AR060974A1 - Compuesto de 4-piridinona, su uso para la preparacion de un medicamento, composicion farmaceutica que lo comprende, proceso para su preparacion y proceso para la preparacion de un compuesto intermediario de utilidad en el anterior - Google Patents
Compuesto de 4-piridinona, su uso para la preparacion de un medicamento, composicion farmaceutica que lo comprende, proceso para su preparacion y proceso para la preparacion de un compuesto intermediario de utilidad en el anteriorInfo
- Publication number
- AR060974A1 AR060974A1 ARP070102297A ARP070102297A AR060974A1 AR 060974 A1 AR060974 A1 AR 060974A1 AR P070102297 A ARP070102297 A AR P070102297A AR P070102297 A ARP070102297 A AR P070102297A AR 060974 A1 AR060974 A1 AR 060974A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- pharmaceutical composition
- piridinone
- composite
- medicinal product
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 4
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000002131 composite material Substances 0.000 title 1
- 229940126601 medicinal product Drugs 0.000 title 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 2
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
- -1 4-pyridinone compound Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 201000004792 malaria Diseases 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/68—One oxygen atom attached in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06381025A EP1862459A1 (en) | 2006-05-31 | 2006-05-31 | Novel heterocyclic compounds |
| EP07380072A EP1967515A1 (en) | 2007-03-08 | 2007-03-08 | Heterocyclic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR060974A1 true AR060974A1 (es) | 2008-07-23 |
Family
ID=38480438
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP070102297A AR060974A1 (es) | 2006-05-31 | 2007-05-29 | Compuesto de 4-piridinona, su uso para la preparacion de un medicamento, composicion farmaceutica que lo comprende, proceso para su preparacion y proceso para la preparacion de un compuesto intermediario de utilidad en el anterior |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US7674808B2 (enExample) |
| EP (1) | EP2024332A1 (enExample) |
| JP (1) | JP2009538873A (enExample) |
| KR (1) | KR20090012342A (enExample) |
| AR (1) | AR060974A1 (enExample) |
| AU (1) | AU2007267093A1 (enExample) |
| BR (1) | BRPI0711783A2 (enExample) |
| CA (1) | CA2653872A1 (enExample) |
| CR (1) | CR10492A (enExample) |
| EA (1) | EA200870545A1 (enExample) |
| IL (1) | IL195158A0 (enExample) |
| MA (1) | MA30487B1 (enExample) |
| MX (1) | MX2008015291A (enExample) |
| NO (1) | NO20085087L (enExample) |
| PE (1) | PE20080453A1 (enExample) |
| TW (1) | TW200817331A (enExample) |
| WO (1) | WO2007138048A1 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050158294A1 (en) | 2003-12-19 | 2005-07-21 | The Procter & Gamble Company | Canine probiotic Bifidobacteria pseudolongum |
| US8877178B2 (en) | 2003-12-19 | 2014-11-04 | The Iams Company | Methods of use of probiotic bifidobacteria for companion animals |
| WO2006130187A1 (en) | 2005-05-31 | 2006-12-07 | The Iams Company | Feline probiotic lactobacilli |
| JP4938006B2 (ja) | 2005-05-31 | 2012-05-23 | ザ・アイムス・カンパニー | ネコ科動物プロバイオティク・ビフィドバクテリア |
| RU2436581C2 (ru) | 2007-02-01 | 2011-12-20 | Дзе Иамс Компани | Способ уменьшения воспаления и снижения стресса у млекопитающего |
| EP2220043A1 (en) * | 2007-11-30 | 2010-08-25 | Glaxo Group Limited | Crystalline form of an antimalarial compound |
| US9771199B2 (en) * | 2008-07-07 | 2017-09-26 | Mars, Incorporated | Probiotic supplement, process for making, and packaging |
| US9232813B2 (en) * | 2008-07-07 | 2016-01-12 | The Iams Company | Probiotic supplement, process for making, and packaging |
| WO2010081904A1 (en) | 2009-01-19 | 2010-07-22 | Glaxo Group Limited | 4 ( 1h) -pyridinone derivatives and their use as antimalaria agents |
| EP2246329A1 (en) | 2009-01-19 | 2010-11-03 | Glaxo Group Limited | 4(1H)-pyridinone derivatives and their use as antimalaria agents |
| TW201039834A (en) | 2009-02-20 | 2010-11-16 | Glaxo Group Ltd | Novel heterocyclic compounds |
| WO2010142741A1 (en) * | 2009-06-12 | 2010-12-16 | Glaxo Group Limited | Phenylpyridylpyridones for use as antimalarial agents |
| US10104903B2 (en) | 2009-07-31 | 2018-10-23 | Mars, Incorporated | Animal food and its appearance |
| US10206677B2 (en) * | 2014-09-26 | 2019-02-19 | Ethicon Llc | Surgical staple and driver arrangements for staple cartridges |
| JOP20180072A1 (ar) | 2014-09-11 | 2019-01-30 | Lilly Co Eli | علاج الأعراض المرتبطة بالعلاج بالحرمان من الأندروجين |
| WO2016169908A1 (en) * | 2015-04-21 | 2016-10-27 | Glaxosmithkline Intellectual Property Development Limited | Uracil derivatives for the treatment of malaria |
| GB201809627D0 (en) * | 2018-06-12 | 2018-07-25 | Biorelevant Com Ltd | Methods for preparing buffer solutions suitable for in vitro drug dissolution testing, drug solubility testing and/or drug profiling |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9005518D0 (en) * | 1990-03-12 | 1990-05-09 | Wellcome Found | Heterocyclic compounds |
| US5403934A (en) * | 1990-03-12 | 1995-04-04 | Burroughs Wellcome Co. | Heterocyclic compounds |
| GB9100465D0 (en) * | 1991-01-09 | 1991-02-20 | Hider Robert C | Pharmaceutical compositions |
-
2007
- 2007-05-29 MX MX2008015291A patent/MX2008015291A/es unknown
- 2007-05-29 EA EA200870545A patent/EA200870545A1/ru unknown
- 2007-05-29 PE PE2007000667A patent/PE20080453A1/es not_active Application Discontinuation
- 2007-05-29 WO PCT/EP2007/055188 patent/WO2007138048A1/en not_active Ceased
- 2007-05-29 JP JP2009512577A patent/JP2009538873A/ja active Pending
- 2007-05-29 KR KR1020087029153A patent/KR20090012342A/ko not_active Withdrawn
- 2007-05-29 AU AU2007267093A patent/AU2007267093A1/en not_active Abandoned
- 2007-05-29 EP EP07729610A patent/EP2024332A1/en not_active Withdrawn
- 2007-05-29 US US11/754,382 patent/US7674808B2/en not_active Expired - Fee Related
- 2007-05-29 CA CA002653872A patent/CA2653872A1/en not_active Abandoned
- 2007-05-29 AR ARP070102297A patent/AR060974A1/es not_active Application Discontinuation
- 2007-05-29 BR BRPI0711783-3A patent/BRPI0711783A2/pt not_active IP Right Cessation
- 2007-05-29 TW TW096119056A patent/TW200817331A/zh unknown
- 2007-05-31 US US11/755,849 patent/US7629365B2/en not_active Expired - Fee Related
-
2008
- 2008-11-06 IL IL195158A patent/IL195158A0/en unknown
- 2008-12-01 MA MA31430A patent/MA30487B1/fr unknown
- 2008-12-05 NO NO20085087A patent/NO20085087L/no not_active Application Discontinuation
- 2008-12-10 CR CR10492A patent/CR10492A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007138048A1 (en) | 2007-12-06 |
| EP2024332A1 (en) | 2009-02-18 |
| TW200817331A (en) | 2008-04-16 |
| US20080021073A1 (en) | 2008-01-24 |
| BRPI0711783A2 (pt) | 2011-11-29 |
| NO20085087L (no) | 2009-02-20 |
| AU2007267093A1 (en) | 2007-12-06 |
| CA2653872A1 (en) | 2007-12-06 |
| US7629365B2 (en) | 2009-12-08 |
| US7674808B2 (en) | 2010-03-09 |
| US20070281977A1 (en) | 2007-12-06 |
| PE20080453A1 (es) | 2008-05-29 |
| EA200870545A1 (ru) | 2009-12-30 |
| JP2009538873A (ja) | 2009-11-12 |
| CR10492A (es) | 2009-01-27 |
| MX2008015291A (es) | 2008-12-12 |
| IL195158A0 (en) | 2009-08-03 |
| KR20090012342A (ko) | 2009-02-03 |
| MA30487B1 (fr) | 2009-06-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |