AR063708A1 - Derivados de isoserina, un proceso para su preparacion y su empleo en la produccion de un medicamento para el tratamiento o profilaxis de enfermedades mediadas por la inhibicion del factor ixa de la coagulacion sanguinea. - Google Patents

Derivados de isoserina, un proceso para su preparacion y su empleo en la produccion de un medicamento para el tratamiento o profilaxis de enfermedades mediadas por la inhibicion del factor ixa de la coagulacion sanguinea.

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Publication number
AR063708A1
AR063708A1 ARP070104012A ARP070104012A AR063708A1 AR 063708 A1 AR063708 A1 AR 063708A1 AR P070104012 A ARP070104012 A AR P070104012A AR P070104012 A ARP070104012 A AR P070104012A AR 063708 A1 AR063708 A1 AR 063708A1
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AR
Argentina
Prior art keywords
trisubstituted
mono
aryl
het
substituted
Prior art date
Application number
ARP070104012A
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English (en)
Spanish (es)
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Sanofi Aventis
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Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of AR063708A1 publication Critical patent/AR063708A1/es

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    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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ARP070104012A 2006-09-13 2007-09-11 Derivados de isoserina, un proceso para su preparacion y su empleo en la produccion de un medicamento para el tratamiento o profilaxis de enfermedades mediadas por la inhibicion del factor ixa de la coagulacion sanguinea. AR063708A1 (es)

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WO2006084033A1 (en) 2005-02-03 2006-08-10 Signum Biosciences, Inc. Compositions and methods for enhancing cognitive function
US7923041B2 (en) 2005-02-03 2011-04-12 Signum Biosciences, Inc. Compositions and methods for enhancing cognitive function
EP2049543B1 (en) * 2006-09-07 2014-11-05 Callaghan Innovation Research Limited Acyclic amine inhibitors of 5'-methylthioadenosine phosphorylase and nucleosidase
WO2009132051A1 (en) 2008-04-21 2009-10-29 Signum Biosciences, Inc. Compounds, compositions and methods for making the same
AU2009322342A1 (en) 2008-12-05 2011-06-30 Merck Sharp & Dohme Corp. Morpholinone compounds as factor IXa inhibitors
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AU2007297013A1 (en) 2008-03-20
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