MX2013014009A - Metodo de produccion de derivados de imidazol. - Google Patents

Metodo de produccion de derivados de imidazol.

Info

Publication number
MX2013014009A
MX2013014009A MX2013014009A MX2013014009A MX2013014009A MX 2013014009 A MX2013014009 A MX 2013014009A MX 2013014009 A MX2013014009 A MX 2013014009A MX 2013014009 A MX2013014009 A MX 2013014009A MX 2013014009 A MX2013014009 A MX 2013014009A
Authority
MX
Mexico
Prior art keywords
production method
compound
imidazole derivatives
reagent
reacting
Prior art date
Application number
MX2013014009A
Other languages
English (en)
Inventor
Yoichi Kawabata
Yasuhiro Sawai
Kazuaki Kanno
Naotaka Sawada
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46458578&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2013014009(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of MX2013014009A publication Critical patent/MX2013014009A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28—Antiandrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

La presente invención se refiere a un método de producción ventajoso de un derivado de imidazol, que es apropiado para la producción industrial. El compuesto (VI) se produce haciendo reaccionar el compuesto (I) con un reactivo de Grignard o un reactivo de magnesio y un reactivo de litio y luego haciendo reaccionar del compuesto resultante con el compuesto (V).
MX2013014009A 2011-06-15 2012-06-14 Metodo de produccion de derivados de imidazol. MX2013014009A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2011133712 2011-06-15
PCT/JP2012/065795 WO2012173280A1 (en) 2011-06-15 2012-06-14 Production method of imidazole derivatives

Publications (1)

Publication Number Publication Date
MX2013014009A true MX2013014009A (es) 2014-03-12

Family

ID=46458578

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013014009A MX2013014009A (es) 2011-06-15 2012-06-14 Metodo de produccion de derivados de imidazol.

Country Status (26)

Country Link
US (2) US9278938B2 (es)
EP (1) EP2721010B1 (es)
JP (1) JP6082353B2 (es)
KR (1) KR20140028069A (es)
CN (1) CN103608334B (es)
AR (1) AR086926A1 (es)
AU (1) AU2012270496A1 (es)
BR (1) BR112013030888A2 (es)
CA (1) CA2838971C (es)
CL (1) CL2013003492A1 (es)
CO (1) CO6852075A2 (es)
CR (1) CR20130655A (es)
DO (1) DOP2013000287A (es)
EA (1) EA201490019A1 (es)
EC (1) ECSP14013128A (es)
ES (1) ES2554454T3 (es)
IL (1) IL229566A0 (es)
MA (1) MA35809B1 (es)
MX (1) MX2013014009A (es)
PE (1) PE20141326A1 (es)
SG (1) SG195036A1 (es)
TN (1) TN2013000481A1 (es)
TW (1) TW201307295A (es)
UY (1) UY34130A (es)
WO (1) WO2012173280A1 (es)
ZA (1) ZA201308884B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016054129A1 (en) * 2014-09-30 2016-04-07 Stc.Unm Graphene-based inorganic-organic hybrid materials and separation of racemic mixtures
US20200033307A1 (en) * 2018-07-25 2020-01-30 Honeywell International Inc. Method of determining an amount of water in a sample using a derivative of imidazole and a hydrogen halide donor
KR102253950B1 (ko) * 2019-07-24 2021-05-20 (주)에니켐텍 신규한 메데토미딘 제조방법

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5832880A (ja) * 1981-08-24 1983-02-25 Isukura Sangyo Kk ハリントニンの部分合成方法
EP1193258A4 (en) 1999-06-22 2002-11-13 Takeda Chemical Industries Ltd PROCESS FOR THE PREPARATION OF IMIDAZOLE DERIVATIVES
PE20010781A1 (es) 1999-10-22 2001-08-08 Takeda Chemical Industries Ltd Compuestos 1-(1h-imidazol-4-il)-1-(naftil-2-sustituido)etanol, su produccion y utilizacion
DE10031604A1 (de) 2000-06-29 2002-01-17 Consortium Elektrochem Ind Verfahren zur Herstellung von beta-Hydroxy- und beta-Aminocarbonylverbindungen
AU2002214296C1 (en) 2000-11-17 2006-04-13 Takeda Pharmaceutical Company Limited Novel imidazole derivatives, production method thereof and use thereof
DE60212454T2 (de) 2002-01-04 2007-02-01 Koninklijke Philips Electronics N.V. Gesinterte formkörper und elektrische lampe
US7662974B2 (en) * 2002-01-10 2010-02-16 Takeda Pharmaceutical Company Limited Process for producing fused imidazole compound, reformatsky reagent in stable form, and process for producing the same
EP1394140A1 (de) * 2002-08-14 2004-03-03 Consortium für elektrochemische Industrie GmbH Enantioselektives Reformatsky-Verfahren zur Herstellung von optisch aktiven Alkoholen, Aminen und deren Derivaten
KR20100047854A (ko) 2007-06-29 2010-05-10 아테로메드, 아이엔씨. 죽종 절제 장치, 시스템 및 방법

Also Published As

Publication number Publication date
WO2012173280A1 (en) 2012-12-20
EP2721010B1 (en) 2015-09-09
TN2013000481A1 (en) 2015-03-30
US20140100373A1 (en) 2014-04-10
DOP2013000287A (es) 2014-02-16
CN103608334A (zh) 2014-02-26
SG195036A1 (en) 2013-12-30
CN103608334B (zh) 2015-12-23
US20160244454A1 (en) 2016-08-25
JP6082353B2 (ja) 2017-02-15
BR112013030888A2 (pt) 2017-03-21
MA35809B1 (fr) 2014-12-01
CL2013003492A1 (es) 2014-07-18
US10005780B2 (en) 2018-06-26
CA2838971C (en) 2019-07-30
JP2014520066A (ja) 2014-08-21
KR20140028069A (ko) 2014-03-07
US9278938B2 (en) 2016-03-08
ZA201308884B (en) 2015-02-25
EA201490019A1 (ru) 2014-04-30
AU2012270496A1 (en) 2013-12-19
ECSP14013128A (es) 2014-02-28
IL229566A0 (en) 2014-01-30
UY34130A (es) 2013-01-31
ES2554454T3 (es) 2015-12-21
PE20141326A1 (es) 2014-10-16
CO6852075A2 (es) 2014-01-30
EP2721010A1 (en) 2014-04-23
CR20130655A (es) 2014-03-03
AR086926A1 (es) 2014-01-29
CA2838971A1 (en) 2012-12-20
TW201307295A (zh) 2013-02-16

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