AT321917B - Verfahren zur herstellung von neuen alpha-aryl-4-subst. piperidinoalkanolderivaten und ihren pharmazeutisch annehmbaren säureadditionssalzen - Google Patents
Verfahren zur herstellung von neuen alpha-aryl-4-subst. piperidinoalkanolderivaten und ihren pharmazeutisch annehmbaren säureadditionssalzenInfo
- Publication number
- AT321917B AT321917B AT1115372A AT1115372A AT321917B AT 321917 B AT321917 B AT 321917B AT 1115372 A AT1115372 A AT 1115372A AT 1115372 A AT1115372 A AT 1115372A AT 321917 B AT321917 B AT 321917B
- Authority
- AT
- Austria
- Prior art keywords
- alcanol
- subst
- piperidino
- aryl
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22182172A | 1972-01-28 | 1972-01-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AT321917B true AT321917B (de) | 1975-04-25 |
Family
ID=22829539
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT246074*1A AT323742B (de) | 1972-01-28 | 1972-12-29 | Verfahren zur herstellung von neuen alpha-aryl-4-substituierten piperidinoalkanolderivaten und ihren pharmazeutisch annehmbaren saureadditionssalzen |
| AT1115372A AT321917B (de) | 1972-01-28 | 1972-12-29 | Verfahren zur herstellung von neuen alpha-aryl-4-subst. piperidinoalkanolderivaten und ihren pharmazeutisch annehmbaren säureadditionssalzen |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT246074*1A AT323742B (de) | 1972-01-28 | 1972-12-29 | Verfahren zur herstellung von neuen alpha-aryl-4-substituierten piperidinoalkanolderivaten und ihren pharmazeutisch annehmbaren saureadditionssalzen |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS5115035B2 (xx) |
| AR (1) | AR195314A1 (xx) |
| AT (2) | AT323742B (xx) |
| AU (1) | AU467361B2 (xx) |
| BE (1) | BE794597A (xx) |
| CA (1) | CA978946A (xx) |
| CH (2) | CH587820A5 (xx) |
| CS (1) | CS177834B2 (xx) |
| DD (1) | DD103239A5 (xx) |
| DE (1) | DE2303306C3 (xx) |
| DK (1) | DK136713B (xx) |
| ES (1) | ES410731A1 (xx) |
| FR (1) | FR2181690B1 (xx) |
| GB (1) | GB1413138A (xx) |
| HU (1) | HU166477B (xx) |
| IE (1) | IE36983B1 (xx) |
| IL (1) | IL41060A (xx) |
| LU (1) | LU66916A1 (xx) |
| NL (1) | NL175410C (xx) |
| NO (1) | NO140057C (xx) |
| PH (1) | PH10264A (xx) |
| PL (1) | PL89095B1 (xx) |
| SE (1) | SE382058B (xx) |
| SU (1) | SU464997A3 (xx) |
| YU (1) | YU36013B (xx) |
| ZA (1) | ZA728544B (xx) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3941795A (en) | 1974-02-08 | 1976-03-02 | Richardson-Merrell Inc. | α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES |
| US4254130A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| US4254129A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| IT1200123B (it) * | 1985-09-27 | 1989-01-05 | Ind Chimica Srl | Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo |
| US4742175A (en) * | 1986-05-07 | 1988-05-03 | Merrell Dow Pharmaceuticals Inc. | Preparation of polymorphically pure terfenadine |
| JPS63101760U (xx) * | 1986-12-19 | 1988-07-02 | ||
| IT1205685B (it) * | 1987-05-26 | 1989-03-31 | Erregierre Spa | Processo per la preparazione di alfa-(alchilfenil)-4-(idrossi difenilmetil)-1-piperidina butanolo |
| IL93499A0 (en) * | 1989-02-28 | 1990-11-29 | Merrell Dow Pharma | Preparation of the low melting polymorphic form of terfenadine |
| CA2015390A1 (en) * | 1989-05-01 | 1990-11-01 | Frederick J. Mccarty | Process for the preparation of the high melting polymorphic of terfenadine |
| DE3917241A1 (de) * | 1989-05-26 | 1990-11-29 | Schaper & Bruemmer Gmbh | 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate |
| EP0596120A4 (en) * | 1991-08-09 | 1994-07-06 | Yoshitomi Pharmaceutical | Thiophene compound. |
| CN1183769A (zh) * | 1995-05-08 | 1998-06-03 | 赫彻斯特马里恩鲁斯公司 | α-(取代的烷基苯基)-4-(羟基二苯基甲基)-1-哌啶丁醇衍生物,其制备和其用作抗组胺剂、抗变应性剂和支气管扩张药的用途 |
| EP0864653B1 (de) * | 1997-03-11 | 2004-03-03 | Aventis Pharmaceuticals Inc. | Verfahren zur Herstellung von 4-(4-(4-(Hydroxydiphenyl)-1-piperidinyl)-1-hydroxybutyl)-alpha,alpha-dimenthylphenylessigsäure und phosphorylierter Derivate |
| US7498345B2 (en) * | 2004-09-17 | 2009-03-03 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| JPWO2006043691A1 (ja) * | 2004-10-18 | 2008-05-29 | 株式会社リバース・プロテオミクス研究所 | 創薬標的タンパク質及び標的遺伝子、並びにスクリーニング方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3081303A (en) * | 1961-10-13 | 1963-03-12 | Searle & Co | 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols |
| GB1242169A (en) * | 1969-04-09 | 1971-08-11 | Ucb Sa | Piperidine derivatives |
-
1972
- 1972-12-04 ZA ZA728544A patent/ZA728544B/xx unknown
- 1972-12-05 IE IE1689/72A patent/IE36983B1/xx unknown
- 1972-12-08 PH PH14156A patent/PH10264A/en unknown
- 1972-12-11 AU AU49893/72A patent/AU467361B2/en not_active Ceased
- 1972-12-12 IL IL41060A patent/IL41060A/xx unknown
- 1972-12-15 GB GB5799572A patent/GB1413138A/en not_active Expired
- 1972-12-20 CH CH1854272A patent/CH587820A5/xx not_active IP Right Cessation
- 1972-12-20 CH CH1381476A patent/CH593259A5/xx not_active IP Right Cessation
- 1972-12-27 JP JP47130136A patent/JPS5115035B2/ja not_active Expired
- 1972-12-29 AT AT246074*1A patent/AT323742B/de not_active IP Right Cessation
- 1972-12-29 AT AT1115372A patent/AT321917B/de not_active IP Right Cessation
-
1973
- 1973-01-08 YU YU34/73A patent/YU36013B/xx unknown
- 1973-01-16 CA CA161,413A patent/CA978946A/en not_active Expired
- 1973-01-17 HU HURI498A patent/HU166477B/hu unknown
- 1973-01-18 ES ES410731A patent/ES410731A1/es not_active Expired
- 1973-01-22 NL NLAANVRAGE7300873,A patent/NL175410C/xx not_active IP Right Cessation
- 1973-01-24 SE SE7300974A patent/SE382058B/xx active Protection Beyond IP Right Term
- 1973-01-24 FR FR7302503A patent/FR2181690B1/fr not_active Expired
- 1973-01-24 DE DE2303306A patent/DE2303306C3/de not_active Expired
- 1973-01-25 DD DD168482A patent/DD103239A5/xx unknown
- 1973-01-26 PL PL1973160419A patent/PL89095B1/pl unknown
- 1973-01-26 LU LU66916A patent/LU66916A1/xx unknown
- 1973-01-26 DK DK44973AA patent/DK136713B/da not_active IP Right Cessation
- 1973-01-26 NO NO326/73A patent/NO140057C/no unknown
- 1973-01-26 CS CS630A patent/CS177834B2/cs unknown
- 1973-01-26 BE BE794597D patent/BE794597A/xx not_active IP Right Cessation
- 1973-01-26 AR AR246313A patent/AR195314A1/es active
- 1973-01-27 SU SU1878074A patent/SU464997A3/ru active
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EFA | Change in the company name | ||
| ELA | Expired due to lapse of time |