AT356115B - METHOD FOR PRODUCING SUBSTITUTED AMINO-CHINAZOLINE DERIVATIVES AND THEIR SALTS - Google Patents

METHOD FOR PRODUCING SUBSTITUTED AMINO-CHINAZOLINE DERIVATIVES AND THEIR SALTS

Info

Publication number
AT356115B
AT356115B AT386977A AT386977A AT356115B AT 356115 B AT356115 B AT 356115B AT 386977 A AT386977 A AT 386977A AT 386977 A AT386977 A AT 386977A AT 356115 B AT356115 B AT 356115B
Authority
AT
Austria
Prior art keywords
salts
substituted amino
producing substituted
chinazoline derivatives
chinazoline
Prior art date
Application number
AT386977A
Other languages
German (de)
Other versions
ATA386977A (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ATA386977A publication Critical patent/ATA386977A/en
Application granted granted Critical
Publication of AT356115B publication Critical patent/AT356115B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT386977A 1976-06-15 1977-06-01 METHOD FOR PRODUCING SUBSTITUTED AMINO-CHINAZOLINE DERIVATIVES AND THEIR SALTS AT356115B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US69620176A 1976-06-15 1976-06-15

Publications (2)

Publication Number Publication Date
ATA386977A ATA386977A (en) 1979-09-15
AT356115B true AT356115B (en) 1980-04-10

Family

ID=24796111

Family Applications (1)

Application Number Title Priority Date Filing Date
AT386977A AT356115B (en) 1976-06-15 1977-06-01 METHOD FOR PRODUCING SUBSTITUTED AMINO-CHINAZOLINE DERIVATIVES AND THEIR SALTS

Country Status (34)

Country Link
JP (1) JPS52153985A (en)
AR (1) AR218251A1 (en)
AT (1) AT356115B (en)
BE (1) BE855656A (en)
BG (3) BG35748A3 (en)
CA (1) CA1068698A (en)
CH (3) CH638203A5 (en)
CS (1) CS202069B2 (en)
DD (1) DD131021A5 (en)
DE (1) DE2725019A1 (en)
DK (1) DK146625C (en)
EG (1) EG12922A (en)
ES (1) ES459364A1 (en)
FI (1) FI66853C (en)
FR (1) FR2355015A1 (en)
GB (1) GB1548856A (en)
GR (1) GR72288B (en)
HK (1) HK31481A (en)
HU (1) HU177883B (en)
IE (1) IE45423B1 (en)
IL (1) IL52167A (en)
LU (1) LU77530A1 (en)
MY (1) MY8100270A (en)
NL (1) NL172543C (en)
NO (1) NO147838C (en)
NZ (1) NZ184168A (en)
PH (1) PH22196A (en)
PL (3) PL111221B1 (en)
PT (1) PT66617B (en)
RO (3) RO73050A (en)
SE (2) SE435380B (en)
SU (2) SU1033002A3 (en)
YU (1) YU40164B (en)
ZA (1) ZA773014B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3346675A1 (en) * 1983-12-23 1985-07-04 Beiersdorf Ag, 2000 Hamburg SUBSTITUTED 1- (4-AMINO-6,7-DIALKOXY-CHINAZOLINYL) -4- CYCLOHEXENYL DERIVATIVES OF PIPERAZINE AND HOMOPIPERAZINE, METHODS FOR THE PRODUCTION THEREOF, AND THEIR USE, AND ITS RELATED PRODUCTS
AT384218B (en) * 1985-12-04 1987-10-12 Gerot Pharmazeutika METHOD FOR PRODUCING NEW CHINAZOLINE DERIVATIVES
CA2077252C (en) * 1992-08-31 2001-04-10 Khashayar Karimian Methods of making ureas and guanidines, and intermediates therefor
IL112249A (en) 1994-01-25 2001-11-25 Warner Lambert Co Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
US5654307A (en) * 1994-01-25 1997-08-05 Warner-Lambert Company Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
IL112248A0 (en) 1994-01-25 1995-03-30 Warner Lambert Co Tricyclic heteroaromatic compounds and pharmaceutical compositions containing them
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3511836A (en) 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines
US3669968A (en) 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines
JPS4966691A (en) * 1972-10-30 1974-06-27
US3935213A (en) 1973-12-05 1976-01-27 Pfizer Inc. Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives
JPS50126682A (en) * 1974-03-25 1975-10-04

Also Published As

Publication number Publication date
SU1033002A3 (en) 1983-07-30
CH638516A5 (en) 1983-09-30
DE2725019A1 (en) 1977-12-22
NO147838C (en) 1983-06-22
IE45423B1 (en) 1982-08-25
FI66853B (en) 1984-08-31
RO77308A (en) 1981-08-17
DK240877A (en) 1977-12-16
FI771741A (en) 1977-12-16
EG12922A (en) 1980-03-31
CA1068698A (en) 1979-12-25
CH638203A5 (en) 1983-09-15
SE450120B (en) 1987-06-09
CH638517A5 (en) 1983-09-30
IL52167A (en) 1981-01-30
PL105558B1 (en) 1979-10-31
AU2558377A (en) 1978-09-07
AR218251A1 (en) 1980-05-30
BG35748A3 (en) 1984-06-15
JPS5543465B2 (en) 1980-11-06
NL7705939A (en) 1977-12-19
NZ184168A (en) 1979-08-31
BG35594A3 (en) 1984-05-15
NO147838B (en) 1983-03-14
BG35747A3 (en) 1984-06-15
LU77530A1 (en) 1979-03-26
SU946402A3 (en) 1982-07-23
RO77330A (en) 1981-06-22
ZA773014B (en) 1978-04-26
DD131021A5 (en) 1978-05-24
ATA386977A (en) 1979-09-15
HK31481A (en) 1981-07-10
IL52167A0 (en) 1977-07-31
JPS52153985A (en) 1977-12-21
SE8107554L (en) 1981-12-16
IE45423L (en) 1977-12-15
PL111221B1 (en) 1980-08-30
PT66617A (en) 1977-06-01
CS202069B2 (en) 1980-12-31
DK146625B (en) 1983-11-21
PH22196A (en) 1988-06-28
DK146625C (en) 1984-06-04
HU177883B (en) 1982-01-28
FR2355015A1 (en) 1978-01-13
PT66617B (en) 1978-10-27
ES459364A1 (en) 1978-03-16
YU40164B (en) 1985-08-31
SE7705745L (en) 1977-12-16
NL172543C (en) 1983-09-16
MY8100270A (en) 1981-12-31
FR2355015B1 (en) 1981-07-24
BE855656A (en) 1977-12-14
YU132677A (en) 1982-08-31
GB1548856A (en) 1979-07-18
RO73050A (en) 1981-08-30
NO771919L (en) 1977-12-16
PL113012B1 (en) 1980-11-29
PL198874A1 (en) 1978-04-10
FI66853C (en) 1984-12-10
SE435380B (en) 1984-09-24
NL172543B (en) 1983-04-18
GR72288B (en) 1983-10-17

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Legal Events

Date Code Title Description
EIH Change in the person of patent owner
ELJ Ceased due to non-payment of the annual fee
ELJ Ceased due to non-payment of the annual fee