AR071956A1 - Derivados de isoindolina, utiles en terapia del dolor - Google Patents
Derivados de isoindolina, utiles en terapia del dolorInfo
- Publication number
- AR071956A1 AR071956A1 ARP090101938A ARP090101938A AR071956A1 AR 071956 A1 AR071956 A1 AR 071956A1 AR P090101938 A ARP090101938 A AR P090101938A AR P090101938 A ARP090101938 A AR P090101938A AR 071956 A1 AR071956 A1 AR 071956A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- alkoxy
- optionally substituted
- fluoro
- r4nr5
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5731908P | 2008-05-30 | 2008-05-30 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR071956A1 true AR071956A1 (es) | 2010-07-28 |
Family
ID=41377344
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090101938A AR071956A1 (es) | 2008-05-30 | 2009-05-29 | Derivados de isoindolina, utiles en terapia del dolor |
Country Status (6)
Country | Link |
---|---|
AR (1) | AR071956A1 (zh) |
CL (1) | CL2009001330A1 (zh) |
PE (1) | PE20091947A1 (zh) |
TW (1) | TW201000447A (zh) |
UY (1) | UY31853A (zh) |
WO (1) | WO2009145719A1 (zh) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013007768A1 (en) | 2011-07-13 | 2013-01-17 | F. Hoffmann-La Roche Ag | Tricyclic heterocyclic compounds, compositions and methods of use thereof as jak inhibitors |
WO2015102929A1 (en) * | 2013-12-30 | 2015-07-09 | Novartis Ag | Tricyclic sulfonamide derivatives |
US11046683B2 (en) | 2016-12-15 | 2021-06-29 | Ono Pharmaceutical Co., Ltd. | Activator of TREK (TWIK RElated K+ channels) channels |
US20220289763A1 (en) | 2019-07-22 | 2022-09-15 | Lupin Limited | Macrocyclic Compounds as Sting Agonists and Methods and Uses Thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200613272A (en) * | 2004-08-13 | 2006-05-01 | Astrazeneca Ab | Isoindolone compounds and their use as metabotropic glutamate receptor potentiators |
TW200804281A (en) * | 2006-02-16 | 2008-01-16 | Astrazeneca Ab | New metabotropic glutamate receptor-potentiating isoindolones |
WO2008008020A1 (en) * | 2006-07-12 | 2008-01-17 | Astrazeneca Ab | 3-oxoisoindoline-1-carboxamide derivatives as analgesic agents |
TW200812962A (en) * | 2006-07-12 | 2008-03-16 | Astrazeneca Ab | New compounds I/418 |
GB0705882D0 (en) * | 2007-03-27 | 2007-05-02 | Glaxo Group Ltd | Novel compounds |
-
2009
- 2009-05-26 TW TW098117512A patent/TW201000447A/zh unknown
- 2009-05-29 AR ARP090101938A patent/AR071956A1/es unknown
- 2009-05-29 PE PE2009000755A patent/PE20091947A1/es not_active Application Discontinuation
- 2009-05-29 WO PCT/SE2009/050616 patent/WO2009145719A1/en active Application Filing
- 2009-05-29 CL CL2009001330A patent/CL2009001330A1/es unknown
- 2009-05-29 UY UY0001031853A patent/UY31853A/es unknown
Also Published As
Publication number | Publication date |
---|---|
WO2009145719A1 (en) | 2009-12-03 |
UY31853A (es) | 2010-01-05 |
CL2009001330A1 (es) | 2010-01-15 |
TW201000447A (en) | 2010-01-01 |
PE20091947A1 (es) | 2010-01-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR107377A2 (es) | Compuestos derivados de tetrahidroquinolina | |
AR108256A2 (es) | Un método para el control de nematodos parásitos de plantas | |
AR079401A1 (es) | Cianobutiratos sustituidos con accion herbicida | |
AR049894A1 (es) | Derivados de prolina y sus usos como inhibodores de la enzima dipeptidilpeptidasa-iv | |
PE20090904A1 (es) | ARILOXAZOLES SUSTITUIDOS COMO LIGANDOS DE LOS RECEPTORES DE ADENOSINA A1 Y/O A2b | |
AR055150A1 (es) | Compuestos de isoindol - imido y composiciones que los comprenden y sus metodos de uso | |
AR060604A1 (es) | Nuevos arilamino n- heteroarilos como inhibidores de mek | |
AR085615A1 (es) | Derivados de fluoropiridinona utiles como agentes antibacterianos y composiciones farmaceuticas que los contienen | |
CO6160323A2 (es) | Derivados de quinazolinona 5-sustituidos como agentes antitumorales | |
PE20160844A1 (es) | Compuestos triciclicos como agentes anticancerigenos | |
AR072952A1 (es) | Compuestos de 2-imino-3-metilpirrolopirimidinona fenilo-sustituida como inhibidores de bace-1, composiciones y su uso | |
PE20090511A1 (es) | Imidazopiridinonas | |
DOP2010000046A (es) | Compuestos de biciclolactama sustituida | |
PE20120693A1 (es) | Compuestos heterociclos como moduladores de la piruvato cinasa m2 (pkm2) | |
CO6150164A2 (es) | Derivados de 2-metilmorfolina pirido-,pirazo-ypirimido-pirimidina como inhibidores de mtor | |
PE20061439A1 (es) | DERIVADOS DE 2-AMIDO-6-AMINO-8-OXO-PURINA COMO MODULADORES DEL RECEPTOR Toll (TLR) | |
AR054790A1 (es) | Metodos para el tratamiento de disfuncion sexual | |
AR069480A1 (es) | Derivados de 2-amino-pirimidina | |
CR11245A (es) | Mejoras en compuestos organicos o relacionadas con los mismos | |
HN2005000239A (es) | Derivados de tetrahidroisoquinolilsulfonamidas, su preparacion y su utilizacion en terapeutica | |
PE20091090A1 (es) | Derivados de piperidina como agonistas de receptores muscarinicos | |
PE20100718A1 (es) | Derivados triciclicos de 1, 4-dihidropiridina [b, e]-condensados como inhibidores de aurora quinasas | |
AR064424A1 (es) | Derivados sustituidos de 1-oxo-ftalazinas y 1-oxo-pirido-piridazinas,composiciones farmaceuticas que los contienen y usos para prevenir y/o tratar enfermedades inflamatorias y alergicas del tracto respiratorio. | |
AR082075A1 (es) | Derivados de dioxima eter microbicidas | |
AR069813A1 (es) | Derivados de 2- amino-pirimidina, una composicion farmaceutica, un metodo de preparacion del compuesto y uso del mismo para preparar un medicamento |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |