AR204003A1 - PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2- (1-PIPERAZINYL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS - Google Patents
PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2- (1-PIPERAZINYL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTSInfo
- Publication number
- AR204003A1 AR204003A1 AR253060A AR25306074A AR204003A1 AR 204003 A1 AR204003 A1 AR 204003A1 AR 253060 A AR253060 A AR 253060A AR 25306074 A AR25306074 A AR 25306074A AR 204003 A1 AR204003 A1 AR 204003A1
- Authority
- AR
- Argentina
- Prior art keywords
- oxopyride
- piperazinyl
- pyrimidine
- procedure
- pharmaceutically acceptable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP3845373A JPS5546400B2 (en) | 1973-04-03 | 1973-04-03 | |
| JP5654473A JPS565753B2 (en) | 1973-05-21 | 1973-05-21 | |
| JP6446473A JPS565755B2 (en) | 1973-06-07 | 1973-06-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR204003A1 true AR204003A1 (en) | 1975-11-12 |
Family
ID=27289838
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR253060A AR204003A1 (en) | 1973-04-03 | 1974-01-01 | PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2- (1-PIPERAZINYL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS |
| AR258571A AR204660A1 (en) | 1973-04-03 | 1975-01-01 | PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2 (1-PIPERAZINIL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR258571A AR204660A1 (en) | 1973-04-03 | 1975-01-01 | PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2 (1-PIPERAZINIL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID |
Country Status (11)
| Country | Link |
|---|---|
| AR (2) | AR204003A1 (en) |
| AT (1) | AT340931B (en) |
| CA (1) | CA1066701A (en) |
| CH (1) | CH593281A5 (en) |
| ES (1) | ES424851A1 (en) |
| FI (1) | FI56011C (en) |
| IE (1) | IE39102B1 (en) |
| NL (1) | NL186087C (en) |
| NO (1) | NO142221C (en) |
| PH (2) | PH10529A (en) |
| SE (1) | SE416051B (en) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1209163B (en) * | 1979-12-21 | 1989-07-10 | Unibios S P A Trecate Novara | PROCEDURE FOR THE MANUFACTURE OF: 6-ALCOSSICARBONIL-8-ETHYL-5-OXO-5,8 DIIDRO-APERTA PAR. SQUARE 2,3-DCHIUSA PAR. SQUARE-PRIMIDINE 2-REPLACED AND ACID CORRESPONDING BOOKS. |
| KR101763656B1 (en) | 2009-06-29 | 2017-08-01 | 인사이트 홀딩스 코포레이션 | Pyrimidinones as pi3k inhibitors |
| WO2011075643A1 (en) | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted heteroaryl fused derivatives as pi3k inhibitors |
| TW201130842A (en) | 2009-12-18 | 2011-09-16 | Incyte Corp | Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors |
| JP5961187B2 (en) | 2010-12-20 | 2016-08-02 | インサイト・ホールディングス・コーポレイションＩｎｃｙｔｅ Ｈｏｌｄｉｎｇｓ Ｃｏｒｐｏｒａｔｉｏｎ | N- (1- (substituted phenyl) ethyl) -9H-purin-6-amine as a PI3K inhibitor |
| WO2013033569A1 (en) | 2011-09-02 | 2013-03-07 | Incyte Corporation | Heterocyclylamines as pi3k inhibitors |
| AR090548A1 (en) | 2012-04-02 | 2014-11-19 | Incyte Corp | BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS |
| WO2015191677A1 (en) | 2014-06-11 | 2015-12-17 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors |
| NZ734993A (en) | 2015-02-27 | 2024-03-22 | Incyte Holdings Corp | Salts of pi3k inhibitor and processes for their preparation |
| US9732097B2 (en) | 2015-05-11 | 2017-08-15 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
| US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
-
1974
- 1974-01-01 AR AR253060A patent/AR204003A1/en active
- 1974-01-30 CA CA191,286A patent/CA1066701A/en not_active Expired
- 1974-02-01 SE SE7401361A patent/SE416051B/en not_active IP Right Cessation
- 1974-02-04 NL NLAANVRAGE7401509,A patent/NL186087C/en not_active IP Right Cessation
- 1974-02-04 FI FI298/74A patent/FI56011C/en active
- 1974-02-04 NO NO740349A patent/NO142221C/en unknown
- 1974-02-14 CH CH205474A patent/CH593281A5/en not_active IP Right Cessation
- 1974-03-25 IE IE00650/74A patent/IE39102B1/en unknown
- 1974-04-02 ES ES424851A patent/ES424851A1/en not_active Expired
- 1974-04-03 AT AT277774A patent/AT340931B/en not_active IP Right Cessation
- 1974-04-03 PH PH15698A patent/PH10529A/en unknown
-
1975
- 1975-01-01 AR AR258571A patent/AR204660A1/en active
- 1975-09-05 PH PH17546A patent/PH10984A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NL186087C (en) | 1990-09-17 |
| CH593281A5 (en) | 1977-11-30 |
| NO740349L (en) | 1974-10-04 |
| NL7401509A (en) | 1974-10-07 |
| ATA277774A (en) | 1977-05-15 |
| NL186087B (en) | 1990-04-17 |
| FI56011B (en) | 1979-07-31 |
| CA1066701A (en) | 1979-11-20 |
| AR204660A1 (en) | 1976-02-20 |
| FI56011C (en) | 1979-11-12 |
| SE416051B (en) | 1980-11-24 |
| IE39102B1 (en) | 1978-08-02 |
| NO142221C (en) | 1980-07-16 |
| AT340931B (en) | 1978-01-10 |
| ES424851A1 (en) | 1976-06-01 |
| PH10529A (en) | 1977-05-30 |
| IE39102L (en) | 1974-10-03 |
| NO142221B (en) | 1980-04-08 |
| PH10984A (en) | 1977-10-18 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MX3859E (en) | PROCEDURE FOR PREPARING METAL SALTS FROM CYCLOHEXANE | |
| AR213086A1 (en) | PROCEDURE FOR THE PREPARATION OF ACID DERIVATIVES 2- (PARA-SUBSTITUTED FENYL) -BENZOXAZOLE-5 OR 6-CARBOXYL, PHARMACEUTICALLY ACTIVE | |
| AR202799A1 (en) | A PROCEDURE FOR PREPARING DERIVATIVES OF 2- (1-PIPERAZINYL) 5,8-DIHYDRO-5-OXYPYRIDE <2,3-D> PYRIMIDIN-6-CARBOXYL ACID | |
| AR204003A1 (en) | PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM 2- (1-PIPERAZINYL) -5-OXOPYRIDE- (2,3-D) PYRIMIDINE-6-CARBOXYL ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS | |
| AR199510A1 (en) | PROCEDURE FOR PREPARING 7-ALPHA-AMINOACIL - 3 - HALO-CEPHALOSPORINS AND THEIR PHARMACEUTICALLY ACCEPTABLE ATONIC SALTS | |
| AR204175A1 (en) | PROCEDURE FOR THE PREPARATION OF 2- (3- (4-DIFENIMETHYL-1-PIPERAZINIL) -PROPYL) -S-TRIAZOL- (1,5-A) PYRIDINE AND ITS ACID ADDITION SALTS | |
| SE421313B (en) | PROCEDURE FOR PREPARING 2- (PHENOXIALKYLTIO) -5-NITROIMIDAZOLES | |
| AR204334A1 (en) | PROCEDURE FOR THE PREPARATION OF 1- (4- (ALKYLTIO-ALCOXY) -PHENOXY) -2-HYDROXY-3-ALKYL-AMINO-PROPAN COMPOUNDS | |
| AR202261A1 (en) | PROCEDURE FOR PREPARING DERIVATIVES OF 7-AMINO-3-MERCAPTOMETIL-CEPHALOSPORANIC ACID | |
| AR207751A1 (en) | PROCEDURE FOR PREPARING DERIVATIVES OF 16ALPHA ACID 17ALPHA -ETILENDIOXI-3,20-DIOXO-1,4-PREGNADIEN-21-OICO AND ITS SODIUM SALTS AND ALKYL ESTERS | |
| AR208068A1 (en) | A PROCEDURE FOR PREPARING DERIVATIVES OF 7-ACILAMIDO-3-HALO-CEFEM-4-CARBOXYL ACIDS, THE ESTERS AND THE PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF | |
| AR200042A1 (en) | PROCESS FOR THE PREPARATION OF LYSINE-CALCIUM CHLORIDE AND ITS PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS | |
| AR211844A1 (en) | PROCEDURE FOR PREPARING NEW DERIVATIVES OF 1,2,3,4 CYCLOHEXANOTEATROL ESTER TETRAACETATE AND ITS PHYSIOLOGICALLY ACCEPTABLE SALTS | |
| RO63034A (en) | PROCESS FOR THE PREPARATION OF 2- (5-NITRO-2-FURRYL) -THIENO- (2,3-D) -PYRIMIDINES DERIVATIVES | |
| AR202476A1 (en) | PROCEDURE FOR THE ELABORATION OF COMPOUNDS OF 2-HYDROXY-3-AMINO-PROPOXI-9,10-DIHIDROANTRACENE AND ITS SALTS | |
| DK137857B (en) | Analogous process for the preparation of 2-amino-1,5-benzodiazocine derivatives or pharmaceutically acceptable salts thereof. | |
| AR204577A1 (en) | PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 7-MESYLAMINO-PHENYLGLYCINAMIDE-3-SUBSTITUTED-3-CEFEM-4-CARBOXYL ACID | |
| MX4655E (en) | PROCEDURE FOR PREPARING ACID DERIVATIVES 3,3, '- TRIARILMETANODICARBOXILICO | |
| AR208282A1 (en) | PROCEDURE FOR PREPARING DERIVATIVES OF 2- (N-PHENYL - (- AMINOALKYL) -AMINOINDANE | |
| AR211381Q (en) | PROCEDURE FOR THE PRODUCTION OF SERICOSIDE (D-GLOCUPYRANOSIDE OF SERICICO ACID), SERICICO ACID AND ETHYLASINE-DIALKYLIC ACID, SALTS AND DERIVATIVES | |
| AR195903A1 (en) | PROCEDURE FOR PREPARING BIEOMYCINIC ACID 3-AMINOPROPYLESTER | |
| AR199285A1 (en) | PROCEDURE FOR PREPARING 1,4,6,9-TETRAHYDRO-4-6-DIOXOPYRIDE <3,2-G> QUINOLIN-2,8-DICARBOXYL ACID COMPOUNDS | |
| AR210248A1 (en) | PROCEDURE FOR PREPARING NEW DERIVATIVES OF-METHYL-3,4-DIHYDROXIFENYLALANINE AND ITS SALTS | |
| AR204250A1 (en) | PROCEDURE FOR PREPARING COMPOUNDS DERIVED FROM TRICHLOROACETAMIDO-6 PENICILANIC ACID-5-OXIDE | |
| AR224221A1 (en) | PROCEDURE FOR PREPARING ACID DERIVATIVES 2-O 3-CEFEM-3-CARBOXI-4-CARBOXILICOS AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS |