AR059327A1 - Monohidrato de rimonabant su procedimiento de preparacion y composiciones farmaceuticas que lo contienen - Google Patents

Monohidrato de rimonabant su procedimiento de preparacion y composiciones farmaceuticas que lo contienen

Info

Publication number
AR059327A1
AR059327A1 ARP070100477A ARP070100477A AR059327A1 AR 059327 A1 AR059327 A1 AR 059327A1 AR P070100477 A ARP070100477 A AR P070100477A AR P070100477 A ARP070100477 A AR P070100477A AR 059327 A1 AR059327 A1 AR 059327A1
Authority
AR
Argentina
Prior art keywords
rimonabant
monohidrate
pharmaceutical compositions
compositions containing
preparation procedure
Prior art date
Application number
ARP070100477A
Other languages
English (en)
Inventor
Olivier Monnier
Baptiste Fours
Helene Duplaa
Philippe Ochsenbein
Gerard Coquerel
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37075667&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR059327(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of AR059327A1 publication Critical patent/AR059327A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Reivindicacion 2: La forma cristalina del monohidrato de rimonabant segun la reivindicacion 1, caracterizada por un pico de fusion entre 95°C+- 5°C y 115°C+- 5°C.
ARP070100477A 2006-02-08 2007-02-06 Monohidrato de rimonabant su procedimiento de preparacion y composiciones farmaceuticas que lo contienen AR059327A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0601253A FR2897060B1 (fr) 2006-02-08 2006-02-08 Le monohydrate de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant

Publications (1)

Publication Number Publication Date
AR059327A1 true AR059327A1 (es) 2008-03-26

Family

ID=37075667

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070100477A AR059327A1 (es) 2006-02-08 2007-02-06 Monohidrato de rimonabant su procedimiento de preparacion y composiciones farmaceuticas que lo contienen

Country Status (20)

Country Link
US (1) US20090048449A1 (es)
EP (1) EP1984341A1 (es)
JP (1) JP2009526025A (es)
KR (1) KR20080093042A (es)
CN (1) CN101405271A (es)
AR (1) AR059327A1 (es)
AU (1) AU2007213649A1 (es)
BR (1) BRPI0707711A2 (es)
CA (1) CA2641494A1 (es)
DO (1) DOP2007000023A (es)
EA (1) EA200870236A1 (es)
FR (1) FR2897060B1 (es)
GT (1) GT200700014A (es)
IL (1) IL192963A0 (es)
MA (1) MA30312B1 (es)
NO (1) NO20083521L (es)
TW (1) TW200804343A (es)
UY (1) UY30137A1 (es)
WO (1) WO2007090949A1 (es)
ZA (1) ZA200806713B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2057144A4 (en) * 2006-09-01 2010-06-02 Hetero Drugs Ltd NEW POLYMORPHIC FROM RIMONABANT
WO2008056377A2 (en) * 2006-11-06 2008-05-15 Cadila Healthcare Limited Polymorphic forms of rimonabant
MX2017007426A (es) * 2014-12-08 2018-04-20 Crystal Pharmatech Co Ltd Formas cristalinas de complejo supramolecular trisodico que comprende valsartan y ahu-377 y metodos de las mismas.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
JP4746931B2 (ja) * 2005-07-22 2011-08-10 株式会社日立製作所 フラットディスプレイパネルモジュール及びフラットディスプレイ装置
EP2057144A4 (en) * 2006-09-01 2010-06-02 Hetero Drugs Ltd NEW POLYMORPHIC FROM RIMONABANT
WO2008035023A1 (en) * 2006-09-19 2008-03-27 Cipla Limited Polymorphs of rimonabant

Also Published As

Publication number Publication date
FR2897060B1 (fr) 2008-07-25
EP1984341A1 (fr) 2008-10-29
GT200700014A (es) 2007-09-19
EA200870236A1 (ru) 2009-02-27
NO20083521L (no) 2008-10-24
IL192963A0 (en) 2009-02-11
WO2007090949A1 (fr) 2007-08-16
MA30312B1 (fr) 2009-04-01
ZA200806713B (en) 2009-10-28
UY30137A1 (es) 2007-09-28
DOP2007000023A (es) 2008-02-15
US20090048449A1 (en) 2009-02-19
AU2007213649A1 (en) 2007-08-16
CA2641494A1 (fr) 2007-08-16
JP2009526025A (ja) 2009-07-16
CN101405271A (zh) 2009-04-08
KR20080093042A (ko) 2008-10-17
TW200804343A (en) 2008-01-16
FR2897060A1 (fr) 2007-08-10
BRPI0707711A2 (pt) 2011-05-10

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