ATA142574A - PROCESS FOR THE PREPARATION OF NEW 7-ALPHA-AMINOACYL-3-HALOGENCEPHALOSPORINES - Google Patents

PROCESS FOR THE PREPARATION OF NEW 7-ALPHA-AMINOACYL-3-HALOGENCEPHALOSPORINES

Info

Publication number
ATA142574A
ATA142574A AT142574A AT142574A ATA142574A AT A142574 A ATA142574 A AT A142574A AT 142574 A AT142574 A AT 142574A AT 142574 A AT142574 A AT 142574A AT A142574 A ATA142574 A AT A142574A
Authority
AT
Austria
Prior art keywords
halogencephalosporines
aminoacyl
alpha
preparation
new
Prior art date
Application number
AT142574A
Other languages
German (de)
Other versions
AT333953B (en
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of ATA142574A publication Critical patent/ATA142574A/en
Application granted granted Critical
Publication of AT333953B publication Critical patent/AT333953B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02—Preparation
    • C07D501/04—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT142574A 1973-02-23 1974-02-21 PROCESS FOR THE PREPARATION OF NEW 7-ALPHA-AMINOACYL-3-HALOGENCEPHALOSPORINES AT333953B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US33538173A 1973-02-23 1973-02-23

Publications (2)

Publication Number Publication Date
ATA142574A true ATA142574A (en) 1976-04-15
AT333953B AT333953B (en) 1976-12-27

Family

ID=23311540

Family Applications (1)

Application Number Title Priority Date Filing Date
AT142574A AT333953B (en) 1973-02-23 1974-02-21 PROCESS FOR THE PREPARATION OF NEW 7-ALPHA-AMINOACYL-3-HALOGENCEPHALOSPORINES

Country Status (37)

Country Link
JP (4) JPS6139313B2 (en)
AR (1) AR199510A1 (en)
AT (1) AT333953B (en)
BE (1) BE811495A (en)
BR (1) BR7401384D0 (en)
CA (1) CA1016537A (en)
CH (1) CH593988A5 (en)
CS (1) CS187409B2 (en)
CY (1) CY1043A (en)
DD (1) DD110278A5 (en)
DE (1) DE2408698C2 (en)
DK (1) DK153157C (en)
EG (1) EG11104A (en)
ES (1) ES423531A1 (en)
FI (1) FI63035C (en)
FR (1) FR2218877B1 (en)
GB (1) GB1461323A (en)
GT (1) GT197432133A (en)
HK (1) HK20080A (en)
HU (1) HU166849B (en)
IE (1) IE39046B1 (en)
IL (1) IL44262A (en)
IN (1) IN139620B (en)
KE (1) KE3027A (en)
MW (1) MW674A1 (en)
MY (1) MY8100024A (en)
NL (1) NL179057C (en)
NO (2) NO148375C (en)
OA (1) OA04809A (en)
PH (1) PH9616A (en)
PL (1) PL88702B1 (en)
RO (1) RO64663A (en)
SE (1) SE411212B (en)
SU (1) SU676166A3 (en)
YU (1) YU36970B (en)
ZA (1) ZA741191B (en)
ZM (1) ZM3574A1 (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT342197B (en) * 1975-02-20 1978-03-28 Ciba Geigy Ag NEW PROCESS FOR PRODUCING 3-CEPHEM CONNECTIONS
CH619233A5 (en) * 1975-07-31 1980-09-15 Ciba Geigy Ag
CH622802A5 (en) * 1975-08-20 1981-04-30 Ciba Geigy Ag
IE45158B1 (en) * 1976-08-16 1982-06-30 Lilly Co Eli 3-chloro-cephem synthesis
DE3508258A1 (en) * 1985-03-08 1986-09-18 Bayer Ag, 5090 Leverkusen SS LACTAMANTIBIOTICS, METHOD FOR THE PRODUCTION AND THEIR USE AS AND IN MEDICINAL PRODUCTS
DE3509618A1 (en) 1985-03-16 1986-09-18 Bayer Ag, 5090 Leverkusen SS LACTAM ANTIBIOTICS, METHOD FOR THE PRODUCTION AND THEIR USE AS A MEDICINAL PRODUCT
JPS6436445U (en) * 1987-08-28 1989-03-06
DE3803169A1 (en) 1988-02-03 1989-08-17 Bayer Ag SS LACTAM ANTIBIOTICS, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS AND IN MEDICINAL PRODUCTS
ES2010075A6 (en) * 1989-01-10 1989-10-16 Antibioticos Sa Process for the preparation of 3-chloro-cefem compounds.
JP2539459Y2 (en) * 1991-12-18 1997-06-25 三重ホーロー株式会社 Assembled garbage incinerator
IT1255458B (en) * 1992-05-11 1995-11-02 Col Marco Da PROCEDURE FOR THE PREPARATION OF HALOGENATED BETA-LACTAMIC DERIVATIVES
ES2079327B1 (en) 1994-12-13 1996-08-01 Lilly Sa PHARMACEUTICAL FORMULATIONS OF CEFACLOR.
CN101805357B (en) * 2010-04-28 2012-01-11 陶灵刚 Cefaclor compound and novel preparation method thereof
CN103588790A (en) * 2013-11-29 2014-02-19 中国科学院长春应用化学研究所 Preparation method of 7-amino-3-chloro-3-cephem-4-carboxylic acid-p-nitrobenzyl ester
CN106632400A (en) * 2016-12-16 2017-05-10 石家庄柏奇化工有限公司 Method for preparing 7-ACCA by removing 4-nitrobenzyl through catalytic hydrogenation of Pd-C

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3641021A (en) * 1969-04-18 1972-02-08 Lilly Co Eli 3 7-(ring-substituted) cephalosporin compounds
FR2143211B1 (en) * 1971-06-24 1975-10-31 Fujisawa Pharmaceutical Co
AR206201A1 (en) * 1972-06-29 1976-07-07 Ciba Geigy Ag PROCEDURE FOR OBTAINING ACID COMPOUNDS 7BETA-AMINO-3-CEFEM-3-01-4-CARBOXILICO0-SUBSTITUIDOS

Also Published As

Publication number Publication date
PH9616A (en) 1976-01-20
JPS49110689A (en) 1974-10-22
NL179057C (en) 1986-07-01
BE811495A (en) 1974-08-22
CS187409B2 (en) 1979-01-31
NO148377C (en) 1983-09-28
NO792681L (en) 1974-08-26
ZA741191B (en) 1975-10-29
MW674A1 (en) 1975-04-09
AU6591674A (en) 1975-08-28
DE2408698C2 (en) 1983-11-10
AT333953B (en) 1976-12-27
DK153157B (en) 1988-06-20
HK20080A (en) 1980-04-25
YU39974A (en) 1982-06-18
IL44262A0 (en) 1974-05-16
NL7402489A (en) 1974-08-27
SE411212B (en) 1979-12-10
NO148375B (en) 1983-06-20
CY1043A (en) 1980-08-01
NO148377B (en) 1983-06-20
JPS6139313B2 (en) 1986-09-03
FI63035B (en) 1982-12-31
YU36970B (en) 1984-08-31
BR7401384D0 (en) 1974-11-05
CH593988A5 (en) 1977-12-30
SU676166A3 (en) 1979-07-25
IE39046B1 (en) 1978-07-19
GT197432133A (en) 1975-08-16
NL179057B (en) 1986-02-03
JPS6140237B2 (en) 1986-09-08
JPS56138190A (en) 1981-10-28
DK153157C (en) 1988-10-31
KE3027A (en) 1980-03-14
NO148375C (en) 1983-09-28
FR2218877B1 (en) 1977-03-11
PL88702B1 (en) 1976-09-30
JPS56138191A (en) 1981-10-28
IL44262A (en) 1977-08-31
FR2218877A1 (en) 1974-09-20
JPS56138192A (en) 1981-10-28
IE39046L (en) 1974-08-23
GB1461323A (en) 1977-01-13
AR199510A1 (en) 1974-09-09
EG11104A (en) 1976-12-31
DE2408698A1 (en) 1974-09-05
JPS6140236B2 (en) 1986-09-08
CA1016537A (en) 1977-08-30
FI63035C (en) 1983-04-11
NO740606L (en) 1974-08-26
RO64663A (en) 1979-02-15
HU166849B (en) 1975-06-28
IN139620B (en) 1976-07-10
OA04809A (en) 1980-08-31
MY8100024A (en) 1981-12-31
DD110278A5 (en) 1974-12-12
JPS6140235B2 (en) 1986-09-08
ZM3574A1 (en) 1975-11-21
ES423531A1 (en) 1976-05-16

Similar Documents

Publication Publication Date Title
AT333726B (en) PROCESS FOR THE PREPARATION OF NEW N-CINNAMOYL OR HYDROCINNAMOYLAMINOBENZOIC ACIDS
AT342793B (en) PROCESS FOR THE PREPARATION OF NEW CHOLESTERANS
AT330761B (en) PROCESS FOR THE PREPARATION OF NEW ACYLAMINOSAUREAMIDES
AT333953B (en) PROCESS FOR THE PREPARATION OF NEW 7-ALPHA-AMINOACYL-3-HALOGENCEPHALOSPORINES
AT337698B (en) PROCESS FOR THE PREPARATION OF NEW 2-HYDROXYPHENYL -1-OXA-4- AZASPIRO-ALKANE DERIVATIVES
AT338247B (en) PROCESS FOR THE PREPARATION OF NEW 2-AMINOALKANOYLAMIDOBENZOPHENONE
AT343292B (en) PROCESS FOR THE PREPARATION OF NEW STEROID-3-OXIME DERIVATIVES
AT330161B (en) PROCESS FOR THE PREPARATION OF NEW BIPHENYLBUTANOLS
AT348536B (en) PROCESS FOR THE PREPARATION OF NEW 4-OXO-2-IMIDAZOLIDINYLIDEN UREA
AT337201B (en) PROCESS FOR THE PREPARATION OF NEW 5-PHENYLSULFINYLBENZIMIDAZOLYL-2-CARBAMINE ALKYLESTERS
AT339283B (en) PROCESS FOR THE PREPARATION OF NEW 3,4-DIAMINO-BENZOPHENONE
AT335449B (en) PROCESS FOR THE PREPARATION OF NEW THIADIAZOLYLIMIDAZOLIDINONES
AT341509B (en) PROCESS FOR THE PREPARATION OF NEW CHLOROACETANILIDES
AT331780B (en) PROCESS FOR THE PREPARATION OF NEW 3-N-BUTYLAMINO-4-PHENOXY-5-ALCOXYMETHYL SULPHAMOYLBENZOIC ACIDS
AT327950B (en) PROCESS FOR THE PREPARATION OF NEW 1,2-OXAPHOSPHOLANES
AT325059B (en) PROCESS FOR THE PREPARATION OF NEW THIAZOLOTRIAZOLYLPHOSPHONOTHIOATES
AT343685B (en) PROCESS FOR THE PREPARATION OF NEW D-XYLOFURANOSE DERIVATIVES
ATA695076A (en) PROCESS FOR THE PREPARATION OF NEW 5-METHYL-7-HYDROXY-ISOFLAVONE DERIVATIVES
ATA722475A (en) PROCESS FOR THE PREPARATION OF NEW 3-N-BUTYLAMINO-4-PHENOXY-5-ALCOXYMETHYL-SULFAMOYLBENZOIC ACIDS
ATA722375A (en) PROCESS FOR THE PREPARATION OF NEW 3-N-BUTYLAMINO-4-PHENOXY-5-ALCOXYMETHYL SULPHAMOYLBENZOIC ACIDS
ATA895175A (en) PROCESS FOR THE PREPARATION OF NEW DERIVATIVES OF DIGITOXIGENIN-ALFA-L-ARABINOSIDE
ATA895275A (en) PROCESS FOR THE PREPARATION OF NEW DERIVATIVES OF DIGITOXIGENIN-ALFA-L-ARABINOSIDE
AT341502B (en) PROCESS FOR THE PREPARATION OF NEW 3,4-DIAMINO-BENZOPHENONE
ATA746976A (en) PROCESS FOR THE PREPARATION OF NEW 3,4-DIAMINO-BENZOPHENONE
ATA691775A (en) PROCESS FOR THE PREPARATION OF NEW 1,1-DIPHENYL -2-HYDROXY-3-AMINOPROPANERIVATIVES

Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee
EWE Authorization for restitution
ELA Expired due to lapse of time
REN Ceased due to non-payment of the annual fee