AR086803A1 - Derivados de oxazetidinas, composiciones farmaceuticas y cosmeticas que los contienen y uso de los mismos para tratar enfermedades dermatologicas fundamentalmente, y del aparato respiratorio, digestivo y cardiovascular, entre otras - Google Patents

Derivados de oxazetidinas, composiciones farmaceuticas y cosmeticas que los contienen y uso de los mismos para tratar enfermedades dermatologicas fundamentalmente, y del aparato respiratorio, digestivo y cardiovascular, entre otras

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Publication number
AR086803A1
AR086803A1 ARP120102343A ARP120102343A AR086803A1 AR 086803 A1 AR086803 A1 AR 086803A1 AR P120102343 A ARP120102343 A AR P120102343A AR P120102343 A ARP120102343 A AR P120102343A AR 086803 A1 AR086803 A1 AR 086803A1
Authority
AR
Argentina
Prior art keywords
pharmaceutical
oxazetidines
digestive
cardiovascular
respiratory
Prior art date
Application number
ARP120102343A
Other languages
English (en)
Inventor
Bouix-Peter Claire
Original Assignee
Galderma Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Galderma Res & Dev filed Critical Galderma Res & Dev
Publication of AR086803A1 publication Critical patent/AR086803A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
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    • A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
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Abstract

La presente se refiere al campo farmacéutico, en particular, al tratamiento de patologías de hipopigmentación y dermatosis fotosensibles. Más específicamente, la presente se refiere a compuestos que son agonistas del receptor MC1R y que exhiben una menor toxicidad con respecto a otros compuestos de la misma clase. Reivindicación 1: Compuesto de la fórmula general (1), en la cual: R¹ representa un grupo ciclopropilmetilo o un grupo 4-hidroxibutilo; R² representa un átomo de hidrógeno o un grupo metilo; y también las sales y enantiómeros de los compuestos de fórmula general (1) correspondientes.
ARP120102343A 2011-06-30 2012-06-29 Derivados de oxazetidinas, composiciones farmaceuticas y cosmeticas que los contienen y uso de los mismos para tratar enfermedades dermatologicas fundamentalmente, y del aparato respiratorio, digestivo y cardiovascular, entre otras AR086803A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161503068P 2011-06-30 2011-06-30
FR1159911A FR2981933B1 (fr) 2011-11-02 2011-11-02 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique

Publications (1)

Publication Number Publication Date
AR086803A1 true AR086803A1 (es) 2014-01-22

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
ARP120102343A AR086803A1 (es) 2011-06-30 2012-06-29 Derivados de oxazetidinas, composiciones farmaceuticas y cosmeticas que los contienen y uso de los mismos para tratar enfermedades dermatologicas fundamentalmente, y del aparato respiratorio, digestivo y cardiovascular, entre otras

Country Status (14)

Country Link
US (2) US9353083B2 (es)
EP (1) EP2726478B1 (es)
JP (1) JP5898310B2 (es)
KR (1) KR101946085B1 (es)
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CA3233305A1 (en) 2019-02-19 2020-08-27 Gilead Sciences, Inc. Solid forms of fxr agonists
WO2021251452A1 (ja) * 2020-06-10 2021-12-16 田辺三菱製薬株式会社 光線性皮膚疾患の予防又は治療剤

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EP2726478A1 (en) 2014-05-07
AU2012277838B2 (en) 2017-04-13
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MX2014000170A (es) 2014-02-19
US20140228342A1 (en) 2014-08-14
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IN2014CN00711A (es) 2015-04-03
CA2840606A1 (en) 2013-01-03
EP2726478B1 (en) 2017-01-11
JP2014518238A (ja) 2014-07-28
KR101946085B1 (ko) 2019-02-08
ES2620476T3 (es) 2017-06-28
CN103827106A (zh) 2014-05-28

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