ATE106886T1 - Azabicycloamide und -ester als 5-ht3-receptor- antagonisten. - Google Patents
Azabicycloamide und -ester als 5-ht3-receptor- antagonisten.Info
- Publication number
- ATE106886T1 ATE106886T1 AT90312218T AT90312218T ATE106886T1 AT E106886 T1 ATE106886 T1 AT E106886T1 AT 90312218 T AT90312218 T AT 90312218T AT 90312218 T AT90312218 T AT 90312218T AT E106886 T1 ATE106886 T1 AT E106886T1
- Authority
- AT
- Austria
- Prior art keywords
- esters
- azabicycloamides
- receptor antagonists
- antagonists
- receptor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US1989/005097 WO1991007402A1 (en) | 1989-11-17 | 1989-11-17 | Azabicyclo amides and esters as 5-ht3 receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE106886T1 true ATE106886T1 (de) | 1994-06-15 |
Family
ID=22215354
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT90312218T ATE106886T1 (de) | 1989-11-17 | 1990-11-08 | Azabicycloamide und -ester als 5-ht3-receptor- antagonisten. |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP0434202B1 (de) |
JP (1) | JPH0699428B2 (de) |
AT (1) | ATE106886T1 (de) |
CA (1) | CA2030077C (de) |
DE (1) | DE69009715T2 (de) |
DK (1) | DK0434202T3 (de) |
ES (1) | ES2055344T3 (de) |
FI (1) | FI922124A (de) |
IE (1) | IE63420B1 (de) |
PT (1) | PT95895A (de) |
WO (1) | WO1991007402A1 (de) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9027111D0 (en) * | 1990-12-13 | 1991-02-06 | Raychem Ltd | Circuit protection device |
GB9214184D0 (en) * | 1992-07-03 | 1992-08-12 | Smithkline Beecham Plc | Pharmaceuticals |
FR2699533A1 (fr) * | 1992-12-21 | 1994-06-24 | Mouhtaram Mohamed | Dérivés de N-((1,4-dialkyl-6-arylpipérazine-2-yl)méthyl)benzamides. (Isomères cis et trans) Propriétés pharmacologiques et applications. |
AU2005319248A1 (en) * | 2004-12-22 | 2006-06-29 | Memory Pharmaceuticals Corporation | Nicotinic alpha-7 receptor ligands and preparation and uses thereof |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3405134A (en) * | 1965-08-17 | 1968-10-08 | Colgate Palmolive Co | Quinuclidyl esters of aromatic acids |
US4467095A (en) * | 1969-02-10 | 1984-08-21 | Fmc Corporation | Anticholinergic compounds |
US3563995A (en) * | 1969-04-17 | 1971-02-16 | Ian Wellings | Alkyl esters of 1-azabicyclo(2.2.2)oct-2-ene-3-(4 - chloro-3-sulfamoylanilino)-2-carboxylic acid |
GB1293446A (en) * | 1970-07-23 | 1972-10-18 | Rech S Et D Applic Scient Soge | Quinuclidine derivatives, the preparation thereof and pharmaceutical compositions containing them |
FR2531955A1 (fr) * | 1982-08-17 | 1984-02-24 | Pharmuka Lab | Nouveau procede de preparation de derives de la quinuclidine substitues en position 3 |
CH667657A5 (de) * | 1985-01-07 | 1988-10-31 | Sandoz Ag | Carbocyclische und heterocyclische carbonylmethylen- und methylpiperidine und -pyrrolidine. |
GB8525844D0 (en) * | 1985-10-19 | 1985-11-20 | Beecham Group Plc | Compounds |
EP0311724A1 (de) * | 1987-10-16 | 1989-04-19 | Synthelabo | Anxiolytische R-N-(1-Azabicyclo[2.2.2]oct-3-yl)-benzamide und -thiobenzamide |
-
1989
- 1989-11-17 WO PCT/US1989/005097 patent/WO1991007402A1/en active Application Filing
-
1990
- 1990-11-08 DK DK90312218.2T patent/DK0434202T3/da active
- 1990-11-08 EP EP90312218A patent/EP0434202B1/de not_active Expired - Lifetime
- 1990-11-08 DE DE69009715T patent/DE69009715T2/de not_active Expired - Fee Related
- 1990-11-08 AT AT90312218T patent/ATE106886T1/de active
- 1990-11-08 ES ES90312218T patent/ES2055344T3/es not_active Expired - Lifetime
- 1990-11-15 PT PT95895A patent/PT95895A/pt not_active Application Discontinuation
- 1990-11-15 CA CA002030077A patent/CA2030077C/en not_active Expired - Fee Related
- 1990-11-16 IE IE413490A patent/IE63420B1/en not_active IP Right Cessation
- 1990-11-16 JP JP31124190A patent/JPH0699428B2/ja not_active Expired - Lifetime
-
1992
- 1992-05-11 FI FI922124A patent/FI922124A/fi not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IE63420B1 (en) | 1995-04-19 |
DE69009715T2 (de) | 1994-09-22 |
FI922124A0 (fi) | 1992-05-11 |
PT95895A (pt) | 1991-09-13 |
WO1991007402A1 (en) | 1991-05-30 |
DK0434202T3 (da) | 1994-07-04 |
FI922124A (fi) | 1992-05-11 |
CA2030077A1 (en) | 1991-05-18 |
EP0434202A1 (de) | 1991-06-26 |
IE904134A1 (en) | 1991-05-22 |
JPH03170480A (ja) | 1991-07-24 |
EP0434202B1 (de) | 1994-06-08 |
DE69009715D1 (de) | 1994-07-14 |
JPH0699428B2 (ja) | 1994-12-07 |
ES2055344T3 (es) | 1994-08-16 |
CA2030077C (en) | 1995-08-22 |
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