BE799202A - Procede de preparation de derives d'ampicilline substitues par un groupe acyle heterocyclique, - Google Patents

Procede de preparation de derives d'ampicilline substitues par un groupe acyle heterocyclique,

Info

Publication number
BE799202A
BE799202A BE130836A BE130836A BE799202A BE 799202 A BE799202 A BE 799202A BE 130836 A BE130836 A BE 130836A BE 130836 A BE130836 A BE 130836A BE 799202 A BE799202 A BE 799202A
Authority
BE
Belgium
Prior art keywords
acyl group
derivatives substituted
heterocyclic acyl
preparing
ampicillin derivatives
Prior art date
Application number
BE130836A
Other languages
English (en)
Inventor
M Murakami
I Isaka
A Koda
N Kawahara
I Kashiwagi
Y Murakami
K Yano
Nakano
I Souzu
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP4511872A external-priority patent/JPS5547036B2/ja
Priority claimed from JP8342472A external-priority patent/JPS4941396A/ja
Priority claimed from JP8510372A external-priority patent/JPS4942693A/ja
Priority claimed from JP8510272A external-priority patent/JPS4942692A/ja
Priority claimed from JP12595272A external-priority patent/JPS4981388A/ja
Priority claimed from JP1991773A external-priority patent/JPS49108092A/ja
Priority claimed from JP3813273A external-priority patent/JPS49125386A/ja
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Publication of BE799202A publication Critical patent/BE799202A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE130836A 1972-05-08 1973-05-07 Procede de preparation de derives d'ampicilline substitues par un groupe acyle heterocyclique, BE799202A (fr)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP4511872A JPS5547036B2 (fr) 1972-05-08 1972-05-08
JP8342472A JPS4941396A (fr) 1972-08-21 1972-08-21
JP8510372A JPS4942693A (fr) 1972-08-25 1972-08-25
JP8510272A JPS4942692A (fr) 1972-08-25 1972-08-25
JP12595272A JPS4981388A (fr) 1972-12-15 1972-12-15
JP1991773A JPS49108092A (fr) 1973-02-18 1973-02-18
JP3813273A JPS49125386A (fr) 1973-04-04 1973-04-04

Publications (1)

Publication Number Publication Date
BE799202A true BE799202A (fr) 1973-08-31

Family

ID=27563884

Family Applications (1)

Application Number Title Priority Date Filing Date
BE130836A BE799202A (fr) 1972-05-08 1973-05-07 Procede de preparation de derives d'ampicilline substitues par un groupe acyle heterocyclique,

Country Status (10)

Country Link
US (1) US3953428A (fr)
AR (2) AR204813A1 (fr)
AT (1) AT331970B (fr)
BE (1) BE799202A (fr)
CA (1) CA1050971A (fr)
DE (1) DE2322750A1 (fr)
DK (1) DK139754B (fr)
FI (1) FI58131C (fr)
FR (1) FR2183895B1 (fr)
GB (1) GB1407566A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3954734A (en) * 1974-01-21 1976-05-04 Parke, Davis & Company Novel antibacterial amide compounds and process means for producing the same

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4202900A (en) * 1972-09-27 1980-05-13 Ciba-Geigy Corporation Derivatives of penam-3-carboxylic acid and a pharmaceutical composition containing the same
JPS5751837B2 (fr) * 1973-04-05 1982-11-04
US3994874A (en) * 1973-11-07 1976-11-30 Richardson-Merrell Inc. 6-[(2-Oxo-1-pyridinyl)acylamino]penicillin derivatives
IL47168A (en) * 1974-05-09 1979-07-25 Toyama Chemical Co Ltd Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
US3989687A (en) * 1974-09-27 1976-11-02 Richardson-Merrell Inc. 4-Oxo-1-pyridinyl penicillin derivatives
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
NZ184434A (en) * 1976-06-30 1979-03-28 Dainippon Pharmaceutical Co Penicillins with a substituted p-hydroxy-benzyl side-chain, and injectable pharmaceutical compositions
GB1579362A (en) * 1977-03-16 1980-11-19 Beecham Group Ltd 6-(a-heterocyclylcarbonyl amino-acetamido)-penicillins and compositions containing them
EP0001041A3 (fr) * 1977-07-27 1979-06-27 Sandoz Ag Alpha(pyridonecarboxylamino)-pénicillines, et céphalosporines, alpha-acétamido-substituées; procédé pour leur préparation, leur usage pharmaceutique; pyridones intermédiaires pour leur préparation
GB2010250B (en) * 1977-12-06 1982-07-14 Nippon Chemiphar Co Penicillin and cephalosporin derivatives and a process for producing the same
US4231928A (en) * 1979-04-24 1980-11-04 Bristol-Myers Company Antibacterial agents
JPS5651488A (en) * 1979-10-02 1981-05-09 Meiji Seika Kaisha Ltd Penicillin derivative and its preparation
US5281612A (en) * 1982-09-09 1994-01-25 Warner-Lambert Company Naphthyridine antibacterial agents
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
IT1215277B (it) * 1985-05-27 1990-01-31 Pomezia Roma A Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi.
US5273973A (en) * 1988-10-24 1993-12-28 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl esters
US5491139A (en) * 1988-10-24 1996-02-13 The Procter & Gamble Company Antimicrobial quinolonyl lactams
EP0366189A3 (fr) * 1988-10-24 1992-01-02 Norwich Eaton Pharmaceuticals, Inc. Lactames-quinolones antimicrobiennes
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
US5180719A (en) * 1988-10-24 1993-01-19 Norwich Eaton Pharmaceuticals, Inc. Antimicrobial quinolonyl lactam esters
CA2001203C (fr) * 1988-10-24 2001-02-13 Thomas P. Demuth, Jr. Dithiocarbamoyl quinolones antimicrobiens
EP0525057B1 (fr) * 1990-04-18 2000-06-14 Procter & Gamble Pharmaceuticals, Inc. Quinolonyle lactames anti-microbiens
FR2713637B1 (fr) * 1993-12-15 1996-01-05 Cird Galderma Nouveaux composés bi-aromatiques dérivés d'amide, compositions pharmaceutiques et cosmétiques les contenant et utilisations.
PL338783A1 (en) * 1997-08-25 2000-11-20 Neurogen Corp Substituted 4-oxo-naphtyridin-3-carboxamides as ligands of cerebral gaba receptors
US6143760A (en) * 1997-08-25 2000-11-07 Neurogen Corporation Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands
EP1765347A4 (fr) * 2004-06-04 2008-10-01 Univ California Composes intervenant dans l'acceleration du transport ionique par le cftr mutant, et utilisations desdits composes
UY33874A (es) * 2011-01-26 2012-08-31 Sanofi Aventis Derivados de ácido 3-heteroaroilamino-propiónico sustituidos y su uso como sustancias farmacéuticas

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1180745A (en) * 1966-10-04 1970-02-11 Beecham Group Ltd Penicillins
US3668198A (en) * 1970-06-01 1972-06-06 Squibb & Sons Inc {60 -ureido-2,4,6-cycloheptatrienylmethylpenicillins
US3711471A (en) * 1971-02-03 1973-01-16 Bristol Myers Co Purification of 6-{8 d-{60 -(3-guanyl-1-ureido)phenylacetamido{9 {0 penicillanic acid

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3954734A (en) * 1974-01-21 1976-05-04 Parke, Davis & Company Novel antibacterial amide compounds and process means for producing the same

Also Published As

Publication number Publication date
US3953428A (en) 1976-04-27
FI58131C (fi) 1980-12-10
DE2322750A1 (de) 1973-11-29
CA1050971A (fr) 1979-03-20
DK139754C (fr) 1979-09-24
ATA399573A (de) 1975-12-15
DK139754B (da) 1979-04-09
AT331970B (de) 1975-12-15
FR2183895B1 (fr) 1976-07-02
FI58131B (fi) 1980-08-29
FR2183895A1 (fr) 1973-12-21
GB1407566A (en) 1975-09-24
AR204162A1 (es) 1975-11-28
AR204813A1 (es) 1976-03-05
AU5504573A (en) 1974-11-07

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