ATA399573A - Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivate - Google Patents

Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivate

Info

Publication number
ATA399573A
ATA399573A AT399573A AT399573A ATA399573A AT A399573 A ATA399573 A AT A399573A AT 399573 A AT399573 A AT 399573A AT 399573 A AT399573 A AT 399573A AT A399573 A ATA399573 A AT A399573A
Authority
AT
Austria
Prior art keywords
aminobenzylpenicillin
derivatives
producing new
new alpha
alpha
Prior art date
Application number
AT399573A
Other languages
English (en)
Other versions
AT331970B (de
Inventor
Masuo Murakami
Ichiro Isaka
Akio Koda
Norio Kawahara
Teruya Kashiwagi
Yukiyasu Murakami
Kuniichiro Yano
Kohzi Nakano
Isao Souzu
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP4511872A external-priority patent/JPS5547036B2/ja
Priority claimed from JP8342472A external-priority patent/JPS4941396A/ja
Priority claimed from JP8510272A external-priority patent/JPS4942692A/ja
Priority claimed from JP8510372A external-priority patent/JPS4942693A/ja
Priority claimed from JP12595272A external-priority patent/JPS4981388A/ja
Priority claimed from JP1991773A external-priority patent/JPS49108092A/ja
Priority claimed from JP3813273A external-priority patent/JPS49125386A/ja
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Application granted granted Critical
Publication of AT331970B publication Critical patent/AT331970B/de
Publication of ATA399573A publication Critical patent/ATA399573A/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT399573A 1972-05-08 1973-05-07 Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivate AT331970B (de)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP4511872A JPS5547036B2 (de) 1972-05-08 1972-05-08
JP8342472A JPS4941396A (de) 1972-08-21 1972-08-21
JP8510272A JPS4942692A (de) 1972-08-25 1972-08-25
JP8510372A JPS4942693A (de) 1972-08-25 1972-08-25
JP12595272A JPS4981388A (de) 1972-12-15 1972-12-15
JP1991773A JPS49108092A (de) 1973-02-18 1973-02-18
JP3813273A JPS49125386A (de) 1973-04-04 1973-04-04

Publications (2)

Publication Number Publication Date
AT331970B AT331970B (de) 1975-12-15
ATA399573A true ATA399573A (de) 1975-12-15

Family

ID=27563884

Family Applications (1)

Application Number Title Priority Date Filing Date
AT399573A AT331970B (de) 1972-05-08 1973-05-07 Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivate

Country Status (10)

Country Link
US (1) US3953428A (de)
AR (2) AR204162A1 (de)
AT (1) AT331970B (de)
BE (1) BE799202A (de)
CA (1) CA1050971A (de)
DE (1) DE2322750A1 (de)
DK (1) DK139754B (de)
FI (1) FI58131C (de)
FR (1) FR2183895B1 (de)
GB (1) GB1407566A (de)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4202900A (en) * 1972-09-27 1980-05-13 Ciba-Geigy Corporation Derivatives of penam-3-carboxylic acid and a pharmaceutical composition containing the same
JPS5751837B2 (de) * 1973-04-05 1982-11-04
US3994874A (en) * 1973-11-07 1976-11-30 Richardson-Merrell Inc. 6-[(2-Oxo-1-pyridinyl)acylamino]penicillin derivatives
US3954734A (en) * 1974-01-21 1976-05-04 Parke, Davis & Company Novel antibacterial amide compounds and process means for producing the same
IL47168A (en) * 1974-05-09 1979-07-25 Toyama Chemical Co Ltd Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
US3989687A (en) * 1974-09-27 1976-11-02 Richardson-Merrell Inc. 4-Oxo-1-pyridinyl penicillin derivatives
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
NZ184434A (en) * 1976-06-30 1979-03-28 Dainippon Pharmaceutical Co Penicillins with a substituted p-hydroxy-benzyl side-chain, and injectable pharmaceutical compositions
GB1579362A (en) * 1977-03-16 1980-11-19 Beecham Group Ltd 6-(a-heterocyclylcarbonyl amino-acetamido)-penicillins and compositions containing them
EP0001041A3 (de) * 1977-07-27 1979-06-27 Sandoz Ag Alpha(Pyridonecarboxylamino)Alpha-acetamid-substituierte Penicilline und Cephalosporine, Verfahren zu ihrer Herstellung, ihre Verwendung als Arzneimittel; Pyridone für ihre Herstellung
US4219477A (en) * 1977-12-06 1980-08-26 Nippon Chemiphar Company Limited Penicillin derivatives
US4231928A (en) * 1979-04-24 1980-11-04 Bristol-Myers Company Antibacterial agents
JPS5651488A (en) * 1979-10-02 1981-05-09 Meiji Seika Kaisha Ltd Penicillin derivative and its preparation
US5281612A (en) * 1982-09-09 1994-01-25 Warner-Lambert Company Naphthyridine antibacterial agents
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
IT1215277B (it) * 1985-05-27 1990-01-31 Pomezia Roma A Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi.
US5273973A (en) * 1988-10-24 1993-12-28 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl esters
CA2001203C (en) * 1988-10-24 2001-02-13 Thomas P. Demuth, Jr. Novel antimicrobial dithiocarbamoyl quinolones
US5180719A (en) * 1988-10-24 1993-01-19 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl lactam esters
US5491139A (en) * 1988-10-24 1996-02-13 The Procter & Gamble Company Antimicrobial quinolonyl lactams
EP0997466A1 (de) * 1988-10-24 2000-05-03 PROCTER & GAMBLE PHARMACEUTICALS, INC. Antimikrobielle Laktamchinolone
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
WO1991016327A1 (en) * 1990-04-18 1991-10-31 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl lactams
FR2713637B1 (fr) * 1993-12-15 1996-01-05 Cird Galderma Nouveaux composés bi-aromatiques dérivés d'amide, compositions pharmaceutiques et cosmétiques les contenant et utilisations.
BR9811362A (pt) * 1997-08-25 2000-08-22 Neurogen Corp Composto
US6143760A (en) 1997-08-25 2000-11-07 Neurogen Corporation Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands
EP1765347A4 (de) * 2004-06-04 2008-10-01 Univ California Verbindungen mit ionentransporterhöhender wirkung durch mutanten cftr und ihre verwendung
AR085013A1 (es) * 2011-01-26 2013-08-07 Sanofi Aventis Derivados de acido 3-heteroaroilamino-propionico sustituidos y su uso como sustancias farmaceuticas

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1180745A (en) * 1966-10-04 1970-02-11 Beecham Group Ltd Penicillins
US3668198A (en) * 1970-06-01 1972-06-06 Squibb & Sons Inc {60 -ureido-2,4,6-cycloheptatrienylmethylpenicillins
US3711471A (en) * 1971-02-03 1973-01-16 Bristol Myers Co Purification of 6-{8 d-{60 -(3-guanyl-1-ureido)phenylacetamido{9 {0 penicillanic acid

Also Published As

Publication number Publication date
FI58131C (fi) 1980-12-10
AT331970B (de) 1975-12-15
DK139754B (da) 1979-04-09
AU5504573A (en) 1974-11-07
DK139754C (de) 1979-09-24
AR204162A1 (es) 1975-11-28
GB1407566A (en) 1975-09-24
FR2183895A1 (de) 1973-12-21
US3953428A (en) 1976-04-27
FI58131B (fi) 1980-08-29
FR2183895B1 (de) 1976-07-02
CA1050971A (en) 1979-03-20
DE2322750A1 (de) 1973-11-29
BE799202A (fr) 1973-08-31
AR204813A1 (es) 1976-03-05

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Legal Events

Date Code Title Description
ELA Expired due to lapse of time
ELJ Ceased due to non-payment of the annual fee