FI56011B - PROCEDURE FOR FRAMSTATING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5 8-DIHYDRO-5-OXOPYRIDO (2 3-D) -PYRIMIDIN-6-CARBOXYL - Google Patents

PROCEDURE FOR FRAMSTATING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5 8-DIHYDRO-5-OXOPYRIDO (2 3-D) -PYRIMIDIN-6-CARBOXYL

Info

Publication number
FI56011B
FI56011B FI298/74A FI29874A FI56011B FI 56011 B FI56011 B FI 56011B FI 298/74 A FI298/74 A FI 298/74A FI 29874 A FI29874 A FI 29874A FI 56011 B FI56011 B FI 56011B
Authority
FI
Finland
Prior art keywords
piperazinyl
framstating
oxopyrido
eller
pyrimidin
Prior art date
Application number
FI298/74A
Other languages
Finnish (fi)
Other versions
FI56011C (en
Inventor
Shinsaku Minami
Jun-Ichi Matsumoto
Kazuyo Kawaguchi
Shinsaku Mishio
Masanao Shimizu
Yoshiyuki Takase
Shinichi Nakamura
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Application granted granted Critical
Publication of FI56011B publication Critical patent/FI56011B/en
Publication of FI56011C publication Critical patent/FI56011C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI298/74A 1973-04-03 1974-02-04 PROCEDURE FOR FRAMSTAELLNING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5,8-DIHYDRO-5-OXOPYRIDO (2,3-D) -PYRIMIDIN-6- CARBOXYLSYROR FI56011C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (en) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (en) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (en) 1973-06-07 1973-06-07

Publications (2)

Publication Number Publication Date
FI56011B true FI56011B (en) 1979-07-31
FI56011C FI56011C (en) 1979-11-12

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
FI298/74A FI56011C (en) 1973-04-03 1974-02-04 PROCEDURE FOR FRAMSTAELLNING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5,8-DIHYDRO-5-OXOPYRIDO (2,3-D) -PYRIMIDIN-6- CARBOXYLSYROR

Country Status (11)

Country Link
AR (2) AR204003A1 (en)
AT (1) AT340931B (en)
CA (1) CA1066701A (en)
CH (1) CH593281A5 (en)
ES (1) ES424851A1 (en)
FI (1) FI56011C (en)
IE (1) IE39102B1 (en)
NL (1) NL186087C (en)
NO (1) NO142221C (en)
PH (2) PH10529A (en)
SE (1) SE416051B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (en) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara PROCEDURE FOR THE MANUFACTURE OF: 6-ALCOSSICARBONIL-8-ETHYL-5-OXO-5,8 DIIDRO-APERTA PAR. SQUARE 2,3-DCHIUSA PAR. SQUARE-PRIMIDINE 2-REPLACED AND ACID CORRESPONDING BOOKS.
AR077280A1 (en) 2009-06-29 2011-08-17 Incyte Corp PYRIMIDINONES AS PI3K INHIBITORS, AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
AR079529A1 (en) 2009-12-18 2012-02-01 Incyte Corp ARILO AND HETEROARILO DERIVATIVES REPLACED AND FOUNDED AS INHIBITORS OF THE PI3K
CA2822070C (en) 2010-12-20 2019-09-17 Incyte Corporation N-(1-(substituted-phenyl)ethyl)-9h-purin-6-amines as pi3k inhibitors
DK2751109T3 (en) 2011-09-02 2017-01-23 Incyte Holdings Corp HETEROCYCLYLAMINES AS PI3K INHIBITORS
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
TWI748941B (en) 2015-02-27 2021-12-11 美商英塞特公司 Salts and processes of preparing a pi3k inhibitor
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor

Also Published As

Publication number Publication date
FI56011C (en) 1979-11-12
PH10529A (en) 1977-05-30
CA1066701A (en) 1979-11-20
AR204003A1 (en) 1975-11-12
PH10984A (en) 1977-10-18
AT340931B (en) 1978-01-10
NL186087C (en) 1990-09-17
AR204660A1 (en) 1976-02-20
ES424851A1 (en) 1976-06-01
IE39102L (en) 1974-10-03
IE39102B1 (en) 1978-08-02
NO740349L (en) 1974-10-04
NL186087B (en) 1990-04-17
NL7401509A (en) 1974-10-07
SE416051B (en) 1980-11-24
NO142221C (en) 1980-07-16
NO142221B (en) 1980-04-08
CH593281A5 (en) 1977-11-30
ATA277774A (en) 1977-05-15

Similar Documents

Publication Publication Date Title
SE419981B (en) PROCEDURE FOR PREPARING 1ALFA-HYDROXY-VITAMIN D-DERIVATE
SE453667B (en) PROCEDURE FOR PREPARING POLYETERIMIDES
SE423536B (en) PROCEDURE FOR PREPARING MULTIPLE ALCOHOLS
SE423631B (en) PROCEDURE FOR THE PREPARATION OF OXALHYL DIALKYLXANTINES
SE422942B (en) ANALOGY PROCEDURE FOR PENICILLIN PREPARATION
SE7710599L (en) PROCEDURE FOR THE PREPARATION OF BENSISOXAZOLES
SE420720B (en) PROCEDURE FOR PREPARING 2,6-DISUBSTUDE PHENYLAMINOGUANIDE COMPOUNDS
AR199047A1 (en) PROCEDURE FOR SYNTHESIZING METHYL MERCAPTANE
FI56011B (en) PROCEDURE FOR FRAMSTATING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5 8-DIHYDRO-5-OXOPYRIDO (2 3-D) -PYRIMIDIN-6-CARBOXYL
SE411212B (en) PROCEDURE FOR THE PREPARATION OF 3-HALOGEN-CEPHALOSPORINE
SE415834B (en) ANALOGY PROCEDURE FOR PYRAZOLD DERIVATIVE PREPARATION
NO141649C (en) ANALOGY PROCEDURE FOR THE PREPARATION OF NEUROLEPTIC ACTIVE 7-FLUOROUS-SUBSTITUTED PHENOTIAZINES
NO146596C (en) PROCEDURE FOR THE PREPARATION OF 6-DEOXYTE TRACYCLINES
NO790627L (en) PROCEDURE FOR THE PREPARATION OF HYDROXYALKYLXANTINES
SE417601B (en) PROCEDURE FOR THE PREPARATION OF AMIDINOCARBAMIDS
SE405700B (en) PROCEDURE FOR PREHEAMING SHAPES
NO843825L (en) PROCEDURE FOR THE PREPARATION OF 6-DEOXYTHETRACYCLINE
SE421313B (en) PROCEDURE FOR PREPARING 2- (PHENOXIALKYLTIO) -5-NITROIMIDAZOLES
SE417319B (en) ANALOGY PROCEDURE FOR THE PREPARATION OF ERGOPEPTIN
SE421129B (en) PROCEDURE FOR PREPARING POLY-N-ALKYL IMINOALANES
SE420089B (en) ANALOGY PROCEDURE FOR THE PREPARATION OF PHENOXIPROPYLAMINE DERIVATIVES (ACETOPHENONES)
FI55498B (en) PROCEDURE FOR HYPOGLYCEMISIC PYRIDINKARBOXAMID-SULPHONYLUREAFOERENINGAR
SE411211B (en) PROCEDURE FOR THE PREPARATION OF 3-HALOGENCE PHALOSPORINS
SE409994B (en) PROCEDURE FOR THE PREPARATION OF AMIDINOCARBAMIDS
SE413895B (en) PROCEDURE FOR PREPARING 2-SUBSTITUTED ADENOSIN-5'-CARBOXYLATES