BR112013033861A2 - composto, uso de um composto, composição farmacêutica, composição cosmética e uso cosmético de uma composição - Google Patents

composto, uso de um composto, composição farmacêutica, composição cosmética e uso cosmético de uma composição

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Publication number
BR112013033861A2
BR112013033861A2 BR112013033861A BR112013033861A BR112013033861A2 BR 112013033861 A2 BR112013033861 A2 BR 112013033861A2 BR 112013033861 A BR112013033861 A BR 112013033861A BR 112013033861 A BR112013033861 A BR 112013033861A BR 112013033861 A2 BR112013033861 A2 BR 112013033861A2
Authority
BR
Brazil
Prior art keywords
composition
compound
cosmetic
pharmaceutical composition
pharmaceutical
Prior art date
Application number
BR112013033861A
Other languages
English (en)
Other versions
BR112013033861B1 (pt
Inventor
Bouix-Peter Clarie
Original Assignee
Galderma Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Galderma Res & Dev filed Critical Galderma Res & Dev
Publication of BR112013033861A2 publication Critical patent/BR112013033861A2/pt
Publication of BR112013033861B1 publication Critical patent/BR112013033861B1/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
    • A61K8/4946—Imidazoles or their condensed derivatives, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
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BR112013033861-0A 2011-06-30 2012-06-28 Compostos agonistas do receptor de mc1r, usos de ditos compostos, composição farmacêutica, composição cosmética e usos cosméticos de compostos agonistas do receptor de mc1r BR112013033861B1 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161503068P 2011-06-30 2011-06-30
US61/503,068 2011-06-30
FR1159911A FR2981933B1 (fr) 2011-11-02 2011-11-02 Derives d'oxoazetidine, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique
FR1159911 2011-11-02
PCT/EP2012/062622 WO2013001030A1 (en) 2011-06-30 2012-06-28 Oxazetidine derivatives, process for preparing them and use thereof in human medicine and in cosmetics

Publications (2)

Publication Number Publication Date
BR112013033861A2 true BR112013033861A2 (pt) 2017-12-19
BR112013033861B1 BR112013033861B1 (pt) 2021-11-09

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BR112013033861-0A BR112013033861B1 (pt) 2011-06-30 2012-06-28 Compostos agonistas do receptor de mc1r, usos de ditos compostos, composição farmacêutica, composição cosmética e usos cosméticos de compostos agonistas do receptor de mc1r

Country Status (14)

Country Link
US (2) US9353083B2 (pt)
EP (1) EP2726478B1 (pt)
JP (1) JP5898310B2 (pt)
KR (1) KR101946085B1 (pt)
AR (1) AR086803A1 (pt)
AU (1) AU2012277838B2 (pt)
BR (1) BR112013033861B1 (pt)
CA (1) CA2840606A1 (pt)
ES (1) ES2620476T3 (pt)
FR (1) FR2981933B1 (pt)
IN (1) IN2014CN00711A (pt)
MX (1) MX2014000170A (pt)
RU (1) RU2624011C2 (pt)
WO (1) WO2013001030A1 (pt)

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EP2825187A1 (en) * 2012-03-15 2015-01-21 Galderma Research & Development Combination of a mc1r receptor agonist and uvb for the treatment and/or prevention of pigmentation disorders
CA2968836A1 (en) 2016-06-13 2017-12-13 Gilead Sciences, Inc. Fxr (nr1h4) modulating compounds
CA3050630A1 (en) * 2017-02-01 2018-08-09 Clinuvel Pharmaceuticals Ltd Alpha-msh analogues used in the treatment of xeroderma pigmentosum
AU2018243719B2 (en) 2017-03-28 2021-01-21 Gilead Sciences, Inc. Therapeutic combinations for treating liver diseases
CA3233305A1 (en) 2019-02-19 2020-08-27 Gilead Sciences, Inc. Solid forms of fxr agonists
WO2021251452A1 (ja) * 2020-06-10 2021-12-16 田辺三菱製薬株式会社 光線性皮膚疾患の予防又は治療剤

Family Cites Families (5)

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MY128261A (en) * 1992-10-27 2007-01-31 Merck Sharp & Dohme New substituted azetidinones as anti-inflammatory and antidegenerative agents
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FR2981933A1 (fr) 2013-05-03
US9353083B2 (en) 2016-05-31
WO2013001030A1 (en) 2013-01-03
EP2726478A1 (en) 2014-05-07
AU2012277838B2 (en) 2017-04-13
JP5898310B2 (ja) 2016-04-06
AU2012277838A1 (en) 2014-01-23
KR20140050019A (ko) 2014-04-28
MX2014000170A (es) 2014-02-19
US20140228342A1 (en) 2014-08-14
US20160237065A1 (en) 2016-08-18
FR2981933B1 (fr) 2013-11-15
RU2624011C2 (ru) 2017-06-30
US9981952B2 (en) 2018-05-29
RU2014102966A (ru) 2015-08-10
IN2014CN00711A (pt) 2015-04-03
CA2840606A1 (en) 2013-01-03
EP2726478B1 (en) 2017-01-11
JP2014518238A (ja) 2014-07-28
AR086803A1 (es) 2014-01-22
KR101946085B1 (ko) 2019-02-08
ES2620476T3 (es) 2017-06-28
CN103827106A (zh) 2014-05-28

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