AR217460A1 - Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales - Google Patents

Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales

Info

Publication number
AR217460A1
AR217460A1 AR270785A AR27078578A AR217460A1 AR 217460 A1 AR217460 A1 AR 217460A1 AR 270785 A AR270785 A AR 270785A AR 27078578 A AR27078578 A AR 27078578A AR 217460 A1 AR217460 A1 AR 217460A1
Authority
AR
Argentina
Prior art keywords
isoquinolein
isoquinolyl
thiazol
imino
tetrahydro
Prior art date
Application number
AR270785A
Other languages
English (en)
Spanish (es)
Original Assignee
Rhone Poulenc Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7701516A external-priority patent/FR2378030A1/fr
Priority claimed from FR7739028A external-priority patent/FR2412545A1/fr
Application filed by Rhone Poulenc Ind filed Critical Rhone Poulenc Ind
Application granted granted Critical
Publication of AR217460A1 publication Critical patent/AR217460A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C07D217/16Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
AR270785A 1977-01-20 1978-01-20 Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales AR217460A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7701516A FR2378030A1 (fr) 1977-01-20 1977-01-20 Nouveau derive de l'isoquinoleine, sa preparation et les compositions qui le contiennent
FR7739028A FR2412545A1 (fr) 1977-12-23 1977-12-23 Nouveaux derives de l'isoquinoleine, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
AR217460A1 true AR217460A1 (es) 1980-03-31

Family

ID=26219809

Family Applications (2)

Application Number Title Priority Date Filing Date
AR270785A AR217460A1 (es) 1977-01-20 1978-01-20 Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales
AR275407A AR219963A1 (es) 1977-01-20 1979-02-05 Procedimiento para preparar nuevos derivados de (alcoil(c1-c10)-3-isoquinolil-5-imino)-3-tetrahidro-1,5,10,10a-tiazol(3,4-b)- isoquinoleina

Family Applications After (1)

Application Number Title Priority Date Filing Date
AR275407A AR219963A1 (es) 1977-01-20 1979-02-05 Procedimiento para preparar nuevos derivados de (alcoil(c1-c10)-3-isoquinolil-5-imino)-3-tetrahidro-1,5,10,10a-tiazol(3,4-b)- isoquinoleina

Country Status (25)

Country Link
US (1) US4153698A (cs)
JP (1) JPS5914037B2 (cs)
AR (2) AR217460A1 (cs)
AT (1) AT361481B (cs)
AU (1) AU510044B2 (cs)
CA (1) CA1091674A (cs)
CH (1) CH633010A5 (cs)
CS (2) CS195350B2 (cs)
DE (1) DE2802453C3 (cs)
DK (1) DK143343C (cs)
ES (2) ES466192A1 (cs)
FI (1) FI62314C (cs)
GB (1) GB1574281A (cs)
GR (1) GR61726B (cs)
HU (1) HU174219B (cs)
IE (1) IE46375B1 (cs)
IL (1) IL53841A (cs)
LU (1) LU78895A1 (cs)
NL (1) NL7800383A (cs)
NO (1) NO780202L (cs)
NZ (1) NZ186282A (cs)
OA (1) OA05859A (cs)
PT (1) PT67545B (cs)
SE (1) SE7800681L (cs)
SU (2) SU730309A3 (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU797580A3 (ru) * 1977-11-10 1981-01-15 Рон-Пуленк Эндюстри (Фирма) Способ получени производных изохино-лиНА, иХ СОлЕй, РАцЕМАТОВ или ОпТичЕС-КиХ изОМЕРОВ
FR2456098A2 (fr) * 1977-12-23 1980-12-05 Rhone Poulenc Ind Nouveaux derives de l'isoquinoleine, leur preparation et les compositions pharmaceutiques qui les contiennent
NL7908655A (nl) * 1978-12-07 1980-06-10 Rhone Poulenc Ind Nieuwe thienopyridine-derivaten, de bereiding ervan, alsmede farmaceutische preparaten, die de nieuwe derivaten bevatten.
FR2456111A1 (fr) * 1979-05-09 1980-12-05 Rhone Poulenc Ind Nouveaux derives de l'indole, leur preparation et les medicaments qui les contiennent
NL8002540A (nl) * 1979-05-09 1980-11-11 Rhone Poulenc Ind Nieuwe isochinoline derivaten, werkwijzen ter bereiding ervan en farmaceutische preparaten, die de nieuwe derivaten bevatten.
AU6496380A (en) * 1979-12-04 1981-06-11 Rhone-Poulenc Industries Thiazolo(3,4-b) isoquinoline derivatives
US4269842A (en) * 1979-12-05 1981-05-26 Rhone-Poulenc Industries Method for treating rhinoviral complaints
US6582728B1 (en) * 1992-07-08 2003-06-24 Inhale Therapeutic Systems, Inc. Spray drying of macromolecules to produce inhaleable dry powders

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL169076C (nl) * 1975-08-06 1982-06-01 Rhone Poulenc Ind Werkwijze voor het bereiden of vervaardigen van farmacologische preparaten met een analgetische en antipyretische werking, alsmede werkwijze voor het bereiden van geneeskrachtige verbindingen, welke geschikt zijn voor gebruik in dergelijke preparaten.

Also Published As

Publication number Publication date
SU776560A3 (ru) 1980-10-30
DK143343C (da) 1982-01-25
DK27178A (da) 1978-07-21
PT67545B (fr) 1979-06-15
ATA39378A (de) 1980-08-15
FI62314B (fi) 1982-08-31
NZ186282A (en) 1980-02-21
JPS5914037B2 (ja) 1984-04-02
SU730309A3 (ru) 1980-04-25
FI62314C (fi) 1982-12-10
NO780202L (no) 1978-07-21
NL7800383A (nl) 1978-07-24
SE7800681L (sv) 1978-07-21
IL53841A0 (en) 1978-04-30
DE2802453B2 (de) 1981-04-02
AU510044B2 (en) 1980-06-05
CH633010A5 (fr) 1982-11-15
AT361481B (de) 1981-03-10
IE46375B1 (en) 1983-05-18
OA05859A (fr) 1981-05-31
AR219963A1 (es) 1980-09-30
FI780182A7 (fi) 1978-07-21
AU3261178A (en) 1979-08-02
JPS53116399A (en) 1978-10-11
DE2802453A1 (de) 1978-07-27
GR61726B (en) 1978-12-29
LU78895A1 (fr) 1978-09-18
ES466192A1 (es) 1978-10-16
US4153698A (en) 1979-05-08
CS195349B2 (en) 1980-01-31
HU174219B (hu) 1979-11-28
IE780126L (en) 1978-07-20
PT67545A (fr) 1978-02-01
CS195350B2 (en) 1980-01-31
DE2802453C3 (de) 1982-03-25
GB1574281A (en) 1980-09-03
CA1091674A (fr) 1980-12-16
ES468630A1 (es) 1978-12-01
IL53841A (en) 1980-10-26
DK143343B (da) 1981-08-10

Similar Documents

Publication Publication Date Title
AR228444A1 (es) Procedimiento para preparar derivados de 5-bencil-tiazolidin-2,4-diona y sus sales
MX4811E (es) Procedimiento para preparar derivados de prostaglandina
AR220686A1 (es) Procedimiento para obtener derivados de 2 amino-2-desoxi-3-o-(propilcarbamoilmetil)-carbamoilmetil-glucopiranosa y sus sales
AR230270A1 (es) Procedimiento para preparar nuevos derivados de 2-alquiltio-3(-alcanoil alcoxicarbonil)-5-halogeno-6-fenoxi-bencimidazol substituidos
MX4899E (es) Procedimiento para preparar derivados de espirohidantoina
AR227882A1 (es) Procedimiento para la preparacion de nuevos derivados de pirido(1,2-a)pirimidina y sus sales
AR221081A1 (es) Procedimiento para preparar derivados de fenoximetil-piperidino-propoxi-indol
AR222666A1 (es) Procedimiento para preparar derivados de 5-tetrazolil dibenzo-(b,f)tiepinas
AR222311A1 (es) Procedimiento para preparar derivados de 1,2,3,3 alpha,8,8 alpha,hexahidropirrol-(2,3-b)indol y sus sales
AR216438A1 (es) Procedimiento para preparar derivados de difenil-alquil-aza-bicicloalcano
MX151851A (es) Procedimiento mejorado para preparar derivados de triacina
AR223160A1 (es) Procedimiento para preparar derivados de 3-aminoalquiltiazolidindiona(2,4)y sus sales
AR217460A1 (es) Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales
AR213184A1 (es) Procedimiento para preparar derivados de 1,4-etan-6-oxo-perhidroquinoleina y sus sales
AR221352A1 (es) Un procedimiento para preparar derivados de trans-4a-fenil-octahidro-1h2-pirindinas y sus sales
MX4911E (es) Procedimiento para preparar derivados de quinoleina
MX5160E (es) Procedimiento mejorado para preparar derivados de aminoalcoholes
MX5534E (es) Procedimiento para la preparacion de derivados de nicotinamida
AR222310A1 (es) Procedimiento para preparar derivados de 5-bencil-(1,2,4)-oxadiazol
AR229078A1 (es) Procedimiento para obtener derivados de 6,7-dihidro-3h-imidazo(1,2-a)-purin-9-(4h)-ona y sus sales
AR216058A1 (es) Procedimiento de preparacion de sulfoximidas sustituidas,y sus sales
AR231975A1 (es) Procedimiento para preparar derivados de 2-aminoalquil-2-piridilamidas
ES490505A0 (es) Procedimiento de preparacion de nuevos derivados benzo-as- triazinos y de sus sales de adicion acidas, farmaceuticamen-te aceptables
AR228852A1 (es) Procedimiento para preparar derivados de 1,1'bifenil-2-il-alquilamina y sus sales
MX5454E (es) Procedimiento para preparar derivados de la 1,2,4-triazin-5-ona