FI56011C - PROCEDURE FOR FRAMSTAELLNING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5,8-DIHYDRO-5-OXOPYRIDO (2,3-D) -PYRIMIDIN-6- CARBOXYLSYROR - Google Patents

PROCEDURE FOR FRAMSTAELLNING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5,8-DIHYDRO-5-OXOPYRIDO (2,3-D) -PYRIMIDIN-6- CARBOXYLSYROR

Info

Publication number
FI56011C
FI56011C FI298/74A FI29874A FI56011C FI 56011 C FI56011 C FI 56011C FI 298/74 A FI298/74 A FI 298/74A FI 29874 A FI29874 A FI 29874A FI 56011 C FI56011 C FI 56011C
Authority
FI
Finland
Prior art keywords
piperazinyl
carboxylsyror
oxopyrido
eller
framstaellning
Prior art date
Application number
FI298/74A
Other languages
Finnish (fi)
Other versions
FI56011B (en
Inventor
Shinsaku Minami
Jun-Ichi Matsumoto
Kazuyo Kawaguchi
Shinsaku Mishio
Masanao Shimizu
Yoshiyuki Takase
Shinichi Nakamura
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of FI56011B publication Critical patent/FI56011B/en
Application granted granted Critical
Publication of FI56011C publication Critical patent/FI56011C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI298/74A 1973-04-03 1974-02-04 PROCEDURE FOR FRAMSTAELLNING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5,8-DIHYDRO-5-OXOPYRIDO (2,3-D) -PYRIMIDIN-6- CARBOXYLSYROR FI56011C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (en) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (en) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (en) 1973-06-07 1973-06-07

Publications (2)

Publication Number Publication Date
FI56011B FI56011B (en) 1979-07-31
FI56011C true FI56011C (en) 1979-11-12

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
FI298/74A FI56011C (en) 1973-04-03 1974-02-04 PROCEDURE FOR FRAMSTAELLNING AV 2- (1-PIPERAZINYL) - ELLER 2- (4-ALKYL-1-PIPERAZINYL) -8-ETHYL-5,8-DIHYDRO-5-OXOPYRIDO (2,3-D) -PYRIMIDIN-6- CARBOXYLSYROR

Country Status (11)

Country Link
AR (2) AR204003A1 (en)
AT (1) AT340931B (en)
CA (1) CA1066701A (en)
CH (1) CH593281A5 (en)
ES (1) ES424851A1 (en)
FI (1) FI56011C (en)
IE (1) IE39102B1 (en)
NL (1) NL186087C (en)
NO (1) NO142221C (en)
PH (2) PH10529A (en)
SE (1) SE416051B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (en) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara PROCEDURE FOR THE MANUFACTURE OF: 6-ALCOSSICARBONIL-8-ETHYL-5-OXO-5,8 DIIDRO-APERTA PAR. SQUARE 2,3-DCHIUSA PAR. SQUARE-PRIMIDINE 2-REPLACED AND ACID CORRESPONDING BOOKS.
PE20120493A1 (en) 2009-06-29 2012-05-20 Incyte Corp PYRIMIDINONES AS PI3K INHIBITORS
US8680108B2 (en) 2009-12-18 2014-03-25 Incyte Corporation Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
AR084366A1 (en) 2010-12-20 2013-05-08 Incyte Corp N- (1- (REPLACED PHENYL) ETIL) -9H-PURIN-6-AMINAS AS PI3K INHIBITORS
KR101982475B1 (en) 2011-09-02 2019-05-27 인사이트 홀딩스 코포레이션 Heterocyclylamines as pi3k inhibitors
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
MY187502A (en) 2015-02-27 2021-09-24 Incyte Corp Salts of pi3k inhibitor and processes for their preparation
US9732097B2 (en) 2015-05-11 2017-08-15 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor

Also Published As

Publication number Publication date
PH10529A (en) 1977-05-30
AR204003A1 (en) 1975-11-12
PH10984A (en) 1977-10-18
CA1066701A (en) 1979-11-20
IE39102B1 (en) 1978-08-02
SE416051B (en) 1980-11-24
IE39102L (en) 1974-10-03
FI56011B (en) 1979-07-31
CH593281A5 (en) 1977-11-30
ATA277774A (en) 1977-05-15
NO142221C (en) 1980-07-16
NO142221B (en) 1980-04-08
NL186087C (en) 1990-09-17
NO740349L (en) 1974-10-04
ES424851A1 (en) 1976-06-01
AT340931B (en) 1978-01-10
AR204660A1 (en) 1976-02-20
NL186087B (en) 1990-04-17
NL7401509A (en) 1974-10-07

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