AR214303A1 - Un procedimiento para preparar nuevos derivados de(cicloalquilalquiloxi-(o tio,o-sulfonil-alquil)-(o alquiloxi fenoxi)-1amino-3-propanol-2 - Google Patents

Un procedimiento para preparar nuevos derivados de(cicloalquilalquiloxi-(o tio,o-sulfonil-alquil)-(o alquiloxi fenoxi)-1amino-3-propanol-2

Info

Publication number
AR214303A1
AR214303A1 AR265315A AR26531576A AR214303A1 AR 214303 A1 AR214303 A1 AR 214303A1 AR 265315 A AR265315 A AR 265315A AR 26531576 A AR26531576 A AR 26531576A AR 214303 A1 AR214303 A1 AR 214303A1
Authority
AR
Argentina
Prior art keywords
alkyloxyphenoxy
1amine
cycloalkylalkyloxy
thio
sulfonyl
Prior art date
Application number
AR265315A
Other languages
English (en)
Spanish (es)
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Application granted granted Critical
Publication of AR214303A1 publication Critical patent/AR214303A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
    • C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
    • C07D303/24—Ethers with hydroxy compounds containing no oxirane rings with polyhydroxy compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
AR265315A 1975-11-06 1976-11-02 Un procedimiento para preparar nuevos derivados de(cicloalquilalquiloxi-(o tio,o-sulfonil-alquil)-(o alquiloxi fenoxi)-1amino-3-propanol-2 AR214303A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7533899A FR2330383A1 (fr) 1975-11-06 1975-11-06 Nouveaux ethers de phenols substitues, leurs sels, leur preparation et les medicaments qui les renferment

Publications (1)

Publication Number Publication Date
AR214303A1 true AR214303A1 (es) 1979-05-31

Family

ID=9162099

Family Applications (1)

Application Number Title Priority Date Filing Date
AR265315A AR214303A1 (es) 1975-11-06 1976-11-02 Un procedimiento para preparar nuevos derivados de(cicloalquilalquiloxi-(o tio,o-sulfonil-alquil)-(o alquiloxi fenoxi)-1amino-3-propanol-2

Country Status (24)

Country Link
US (2) US4252984A (de)
JP (1) JPS5848543B2 (de)
AR (1) AR214303A1 (de)
AT (1) AT344683B (de)
AU (1) AU501581B2 (de)
BE (1) BE847801A (de)
CA (1) CA1072981A (de)
CH (1) CH602582A5 (de)
DE (1) DE2649605C3 (de)
DK (1) DK145119C (de)
ES (1) ES452920A1 (de)
FI (1) FI62829C (de)
FR (1) FR2330383A1 (de)
GB (1) GB1515978A (de)
GR (1) GR61363B (de)
IE (1) IE43645B1 (de)
IL (1) IL50814A (de)
LU (1) LU76117A1 (de)
NL (1) NL179051C (de)
NO (1) NO142034C (de)
NZ (1) NZ182498A (de)
PT (1) PT65780B (de)
SE (1) SE433208B (de)
ZA (1) ZA766338B (de)

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DE3125870C2 (de) * 1980-07-09 1994-09-15 William John Louis 3-Aminopropoxyphenyl Derivate, ihre Herstellung und sie enthaltende Arzneimittel
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JPS57108047A (en) * 1980-11-06 1982-07-05 Sandoz Ag 3-aminopropoxyphenyl derivative, manufacture and pharmaceutical composition containing same
FI76551C (fi) 1980-11-06 1988-11-10 Sandoz Ag Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 3-aminopropoxifenylderivat.
US5347050A (en) * 1980-11-06 1994-09-13 Richard Berthold 3-aminopropoxyphenyl derivatives, their preparation and pharmaceutical compositions containing them
DE3125636A1 (de) * 1981-06-30 1983-01-13 Merck Patent Gmbh, 6100 Darmstadt 1-(p-2-isopropoxyethoxymethyl-phenoxy)-3-isopropylamino-propan-2-ol zur senkung des augeninnendrucks und ophtalmikum, enthalten diese verbindung
FR2512443A1 (fr) * 1981-09-10 1983-03-11 Synthelabo Derives de phenoxy-3 propanol-2, leur preparation et leur application en therapeutique
DE3151201A1 (de) * 1981-12-23 1983-07-28 Beiersdorf Ag, 2000 Hamburg Substituierte phenoxyalkanolamine und phenoxyalkanol-cycloalkylamine, verfahren zu ihrer herstellung, diese verbindungen enthaltende pharmazeutische zubereitungen und zwischenprodukte
US4450172A (en) * 1982-03-10 1984-05-22 E. I. Du Pont De Nemours And Company Antihypertensive polyhalohydroxyisopropyl phenylalka(e)noic acid esters of alkylaminohydroxypropyloxyphenylalkyl alcohols
FR2536390B1 (fr) * 1982-11-22 1986-03-21 Synthelabo Isomere s du betaxolol, sa preparation et son application en therapeutique
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CA1262729A (en) * 1983-10-19 1989-11-07 Leo Alig Phenoxypropanolamines
NZ211815A (en) * 1984-05-15 1988-11-29 Warner Lambert Co Preparation of 1-((3,4-dimethoxyphenethyl)amino)-3- (3-tolyloxy)-2-propanol
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ES8609190A1 (es) * 1985-02-07 1986-07-16 Pharma Investi S A Un procedimiento para preparar eteres fenolicos
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EP0252007A3 (de) * 1986-06-28 1989-07-05 Ciba-Geigy Ag 2-Propanolderivate als Korrosionsinhibitoren
US4694022A (en) * 1986-12-24 1987-09-15 Alcon Laboratories, Inc. Fatty acid salts of betaxolol useful in the treatment of glaucoma
DE3866984D1 (en) * 1987-07-21 1992-01-30 Hoffmann La Roche Phenoxypropanolamine.
FR2672594B1 (fr) * 1991-02-08 1994-07-01 Synthelabo Derives d'ethers de phenols, leur preparation et leur application en therapeutique.
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US5942633A (en) * 1996-06-19 1999-08-24 Abbott Laboratories Process for the selective alkylation of betaxolol intermediates
US5731463A (en) * 1996-09-23 1998-03-24 Abbott Laboratories Selective alkylation of an alcohol substituted phenol compound
CA2330611A1 (en) 1998-05-22 1999-12-02 The Board Of Trustees Of The Leland Stanford Junior University Bifunctional molecules and therapies based thereon
US6258350B1 (en) 1999-01-20 2001-07-10 Alcon Manufacturing, Ltd. Sustained release ophthalmic formulation
BR0015938A (pt) 1999-11-30 2002-08-27 Alcon Inc Uso de antagonistas beta-adrenoceptores para a fabricação de um medicamento para o tratamento de desordens da retina externa
JP2004511435A (ja) * 2000-07-27 2004-04-15 ファルマシア・コーポレーション うっ血性心不全の処置のための、エポキシ−ステロイド型アルドステロン拮抗薬とβ−アドレナリン作動性拮抗薬の併用療法
DE60234057D1 (de) 2001-07-25 2009-11-26 Raptor Pharmaceutical Inc Zusammensetzungen und verfahren zur modulation des transports durch die blut-hirn-schranke
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AT323131B (de) * 1935-11-15 1975-06-25 Boehringer Sohn Ingelheim Verfahren zur herstellung von neuen racemischen oder optisch aktiven n,n'-bis-(3-subst.phenoxy-2-hydroxy-1-propyl)-alpha,omega-diaminoalkanen sowie deren saureadditionssalzen
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CA956632A (en) * 1969-05-16 1974-10-22 Yoshitomi Pharmaceutical Industries Phenoxy-aminopropanol derivatives
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Also Published As

Publication number Publication date
DK145119C (da) 1983-02-14
JPS5285146A (en) 1977-07-15
CA1072981A (en) 1980-03-04
AU1925976A (en) 1978-05-11
FI763132A (de) 1977-05-07
US4252984A (en) 1981-02-24
ES452920A1 (es) 1977-11-01
CH602582A5 (de) 1978-07-31
NO142034C (no) 1980-06-18
FI62829B (fi) 1982-11-30
FI62829C (fi) 1983-03-10
PT65780A (fr) 1976-12-01
SE7612177L (sv) 1977-05-07
DE2649605B2 (de) 1980-07-10
FR2330383B1 (de) 1979-09-21
ATA812076A (de) 1977-12-15
IL50814A (en) 1979-11-30
IE43645L (en) 1977-05-06
NL7612123A (nl) 1977-05-10
NO763732L (no) 1977-05-09
NZ182498A (en) 1978-04-03
JPS5848543B2 (ja) 1983-10-28
NL179051B (nl) 1986-02-03
US4311708A (en) 1982-01-19
GR61363B (en) 1978-10-30
DK145119B (da) 1982-09-06
IE43645B1 (en) 1981-04-22
AU501581B2 (en) 1979-06-21
LU76117A1 (de) 1978-07-10
NL179051C (nl) 1986-07-01
AT344683B (de) 1978-08-10
NO142034B (no) 1980-03-10
GB1515978A (en) 1978-06-28
SE433208B (sv) 1984-05-14
DK495476A (da) 1977-05-07
BE847801A (fr) 1977-02-14
DE2649605C3 (de) 1981-04-02
DE2649605A1 (de) 1977-05-18
IL50814A0 (en) 1977-01-31
PT65780B (fr) 1978-05-10
ZA766338B (en) 1977-10-26
FR2330383A1 (fr) 1977-06-03

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