ES528066A0 - Procedimiento para preparar nuevos derivados del azabiciclo heptano. - Google Patents

Procedimiento para preparar nuevos derivados del azabiciclo heptano.

Info

Publication number
ES528066A0
ES528066A0 ES528066A ES528066A ES528066A0 ES 528066 A0 ES528066 A0 ES 528066A0 ES 528066 A ES528066 A ES 528066A ES 528066 A ES528066 A ES 528066A ES 528066 A0 ES528066 A0 ES 528066A0
Authority
ES
Spain
Prior art keywords
azabiciclo
heptane
procedure
new derivatives
prepare new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES528066A
Other languages
English (en)
Other versions
ES8501401A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Publication of ES8501401A1 publication Critical patent/ES8501401A1/es
Publication of ES528066A0 publication Critical patent/ES528066A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES528066A 1982-12-17 1983-12-15 Procedimiento para preparar nuevos derivados del azabiciclo heptano. Granted ES528066A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19823246757 DE3246757A1 (de) 1982-12-17 1982-12-17 Neue 2-azabicyclo(2.2.1)heptan-derivate, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie 2-azabicyclo(2.2.1)heptan-derivate als zwischenprodukte und verfahren zu deren herstellung

Publications (2)

Publication Number Publication Date
ES8501401A1 ES8501401A1 (es) 1984-11-16
ES528066A0 true ES528066A0 (es) 1984-11-16

Family

ID=6180952

Family Applications (2)

Application Number Title Priority Date Filing Date
ES528066A Granted ES528066A0 (es) 1982-12-17 1983-12-15 Procedimiento para preparar nuevos derivados del azabiciclo heptano.
ES530388A Expired ES8500946A1 (es) 1982-12-17 1984-03-08 Procedimiento para preparar derivados del 2-azabiciclo-2.2.1-heptano.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES530388A Expired ES8500946A1 (es) 1982-12-17 1984-03-08 Procedimiento para preparar derivados del 2-azabiciclo-2.2.1-heptano.

Country Status (10)

Country Link
EP (1) EP0113880A3 (es)
JP (1) JPS59130268A (es)
KR (1) KR840006971A (es)
AU (1) AU2249583A (es)
DE (1) DE3246757A1 (es)
DK (1) DK581183A (es)
ES (2) ES528066A0 (es)
GR (1) GR79480B (es)
PT (1) PT77825B (es)
ZA (1) ZA839347B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3303344A1 (de) 1983-02-02 1984-08-02 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung von n-alkylierten aminosaeuren und deren estern
US5684016A (en) * 1984-04-12 1997-11-04 Hoechst Aktiengesellschaft Method of treating cardiac insufficiency
DE3839127A1 (de) * 1988-11-19 1990-05-23 Hoechst Ag Pyrrolidon-2-carbonsaeure-derivate mit psychotroper wirkung
DD284030A5 (de) 1988-11-24 1990-10-31 Hoechst Ag,De Verfahren zur herstellung von peptiden mit bradykinin-antagonistischer wirkung
FR2655989B1 (fr) * 1989-12-20 1992-02-28 Adir Nouveaux derives d'amino-acides substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US6121280A (en) * 1998-03-24 2000-09-19 Pfizer Inc. Azabicyclic rotomase inhibitors
RU2712097C1 (ru) * 2018-09-28 2020-01-24 Общество с ограниченной ответственностью "Необиотек" Ингибитор дипептидилпептидазы-4 для лечения сахарного диабета 2-го типа, соединения (варианты)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492381A1 (fr) * 1980-10-21 1982-04-23 Science Union & Cie Nouveaux acides aza bicyclo alcane carboxyliques substitues leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme

Also Published As

Publication number Publication date
ES530388A0 (es) 1984-11-01
PT77825A (de) 1984-01-01
DK581183D0 (da) 1983-12-16
ES8501401A1 (es) 1984-11-16
ES8500946A1 (es) 1984-11-01
EP0113880A3 (en) 1984-09-26
KR840006971A (ko) 1984-12-07
AU2249583A (en) 1984-06-21
DK581183A (da) 1984-06-18
JPS59130268A (ja) 1984-07-26
PT77825B (de) 1986-05-27
DE3246757A1 (de) 1984-06-20
EP0113880A2 (de) 1984-07-25
GR79480B (es) 1984-10-30
ZA839347B (en) 1984-08-29

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19980504