AR086926A1 - Metodo de produccion de derivados de imidazol - Google Patents
Metodo de produccion de derivados de imidazolInfo
- Publication number
- AR086926A1 AR086926A1 ARP120102106A ARP120102106A AR086926A1 AR 086926 A1 AR086926 A1 AR 086926A1 AR P120102106 A ARP120102106 A AR P120102106A AR P120102106 A ARP120102106 A AR P120102106A AR 086926 A1 AR086926 A1 AR 086926A1
- Authority
- AR
- Argentina
- Prior art keywords
- formula
- compound
- compound represented
- alkyl group
- aryl group
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- RAXXELZNTBOGNW-UHFFFAOYSA-N 1H-imidazole Chemical class C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 12
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 125000003118 aryl group Chemical group 0.000 abstract 3
- ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical group [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 abstract 2
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 2
- 239000003153 chemical reaction reagent Substances 0.000 abstract 2
- 229910052740 iodine Inorganic materials 0.000 abstract 2
- 239000011777 magnesium Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000007818 Grignard reagent Substances 0.000 abstract 1
- WHXSMMKQMYFTQS-UHFFFAOYSA-N Lithium Chemical compound [Li] WHXSMMKQMYFTQS-UHFFFAOYSA-N 0.000 abstract 1
- FYYHWMGAXLPEAU-UHFFFAOYSA-N Magnesium Chemical compound [Mg] FYYHWMGAXLPEAU-UHFFFAOYSA-N 0.000 abstract 1
- 239000003098 androgen Substances 0.000 abstract 1
- 229940030486 androgens Drugs 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
- 229940011871 estrogen Drugs 0.000 abstract 1
- 150000004795 grignard reagents Chemical class 0.000 abstract 1
- 150000002460 imidazoles Chemical class 0.000 abstract 1
- 238000009776 industrial production Methods 0.000 abstract 1
- 229910052744 lithium Inorganic materials 0.000 abstract 1
- 229910052749 magnesium Inorganic materials 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2011133712 | 2011-06-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR086926A1 true AR086926A1 (es) | 2014-01-29 |
Family
ID=46458578
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP120102106A AR086926A1 (es) | 2011-06-15 | 2012-06-14 | Metodo de produccion de derivados de imidazol |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US9278938B2 (https=) |
| EP (1) | EP2721010B1 (https=) |
| JP (1) | JP6082353B2 (https=) |
| KR (1) | KR20140028069A (https=) |
| CN (1) | CN103608334B (https=) |
| AR (1) | AR086926A1 (https=) |
| AU (1) | AU2012270496A1 (https=) |
| BR (1) | BR112013030888A2 (https=) |
| CA (1) | CA2838971C (https=) |
| CL (1) | CL2013003492A1 (https=) |
| CO (1) | CO6852075A2 (https=) |
| CR (1) | CR20130655A (https=) |
| DO (1) | DOP2013000287A (https=) |
| EA (1) | EA201490019A1 (https=) |
| EC (1) | ECSP14013128A (https=) |
| ES (1) | ES2554454T3 (https=) |
| IL (1) | IL229566A0 (https=) |
| MA (1) | MA35809B1 (https=) |
| MX (1) | MX2013014009A (https=) |
| PE (1) | PE20141326A1 (https=) |
| PH (1) | PH12013502567A1 (https=) |
| SG (1) | SG195036A1 (https=) |
| TN (1) | TN2013000481A1 (https=) |
| TW (1) | TW201307295A (https=) |
| UY (1) | UY34130A (https=) |
| WO (1) | WO2012173280A1 (https=) |
| ZA (1) | ZA201308884B (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016054129A1 (en) * | 2014-09-30 | 2016-04-07 | Stc.Unm | Graphene-based inorganic-organic hybrid materials and separation of racemic mixtures |
| US20200033307A1 (en) * | 2018-07-25 | 2020-01-30 | Honeywell International Inc. | Method of determining an amount of water in a sample using a derivative of imidazole and a hydrogen halide donor |
| KR102253950B1 (ko) * | 2019-07-24 | 2021-05-20 | (주)에니켐텍 | 신규한 메데토미딘 제조방법 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5832880A (ja) * | 1981-08-24 | 1983-02-25 | Isukura Sangyo Kk | ハリントニンの部分合成方法 |
| WO2000078727A1 (en) | 1999-06-22 | 2000-12-28 | Takeda Chemical Industries, Ltd. | Process for the preparation of imidazole derivatives |
| PE20010781A1 (es) | 1999-10-22 | 2001-08-08 | Takeda Chemical Industries Ltd | Compuestos 1-(1h-imidazol-4-il)-1-(naftil-2-sustituido)etanol, su produccion y utilizacion |
| DE10031604A1 (de) | 2000-06-29 | 2002-01-17 | Consortium Elektrochem Ind | Verfahren zur Herstellung von beta-Hydroxy- und beta-Aminocarbonylverbindungen |
| PE20020596A1 (es) * | 2000-11-17 | 2002-08-13 | Takeda Chemical Industries Ltd | Derivados de imidazol, metodos de produccion e intermediarios del mismo |
| EP1463691B1 (en) | 2002-01-04 | 2006-06-14 | Koninklijke Philips Electronics N.V. | Sintered body and electric lamp |
| US7662974B2 (en) | 2002-01-10 | 2010-02-16 | Takeda Pharmaceutical Company Limited | Process for producing fused imidazole compound, reformatsky reagent in stable form, and process for producing the same |
| EP1394140A1 (de) * | 2002-08-14 | 2004-03-03 | Consortium für elektrochemische Industrie GmbH | Enantioselektives Reformatsky-Verfahren zur Herstellung von optisch aktiven Alkoholen, Aminen und deren Derivaten |
| EP2164409B1 (en) | 2007-06-29 | 2018-08-08 | Atheromed, Inc. | Atherectomy system |
-
2012
- 2012-06-14 JP JP2013549084A patent/JP6082353B2/ja not_active Expired - Fee Related
- 2012-06-14 EA EA201490019A patent/EA201490019A1/ru unknown
- 2012-06-14 PE PE2013002711A patent/PE20141326A1/es not_active Application Discontinuation
- 2012-06-14 WO PCT/JP2012/065795 patent/WO2012173280A1/en not_active Ceased
- 2012-06-14 CN CN201280029606.7A patent/CN103608334B/zh not_active Expired - Fee Related
- 2012-06-14 PH PH1/2013/502567A patent/PH12013502567A1/en unknown
- 2012-06-14 KR KR1020137032819A patent/KR20140028069A/ko not_active Withdrawn
- 2012-06-14 US US14/123,381 patent/US9278938B2/en not_active Expired - Fee Related
- 2012-06-14 CA CA2838971A patent/CA2838971C/en not_active Expired - Fee Related
- 2012-06-14 UY UY0001034130A patent/UY34130A/es not_active Application Discontinuation
- 2012-06-14 TW TW101121273A patent/TW201307295A/zh unknown
- 2012-06-14 EP EP12732719.5A patent/EP2721010B1/en active Active
- 2012-06-14 AR ARP120102106A patent/AR086926A1/es unknown
- 2012-06-14 SG SG2013085345A patent/SG195036A1/en unknown
- 2012-06-14 ES ES12732719.5T patent/ES2554454T3/es active Active
- 2012-06-14 MX MX2013014009A patent/MX2013014009A/es unknown
- 2012-06-14 AU AU2012270496A patent/AU2012270496A1/en not_active Abandoned
- 2012-06-14 BR BR112013030888A patent/BR112013030888A2/pt not_active IP Right Cessation
-
2013
- 2013-11-19 TN TNP2013000481A patent/TN2013000481A1/fr unknown
- 2013-11-21 IL IL229566A patent/IL229566A0/en unknown
- 2013-11-26 ZA ZA2013/08884A patent/ZA201308884B/en unknown
- 2013-12-05 CL CL2013003492A patent/CL2013003492A1/es unknown
- 2013-12-06 DO DO2013000287A patent/DOP2013000287A/es unknown
- 2013-12-13 CR CR20130655A patent/CR20130655A/es not_active Application Discontinuation
-
2014
- 2014-01-08 EC ECSP14013128 patent/ECSP14013128A/es unknown
- 2014-01-10 MA MA36668A patent/MA35809B1/fr unknown
- 2014-01-14 CO CO14006049A patent/CO6852075A2/es not_active Application Discontinuation
-
2016
- 2016-01-21 US US15/002,692 patent/US10005780B2/en not_active Expired - Fee Related
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |