AR202224A1 - Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas - Google Patents

Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas

Info

Publication number
AR202224A1
AR202224A1 AR254832A AR25483274A AR202224A1 AR 202224 A1 AR202224 A1 AR 202224A1 AR 254832 A AR254832 A AR 254832A AR 25483274 A AR25483274 A AR 25483274A AR 202224 A1 AR202224 A1 AR 202224A1
Authority
AR
Argentina
Prior art keywords
onas
benzodiazepin
procedure
obtaining
Prior art date
Application number
AR254832A
Other languages
English (en)
Spanish (es)
Original Assignee
Crc Ricerca Chim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Crc Ricerca Chim filed Critical Crc Ricerca Chim
Application granted granted Critical
Publication of AR202224A1 publication Critical patent/AR202224A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/28Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AR254832A 1973-07-30 1974-07-22 Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas AR202224A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1105673A CH573928A5 (lt) 1973-07-30 1973-07-30

Publications (1)

Publication Number Publication Date
AR202224A1 true AR202224A1 (es) 1975-05-23

Family

ID=4369623

Family Applications (1)

Application Number Title Priority Date Filing Date
AR254832A AR202224A1 (es) 1973-07-30 1974-07-22 Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas

Country Status (21)

Country Link
US (1) US4010153A (lt)
JP (1) JPS5041886A (lt)
AR (1) AR202224A1 (lt)
AT (1) AT337192B (lt)
BE (1) BE818047A (lt)
CA (1) CA1021778A (lt)
CH (1) CH573928A5 (lt)
DE (1) DE2436744A1 (lt)
DK (1) DK138798B (lt)
ES (1) ES428675A1 (lt)
FI (1) FI227474A (lt)
FR (1) FR2239464B1 (lt)
GB (1) GB1481219A (lt)
HU (1) HU169180B (lt)
IE (1) IE39904B1 (lt)
IL (1) IL45289A (lt)
NL (1) NL7410256A (lt)
NO (1) NO137897C (lt)
SE (2) SE7409708L (lt)
SU (1) SU528872A3 (lt)
ZA (1) ZA744635B (lt)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4820834A (en) * 1984-06-26 1989-04-11 Merck & Co., Inc. Benzodiazepine analogs
CA1332410C (en) * 1984-06-26 1994-10-11 Roger M. Freidinger Benzodiazepine analogs
RS63653B1 (sr) 2015-07-22 2022-11-30 Enanta Pharm Inc Benzodiazepinski derivati kao inhibitori rsv
EP3402799B1 (en) 2016-01-15 2022-05-04 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
EP3582784B1 (en) 2017-02-16 2022-06-08 Enanta Pharmaceuticals, Inc. Processes for the preparation of benzodiazepine derivatives
US10752598B2 (en) 2017-06-07 2020-08-25 Enanta Pharmaceuticals, Inc. Aryldiazepine derivatives as RSV inhibitors
US10851115B2 (en) 2017-06-30 2020-12-01 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
WO2019006295A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
EP3687543B1 (en) 2017-09-29 2024-03-20 Enanta Pharmaceuticals, Inc. Combinations of pharmaceutical agents as rsv inhibitors
CN111343990B (zh) * 2017-11-13 2023-08-04 英安塔制药有限公司 苯并二氮杂䓬-2-酮和苯并氮杂䓬-2-酮衍生物的拆分方法
US10647711B2 (en) 2017-11-13 2020-05-12 Enanta Pharmaceuticals, Inc. Azepin-2-one derivatives as RSV inhibitors
WO2019199908A1 (en) 2018-04-11 2019-10-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
CA3133300A1 (en) 2019-03-18 2020-09-24 Enanta Pharmaceuticals, Inc. Benzodiazepine derivatives as rsv inhibitors
WO2020210246A1 (en) 2019-04-09 2020-10-15 Enanta Pharmaceuticals, Inc, Heterocyclic compounds as rsv inhibitors
US11505558B1 (en) 2019-10-04 2022-11-22 Enanta Pharmaceuticals, Inc. Antiviral heterocyclic compounds
UY39032A (es) 2020-01-24 2021-07-30 Enanta Pharm Inc Compuestos heterocíclicos como agentes antivirales
US11534439B2 (en) 2020-07-07 2022-12-27 Enanta Pharmaceuticals, Inc. Dihydroquinoxaline and dihydropyridopyrazine derivatives as RSV inhibitors
WO2022086840A1 (en) 2020-10-19 2022-04-28 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as anti-viral agents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3371085A (en) * 1959-12-10 1968-02-27 Hoffmann La Roche 5-aryl-3h-1,4-benzodiazepin-2(1h)-ones
JPS4426302Y1 (lt) * 1966-04-22 1969-11-05

Also Published As

Publication number Publication date
AT337192B (de) 1977-06-10
DK138798B (da) 1978-10-30
NO137897B (no) 1978-02-06
IL45289A (en) 1979-12-30
FR2239464A1 (lt) 1975-02-28
ZA744635B (en) 1975-08-27
SU528872A3 (ru) 1976-09-15
NL7410256A (nl) 1975-02-03
DE2436744A1 (de) 1975-02-27
FI227474A (lt) 1975-01-31
CA1021778A (en) 1977-11-29
SE7409708L (lt) 1975-01-31
GB1481219A (en) 1977-07-27
JPS5041886A (lt) 1975-04-16
IE39904L (en) 1975-01-30
CH573928A5 (lt) 1976-03-31
DK138798C (lt) 1979-04-09
ATA567674A (de) 1976-10-15
DK393274A (lt) 1975-04-01
IL45289A0 (en) 1974-10-22
FR2239464B1 (lt) 1978-04-14
IE39904B1 (en) 1979-01-31
NO742739L (lt) 1975-02-24
BE818047A (fr) 1974-11-18
US4010153A (en) 1977-03-01
HU169180B (lt) 1976-10-28
NO137897C (no) 1978-05-16
ES428675A1 (es) 1976-09-01
SE7510823L (sv) 1975-09-26

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