AR103317A1 - Moduladores de ciclopropil dihidrobenzofurano de receptores de melatonina - Google Patents

Moduladores de ciclopropil dihidrobenzofurano de receptores de melatonina

Info

Publication number
AR103317A1
AR103317A1 ARP150104335A ARP150104335A AR103317A1 AR 103317 A1 AR103317 A1 AR 103317A1 AR P150104335 A ARP150104335 A AR P150104335A AR P150104335 A ARP150104335 A AR P150104335A AR 103317 A1 AR103317 A1 AR 103317A1
Authority
AR
Argentina
Prior art keywords
cyclopropil
melatonine
dihydrobenzofuran
modulators
receptors
Prior art date
Application number
ARP150104335A
Other languages
English (en)
Original Assignee
Auspex Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Auspex Pharmaceuticals Inc filed Critical Auspex Pharmaceuticals Inc
Publication of AR103317A1 publication Critical patent/AR103317A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A01N43/12—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings condensed with a carbocyclic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system

Abstract

Reivindicación 1: Un compuesto caracterizado por la fórmula estructural (1) o una sal del mismo, en donde: R¹ - R¹⁹ se eligen independientemente de hidrógeno y deuterio; y al menos uno de R¹ - R¹⁹ es deuterio.
ARP150104335A 2014-12-29 2015-12-29 Moduladores de ciclopropil dihidrobenzofurano de receptores de melatonina AR103317A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201462097450P 2014-12-29 2014-12-29

Publications (1)

Publication Number Publication Date
AR103317A1 true AR103317A1 (es) 2017-05-03

Family

ID=56284951

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP150104335A AR103317A1 (es) 2014-12-29 2015-12-29 Moduladores de ciclopropil dihidrobenzofurano de receptores de melatonina

Country Status (3)

Country Link
AR (1) AR103317A1 (es)
TW (1) TW201629029A (es)
WO (1) WO2016109359A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107365288A (zh) * 2016-05-12 2017-11-21 浙江京新药业股份有限公司 他司美琼的晶型
CN108395370B (zh) * 2017-02-08 2021-04-06 中国石化扬子石油化工有限公司 一种氧化苯乙烯制备苯甲醛的方法
BR112020011189A2 (pt) 2017-12-05 2020-11-17 Sunovion Pharmaceuticals Inc. misturas não racêmicas e usos das mesmas
MX2020005517A (es) 2017-12-05 2020-11-09 Sunovion Pharmaceuticals Inc Formas cristalinas y metodos de produccion de las mismas.
CN108663460A (zh) * 2018-08-03 2018-10-16 安徽省金楠医疗科技有限公司 一种盐酸达泊西汀异构体检测方法
CN111362893B (zh) * 2018-12-25 2021-07-02 浙江京新药业股份有限公司 一种他司美琼中间体的制备方法
US11160758B2 (en) 2019-06-04 2021-11-02 Sunovion Pharmaceuticals Inc. Modified release formulations and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100130582A1 (en) * 2008-11-24 2010-05-27 Auspex Pharmaceuticals, Inc. Indolinone modulators of dopamine receptor
KR102317399B1 (ko) * 2012-01-26 2021-10-26 반다 파마슈티칼즈, 인코퍼레이티드. 일주기 리듬 장애의 치료
EP2884275A4 (en) * 2012-07-10 2016-04-13 Astellas Pharma Inc PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OR PREVENTION OF STRESS-RELATED HARNINE CONTINENCE OR MIXED INCONTINENCE AND METHOD FOR SCREENING COMPOUNDS FOR INTRODUCTION TO THIS PHARMACEUTICAL COMPOSITION

Also Published As

Publication number Publication date
WO2016109359A1 (en) 2016-07-07
TW201629029A (zh) 2016-08-16

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