AR106049A1 - Formulaciones de liberación controlada - Google Patents
Formulaciones de liberación controladaInfo
- Publication number
- AR106049A1 AR106049A1 ARP160102828A ARP160102828A AR106049A1 AR 106049 A1 AR106049 A1 AR 106049A1 AR P160102828 A ARP160102828 A AR P160102828A AR P160102828 A ARP160102828 A AR P160102828A AR 106049 A1 AR106049 A1 AR 106049A1
- Authority
- AR
- Argentina
- Prior art keywords
- vomiting
- nausea
- compositions
- preformulation
- controlled release
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0021—Intradermal administration, e.g. through microneedle arrays, needleless injectors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/22—Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Abstract
La presente se refiere a una preformulación inyectable que comprende una mezcla de baja viscosidad de: a) al menos un lípido de diacilo neutro y/o al menos un tocoferol; b) al menos un fosfolípido; c) al menos un solvente orgánico que contiene oxígeno; d) al menos un antagonista de 5HT₃; en donde la preformulación forma, o es capaz de formar, al menos una estructura de fase cristalina líquida tras el contacto con un fluido acuoso. Tales composiciones pueden comprender, además, solventes polares y/o agentes activos adicionales, tales como agonistas y/o antagonistas de opioides. Se proporcionan métodos de tratamiento, en particular para el tratamiento de náuseas y vómitos tales como náuseas y vómitos posoperatorios y/o náuseas y vómitos inducidos por la terapia, así como los correspondientes usos de las composiciones. También se proporcionan dispositivos de administración que comprenden las formulaciones y kits que comprenden los dispositivos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB1516554.1A GB201516554D0 (en) | 2015-09-18 | 2015-09-18 | Controlled-release formulations |
Publications (1)
Publication Number | Publication Date |
---|---|
AR106049A1 true AR106049A1 (es) | 2017-12-06 |
Family
ID=54544453
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP160102828A AR106049A1 (es) | 2015-09-18 | 2016-09-16 | Formulaciones de liberación controlada |
Country Status (13)
Country | Link |
---|---|
US (1) | US20180256496A1 (es) |
EP (1) | EP3349800A1 (es) |
JP (1) | JP2018528964A (es) |
KR (1) | KR20180085716A (es) |
CN (1) | CN108601843A (es) |
AR (1) | AR106049A1 (es) |
AU (1) | AU2016323732A1 (es) |
CA (1) | CA2998966A1 (es) |
GB (1) | GB201516554D0 (es) |
HK (1) | HK1258718A1 (es) |
MX (1) | MX2018003333A (es) |
TW (1) | TW201717946A (es) |
WO (1) | WO2017046384A1 (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR102098980B1 (ko) | 2012-07-26 | 2020-04-08 | 카무러스 에이비 | 오피오이드 제형 |
CA3015557C (en) | 2014-11-07 | 2019-07-16 | Indivior Uk Limited | The use of sustained-release buprenorphine formulations for the treatment of pain or opioid use disorders |
BR112019011053A2 (pt) | 2016-12-07 | 2019-10-15 | Ra Pharmaceuticals Inc | moduladores da atividade do complemento |
US10646484B2 (en) | 2017-06-16 | 2020-05-12 | Indivior Uk Limited | Methods to treat opioid use disorder |
CA3116004A1 (en) * | 2018-10-11 | 2020-04-16 | Indivior Uk Limited | Buprenorphine to treat respiratory depression |
AU2020342591A1 (en) | 2019-09-02 | 2022-03-03 | Camurus Ab | Formulations and treatment methods |
WO2021064580A1 (en) * | 2019-10-01 | 2021-04-08 | Shilpa Medicare Limited | Controlled release injectable ondansetron formulations |
CN113081954A (zh) * | 2021-05-25 | 2021-07-09 | 南昌大学第二附属医院 | 一种凝胶载药贴剂药物输送系统 |
CN115702894A (zh) * | 2021-08-11 | 2023-02-17 | 朱信红 | 一种用于止吐的缓释组合物及其制备方法 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8332556D0 (en) * | 1983-12-06 | 1984-01-11 | Reckitt & Colmann Prod Ltd | Analgesic compositions |
GB0412530D0 (en) * | 2004-06-04 | 2004-07-07 | Camurus Ab | Formulation |
EP1768650B1 (en) * | 2004-06-04 | 2008-07-16 | Camurus Ab | Liquid depot formulations |
CA2594718C (en) * | 2005-01-14 | 2012-01-24 | Camurus Ab | Gnrh analogue formulations |
US9226918B2 (en) * | 2008-12-04 | 2016-01-05 | The Board Of Trustees Of The Leland Stanford Junior University | Methods and compositions for treating or preventing narcotic withdrawal symptoms |
SG11201402673YA (en) * | 2011-12-05 | 2014-06-27 | Camurus Ab | Robust controlled-release formulations |
KR102098980B1 (ko) * | 2012-07-26 | 2020-04-08 | 카무러스 에이비 | 오피오이드 제형 |
KR101586789B1 (ko) * | 2012-12-28 | 2016-01-19 | 주식회사 종근당 | 양이온성 약리학적 활성물질의 서방성 지질 초기제제 및 이를 포함하는 약제학적 조성물 |
US20140323517A1 (en) * | 2013-04-30 | 2014-10-30 | Heron Therapeutics, Inc. | Compositions and methods for injection of a biodegradable polymer-based delivery system |
-
2015
- 2015-09-18 GB GBGB1516554.1A patent/GB201516554D0/en not_active Ceased
-
2016
- 2016-09-14 TW TW105129955A patent/TW201717946A/zh unknown
- 2016-09-16 AU AU2016323732A patent/AU2016323732A1/en not_active Abandoned
- 2016-09-16 US US15/761,053 patent/US20180256496A1/en not_active Abandoned
- 2016-09-16 AR ARP160102828A patent/AR106049A1/es unknown
- 2016-09-16 CA CA2998966A patent/CA2998966A1/en not_active Abandoned
- 2016-09-16 CN CN201680060635.8A patent/CN108601843A/zh active Pending
- 2016-09-16 EP EP16766327.7A patent/EP3349800A1/en not_active Withdrawn
- 2016-09-16 WO PCT/EP2016/072059 patent/WO2017046384A1/en active Application Filing
- 2016-09-16 KR KR1020187010943A patent/KR20180085716A/ko unknown
- 2016-09-16 MX MX2018003333A patent/MX2018003333A/es unknown
- 2016-09-16 JP JP2018514400A patent/JP2018528964A/ja not_active Withdrawn
-
2019
- 2019-01-22 HK HK19101119.3A patent/HK1258718A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
MX2018003333A (es) | 2018-08-15 |
KR20180085716A (ko) | 2018-07-27 |
CN108601843A (zh) | 2018-09-28 |
TW201717946A (zh) | 2017-06-01 |
EP3349800A1 (en) | 2018-07-25 |
GB201516554D0 (en) | 2015-11-04 |
JP2018528964A (ja) | 2018-10-04 |
HK1258718A1 (zh) | 2019-11-15 |
US20180256496A1 (en) | 2018-09-13 |
WO2017046384A1 (en) | 2017-03-23 |
AU2016323732A1 (en) | 2018-04-12 |
CA2998966A1 (en) | 2017-03-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |