AU2249583A - 2-azabicyclo(2,2.1)heptane derivatives and intermediates - Google Patents

2-azabicyclo(2,2.1)heptane derivatives and intermediates

Info

Publication number
AU2249583A
AU2249583A AU22495/83A AU2249583A AU2249583A AU 2249583 A AU2249583 A AU 2249583A AU 22495/83 A AU22495/83 A AU 22495/83A AU 2249583 A AU2249583 A AU 2249583A AU 2249583 A AU2249583 A AU 2249583A
Authority
AU
Australia
Prior art keywords
azabicyclo
intermediates
heptane derivatives
heptane
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU22495/83A
Inventor
Reinhard Becker
Rainer Henning
Hansjorg Urbach
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Publication of AU2249583A publication Critical patent/AU2249583A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU22495/83A 1982-12-17 1983-12-16 2-azabicyclo(2,2.1)heptane derivatives and intermediates Abandoned AU2249583A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3246757 1982-12-17
DE19823246757 DE3246757A1 (en) 1982-12-17 1982-12-17 NEW 2-AZABICYCLO (2.2.1) HEPTAN DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR SUBSTANCES AND THE USE THEREOF, AND 2-AZABICYCLO (2.2.1) HEPTAN DERIVATIVES AS INTERMEDIATE PRODUCTS AND METHOD FOR THE PRODUCTION THEREOF

Publications (1)

Publication Number Publication Date
AU2249583A true AU2249583A (en) 1984-06-21

Family

ID=6180952

Family Applications (1)

Application Number Title Priority Date Filing Date
AU22495/83A Abandoned AU2249583A (en) 1982-12-17 1983-12-16 2-azabicyclo(2,2.1)heptane derivatives and intermediates

Country Status (10)

Country Link
EP (1) EP0113880A3 (en)
JP (1) JPS59130268A (en)
KR (1) KR840006971A (en)
AU (1) AU2249583A (en)
DE (1) DE3246757A1 (en)
DK (1) DK581183A (en)
ES (2) ES8501401A1 (en)
GR (1) GR79480B (en)
PT (1) PT77825B (en)
ZA (1) ZA839347B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU617224B2 (en) * 1988-11-19 1991-11-21 Hoechst Aktiengesellschaft Pyrrolidone-2-carboxylic acid derivatives having a psychotropic action

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3303344A1 (en) 1983-02-02 1984-08-02 Hoechst Ag, 6230 Frankfurt METHOD FOR PRODUCING N-ALKYLATED AMINO ACIDS AND THEIR ESTERS
US5684016A (en) * 1984-04-12 1997-11-04 Hoechst Aktiengesellschaft Method of treating cardiac insufficiency
DD284030A5 (en) 1988-11-24 1990-10-31 Hoechst Ag,De PROCESS FOR THE PREPARATION OF PEPTIDES WITH BRADYKININ-ANTAGONISTIC EFFECT
FR2655989B1 (en) * 1989-12-20 1992-02-28 Adir NOVEL SUBSTITUTED AMINO ACID DERIVATIVES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
US6121280A (en) * 1998-03-24 2000-09-19 Pfizer Inc. Azabicyclic rotomase inhibitors
RU2712097C1 (en) * 2018-09-28 2020-01-24 Общество с ограниченной ответственностью "Необиотек" Dipeptidyl peptidase-4 inhibitor for treating type 2 diabetes mellitus, compounds (versions)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492381A1 (en) * 1980-10-21 1982-04-23 Science Union & Cie NOVEL AZA BICYCLO ALKANE CARBOXYLIC ACIDS SUBSTITUTED IN THEIR PREPARATION METHODS AND THEIR USE AS AN ENZYME INHIBITOR

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU617224B2 (en) * 1988-11-19 1991-11-21 Hoechst Aktiengesellschaft Pyrrolidone-2-carboxylic acid derivatives having a psychotropic action

Also Published As

Publication number Publication date
ES528066A0 (en) 1984-11-16
ZA839347B (en) 1984-08-29
JPS59130268A (en) 1984-07-26
PT77825B (en) 1986-05-27
DE3246757A1 (en) 1984-06-20
KR840006971A (en) 1984-12-07
EP0113880A3 (en) 1984-09-26
ES530388A0 (en) 1984-11-01
ES8500946A1 (en) 1984-11-01
PT77825A (en) 1984-01-01
ES8501401A1 (en) 1984-11-16
GR79480B (en) 1984-10-30
DK581183A (en) 1984-06-18
DK581183D0 (en) 1983-12-16
EP0113880A2 (en) 1984-07-25

Similar Documents

Publication Publication Date Title
AU576317B2 (en) 2-thiol- or 2-alkylthio- imidazoles, and intermediates
AU541843B2 (en) Substituted 1,2-diaminocyclobutene-3,4-diones
AU566510B2 (en) Pharmaceutical 1,4-benzodiazepine-2-ones
AU563950B2 (en) 2,2 -disubstituted-1,3-oxepine derivatives
AU8553282A (en) 1(1,2,4-triazoyl/1,3-diazoyl)-2-hydroxy-(n)-phenyl-alkanes
AU1792983A (en) 2,3-dihydrobenzofurans
AU2249583A (en) 2-azabicyclo(2,2.1)heptane derivatives and intermediates
AU1575383A (en) 1,4-dihyropyridine derivatives
AU2435784A (en) 8,10-dideazaminopterins
AU537214B2 (en) 1,1-alkanediol-penicilin derivatives and analogues
AU2599884A (en) 1,8-dihydroxy-10-acyl-9-anthrones
AU2611884A (en) 1,2,3-oxathiazolidin; 1-oxa-3-aza-2-sila-cyclopentan and 1,3,2-oxaphospholidin derivatives
AU531892B2 (en) 1,1-dioxopenicillanoyloxymethyl 6-(-2-amino-2-phenyl- acetamido)penicillanates
AU564232B2 (en) 2:-substituted-spiro benzofuran(2,1:) cycloalkanes
AU8413382A (en) 1,4-piperizine derivatives
AU563796B2 (en) 1:-substituted-spiro(oxazolidine-5,3:-indoline)- -2,2:4-trione derivatives
AU568295B2 (en) 1,2,4-triazol-i-yl-propionitrile derivatives
EP0093485A3 (en) Process for the preparation of substituted 3-oxa-1-aza-bicyclo(4.2.0)octan-8-ones, and intermediates obtained thereby
AU1968883A (en) 15-cycloaliphatic derivatives of 13,14-didehydro- carboprostacyclins
AU3016084A (en) Substituted benzopentathiepins, process therefor and intermediates
AU551883B2 (en) 2,5-bis-perfluoroalkyl-3,4-dicarbonylalkoxypyrroles
AU1176983A (en) 2,3-dihydro-1h-pyrrolizines
AU8879882A (en) 1,2,3-thiadiazol-5-yl-urea derivatives
AU8879782A (en) 1,2,3-thiadiazol-5-yl-urea derivatives
AU636164B2 (en) 2,3-dihydro-1-hydroxy-3-oxo-2-(1-substituted-4-piperidinyl)- 1N-isoindole derivatives