ATA277774A - PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT - Google Patents

PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT

Info

Publication number
ATA277774A
ATA277774A AT277774A AT277774A ATA277774A AT A277774 A ATA277774 A AT A277774A AT 277774 A AT277774 A AT 277774A AT 277774 A AT277774 A AT 277774A AT A277774 A ATA277774 A AT A277774A
Authority
AT
Austria
Prior art keywords
salt
production
piperazine derivatives
new piperazine
new
Prior art date
Application number
AT277774A
Other languages
German (de)
Other versions
AT340931B (en
Inventor
Shinsaku Minami
Junichi Matsumoto
Kazuyo Kawaguchi
Shinsaku Mishio
Masanao Shimizu
Yoshiyuki Takase
Shinichi Nakamura
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of ATA277774A publication Critical patent/ATA277774A/en
Application granted granted Critical
Publication of AT340931B publication Critical patent/AT340931B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT277774A 1973-04-03 1974-04-03 PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT AT340931B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (en) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (en) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (en) 1973-06-07 1973-06-07

Publications (2)

Publication Number Publication Date
ATA277774A true ATA277774A (en) 1977-05-15
AT340931B AT340931B (en) 1978-01-10

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
AT277774A AT340931B (en) 1973-04-03 1974-04-03 PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT

Country Status (11)

Country Link
AR (2) AR204003A1 (en)
AT (1) AT340931B (en)
CA (1) CA1066701A (en)
CH (1) CH593281A5 (en)
ES (1) ES424851A1 (en)
FI (1) FI56011C (en)
IE (1) IE39102B1 (en)
NL (1) NL186087C (en)
NO (1) NO142221C (en)
PH (2) PH10529A (en)
SE (1) SE416051B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (en) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara PROCEDURE FOR THE MANUFACTURE OF: 6-ALCOSSICARBONIL-8-ETHYL-5-OXO-5,8 DIIDRO-APERTA PAR. SQUARE 2,3-DCHIUSA PAR. SQUARE-PRIMIDINE 2-REPLACED AND ACID CORRESPONDING BOOKS.
JP5677425B2 (en) 2009-06-29 2015-02-25 インサイト・コーポレイションIncyte Corporation Pyrimidinone as a PI3K inhibitor
US8680108B2 (en) 2009-12-18 2014-03-25 Incyte Corporation Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors
WO2011075643A1 (en) 2009-12-18 2011-06-23 Incyte Corporation Substituted heteroaryl fused derivatives as pi3k inhibitors
EP2655374B1 (en) 2010-12-20 2019-10-23 Incyte Holdings Corporation N-(1-(substituted-phenyl)ethyl)-9h-purin-6-amines as pi3k inhibitors
KR102507287B1 (en) 2011-09-02 2023-03-07 인사이트 홀딩스 코포레이션 Heterocyclylamines as pi3k inhibitors
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
PE20180129A1 (en) 2015-02-27 2018-01-18 Incyte Corp PI3K INHIBITOR SALTS AND PREPARATION PROCESSES
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
US9732097B2 (en) 2015-05-11 2017-08-15 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor

Also Published As

Publication number Publication date
IE39102B1 (en) 1978-08-02
FI56011C (en) 1979-11-12
NL7401509A (en) 1974-10-07
CH593281A5 (en) 1977-11-30
NO142221B (en) 1980-04-08
NO740349L (en) 1974-10-04
SE416051B (en) 1980-11-24
AR204003A1 (en) 1975-11-12
CA1066701A (en) 1979-11-20
IE39102L (en) 1974-10-03
NO142221C (en) 1980-07-16
PH10984A (en) 1977-10-18
FI56011B (en) 1979-07-31
NL186087B (en) 1990-04-17
PH10529A (en) 1977-05-30
ES424851A1 (en) 1976-06-01
NL186087C (en) 1990-09-17
AT340931B (en) 1978-01-10
AR204660A1 (en) 1976-02-20

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Legal Events

Date Code Title Description
ELA Expired due to lapse of time