinacoes farmaceuticas contendo eritropoietina e hemoglobinas modificadas
BR9802803A (pt) ação e composições farmacêuticas contendo os mesmos.
ATE83668T1 (de) Pflaster zur transdermalen anwendung.
ES2104456T3 (es) Dispersiones polimeras acuosas.
SE9702793D0 (sv) Novel formulation

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification