AR085989A2 - Composiciones endoparasiticidas y proceso para su preparacion - Google Patents
Composiciones endoparasiticidas y proceso para su preparacionInfo
- Publication number
- AR085989A2 AR085989A2 ARP120101244A ARP120101244A AR085989A2 AR 085989 A2 AR085989 A2 AR 085989A2 AR P120101244 A ARP120101244 A AR P120101244A AR P120101244 A ARP120101244 A AR P120101244A AR 085989 A2 AR085989 A2 AR 085989A2
- Authority
- AR
- Argentina
- Prior art keywords
- composition according
- preparation
- cyclodepsipeptide
- morpholinyl
- compositions
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
- A61K9/0017—Non-human animal skin, e.g. pour-on, spot-on
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/22—Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
Abstract
Composiciones endoparasiticidas, aplicables de manera tópica, que contienen depsipéptidos cíclicos y de cadena abierta, constituidos por aminoácidos y ácidos hidroxicarboxílicos como componentes y que contienen de 6 hasta 30 átomos en el anillo o en la cadena, a su preparación y a su empleo como endoparasiticidas.Reivindicación 1: Composición adecuada para la administración tópica en animales caracterizada porque que comprende un ciclodepsipeptido de la fórmula (1), donde Z representa N-morfolinilo, amino, mono- o dimetilamino, solo o en combinación con otros compuestos activos, y 1,2-isopropiliden glicerina. Reivindicación 2: Composición de acuerdo con la reivindicación 1, caracterizada porque comprende el ciclodepsipeptido donde ambos radicales Z representan N-morfolinilo. Reivindicación 3: Composición de acuerdo con la reivindicación 1 ó 2, caracterizada porque adicionalmente comprende alcohol bencilico y/o propilen glicol diacetato. Reivindicación 5: Composición de acuerdo con cualquiera de las reivindicaciones precedentes, caracterizada porque comprende Praziquantel como compuesto activo adicional.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10008128A DE10008128A1 (de) | 2000-02-22 | 2000-02-22 | Endoparasitizide Mittel |
Publications (1)
Publication Number | Publication Date |
---|---|
AR085989A2 true AR085989A2 (es) | 2013-11-13 |
Family
ID=7631886
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP010100751A AR028218A1 (es) | 2000-02-22 | 2001-02-20 | Composicion endoparasiticidas |
ARP120101244A AR085989A2 (es) | 2000-02-22 | 2012-04-11 | Composiciones endoparasiticidas y proceso para su preparacion |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP010100751A AR028218A1 (es) | 2000-02-22 | 2001-02-20 | Composicion endoparasiticidas |
Country Status (25)
Country | Link |
---|---|
US (1) | US20030125244A1 (es) |
EP (1) | EP1259250B1 (es) |
JP (2) | JP5596249B2 (es) |
KR (1) | KR100755414B1 (es) |
CN (1) | CN1309415C (es) |
AR (2) | AR028218A1 (es) |
AT (1) | ATE343394T1 (es) |
AU (2) | AU2001240605B2 (es) |
BR (1) | BR0108562B1 (es) |
CA (1) | CA2400610C (es) |
CZ (1) | CZ300242B6 (es) |
DE (2) | DE10008128A1 (es) |
DK (1) | DK1259250T3 (es) |
ES (1) | ES2274871T3 (es) |
HK (1) | HK1054326B (es) |
HU (1) | HUP0204554A3 (es) |
IL (2) | IL150988A0 (es) |
MX (1) | MXPA02008210A (es) |
NO (1) | NO328949B1 (es) |
NZ (1) | NZ520856A (es) |
PL (1) | PL203999B1 (es) |
PT (1) | PT1259250E (es) |
RU (1) | RU2292905C2 (es) |
WO (1) | WO2001062268A1 (es) |
ZA (1) | ZA200205982B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10104362A1 (de) * | 2001-02-01 | 2002-08-08 | Bayer Ag | Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit |
US7541336B2 (en) * | 2002-11-12 | 2009-06-02 | The Kitasato Institute | Substance fki-1033 and process for producing the same |
DE10358525A1 (de) | 2003-12-13 | 2005-07-07 | Bayer Healthcare Ag | Endoparasitizide Mittel zur topischen Applikation |
DE102005011779A1 (de) * | 2005-03-11 | 2006-09-14 | Bayer Healthcare Ag | Endoparasitizide Mittel |
CN102149717B (zh) | 2008-08-28 | 2014-05-14 | 辉瑞大药厂 | 二氧杂-双环[3.2.1]辛烷-2,3,4-三醇衍生物 |
DE102009012423A1 (de) | 2009-03-10 | 2010-09-16 | Bayer Animal Health Gmbh | Zubereitung auf Ölbasis |
BR112017024773A2 (pt) | 2015-05-20 | 2018-11-06 | Merial, Inc. | compostos depsipeptídeos anti-helmínticos |
JP6943859B2 (ja) | 2015-12-28 | 2021-10-06 | ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド | 駆虫性デプシペプチド化合物 |
MX2019005628A (es) | 2016-11-16 | 2019-12-18 | Boehringer Ingelheim Animal Health Usa Inc | Compuestos depsipeptidos antihelminticos. |
US20220331314A1 (en) | 2019-08-14 | 2022-10-20 | Vetoquinol Sa | Compositions comprising tigolaner for controlling parasites |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3531545A1 (de) * | 1985-09-04 | 1987-03-05 | Goedecke Ag | Arzneimittel mit einem gehalt an calcium-antagonisten und deren verwendung |
DE3705227A1 (de) * | 1987-02-19 | 1988-09-01 | Bayer Ag | Anthelminthische wirkstoffkombinationen |
AU669883B2 (en) * | 1992-03-17 | 1996-06-27 | Astellas Pharma Inc. | Depsipeptide derivative, production thereof and use thereof |
DE4317458A1 (de) * | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
DE4309830C1 (de) * | 1993-03-26 | 1994-05-05 | Lohmann Therapie Syst Lts | Wirkstoffpflaster für die Abgabe von Estradiol an die Haut |
DE4317432A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4317457A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4400464A1 (de) * | 1994-01-11 | 1995-07-13 | Bayer Ag | Endoparasitizide Mittel |
WO1995021624A1 (fr) * | 1994-02-08 | 1995-08-17 | Nippon Kayaku Kabushiki Kaisha | Preparation sous forme de solution a base d'une forte concentration d'aureobasidine |
DE4417742A1 (de) * | 1994-05-20 | 1995-11-23 | Bayer Ag | Nicht-systemische Bekämpfung von Parasiten |
DE19520275A1 (de) * | 1995-06-02 | 1996-12-05 | Bayer Ag | Endoparasitizide Mittel |
DE19545044A1 (de) * | 1995-12-02 | 1997-06-05 | Bayer Ag | Endoparasitizide Mittel |
GB9803448D0 (en) * | 1998-02-18 | 1998-04-15 | Pharma Mar Sa | Pharmaceutical formulation |
ATE295167T1 (de) * | 1998-03-19 | 2005-05-15 | Merck & Co Inc | Schwefelpentafluorophenylpyrazole zur kontrolle von ektoparasitenbefall |
FR2776191B1 (fr) * | 1998-03-23 | 2002-05-31 | Theramex | Composition hormonale topique a effet systemique |
DE19921887A1 (de) * | 1999-05-12 | 2000-11-16 | Bayer Ag | Endoparasitizide Mittel |
-
2000
- 2000-02-22 DE DE10008128A patent/DE10008128A1/de not_active Withdrawn
-
2001
- 2001-02-09 CN CNB018054005A patent/CN1309415C/zh not_active Expired - Lifetime
- 2001-02-09 RU RU2002125493/15A patent/RU2292905C2/ru not_active IP Right Cessation
- 2001-02-09 AU AU2001240605A patent/AU2001240605B2/en not_active Expired
- 2001-02-09 JP JP2001561333A patent/JP5596249B2/ja not_active Expired - Lifetime
- 2001-02-09 DK DK01911623T patent/DK1259250T3/da active
- 2001-02-09 DE DE50111315T patent/DE50111315D1/de not_active Expired - Lifetime
- 2001-02-09 CZ CZ20022867A patent/CZ300242B6/cs not_active IP Right Cessation
- 2001-02-09 CA CA2400610A patent/CA2400610C/en not_active Expired - Lifetime
- 2001-02-09 PT PT01911623T patent/PT1259250E/pt unknown
- 2001-02-09 NZ NZ520856A patent/NZ520856A/en not_active IP Right Cessation
- 2001-02-09 WO PCT/EP2001/001392 patent/WO2001062268A1/de active IP Right Grant
- 2001-02-09 MX MXPA02008210A patent/MXPA02008210A/es active IP Right Grant
- 2001-02-09 BR BRPI0108562-0A patent/BR0108562B1/pt not_active IP Right Cessation
- 2001-02-09 ES ES01911623T patent/ES2274871T3/es not_active Expired - Lifetime
- 2001-02-09 US US10/204,880 patent/US20030125244A1/en not_active Abandoned
- 2001-02-09 EP EP01911623A patent/EP1259250B1/de not_active Expired - Lifetime
- 2001-02-09 AU AU4060501A patent/AU4060501A/xx active Pending
- 2001-02-09 AT AT01911623T patent/ATE343394T1/de active
- 2001-02-09 IL IL15098801A patent/IL150988A0/xx unknown
- 2001-02-09 HU HU0204554A patent/HUP0204554A3/hu unknown
- 2001-02-09 PL PL357551A patent/PL203999B1/pl unknown
- 2001-02-09 KR KR1020027010032A patent/KR100755414B1/ko active IP Right Grant
- 2001-02-20 AR ARP010100751A patent/AR028218A1/es active IP Right Grant
-
2002
- 2002-07-26 ZA ZA200205982A patent/ZA200205982B/xx unknown
- 2002-07-30 IL IL150988A patent/IL150988A/en active IP Right Grant
- 2002-08-21 NO NO20023976A patent/NO328949B1/no not_active IP Right Cessation
-
2003
- 2003-09-11 HK HK03106540.9A patent/HK1054326B/zh unknown
-
2012
- 2012-01-16 JP JP2012006256A patent/JP2012107024A/ja active Pending
- 2012-04-11 AR ARP120101244A patent/AR085989A2/es unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |