AR052054A1 - Procesos para la preparacion de derivados del acido 3-fenil-2-arilalquilpropionico - Google Patents

Procesos para la preparacion de derivados del acido 3-fenil-2-arilalquilpropionico

Info

Publication number
AR052054A1
AR052054A1 ARP050105310A ARP050105310A AR052054A1 AR 052054 A1 AR052054 A1 AR 052054A1 AR P050105310 A ARP050105310 A AR P050105310A AR P050105310 A ARP050105310 A AR P050105310A AR 052054 A1 AR052054 A1 AR 052054A1
Authority
AR
Argentina
Prior art keywords
processes
preparation
arilalquilpropionico
fenil
acid derivatives
Prior art date
Application number
ARP050105310A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AR052054A1 publication Critical patent/AR052054A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P41/00Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P11/00Preparation of sulfur-containing organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P41/00Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture
    • C12P41/003Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by ester formation, lactone formation or the inverse reactions
    • C12P41/005Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by ester formation, lactone formation or the inverse reactions by esterification of carboxylic acid groups in the enantiomers or the inverse reaction
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P7/00Preparation of oxygen-containing organic compounds
    • C12P7/40Preparation of oxygen-containing organic compounds containing a carboxyl group including Peroxycarboxylic acids
    • C12P7/52Propionic acid; Butyric acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Microbiology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Analytical Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se describen procesos enzimáticos y químicos para la preparacion de ciertos derivados de ácido 3-fenil-2-arilalquiltiopropionico que tienen utilidad en el tratamiento de afecciones clínicas que incluyen trastornos lipídicos (dislipidemias), asociados o no con resistencia a insulina, y otras manifestaciones del síndrome metabolico; y además, ciertos nuevos intermediarios utilizados en estos procesos.
ARP050105310A 2004-12-16 2005-12-16 Procesos para la preparacion de derivados del acido 3-fenil-2-arilalquilpropionico AR052054A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0427524.4A GB0427524D0 (en) 2004-12-16 2004-12-16 Chemical process

Publications (1)

Publication Number Publication Date
AR052054A1 true AR052054A1 (es) 2007-02-28

Family

ID=34090119

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050105310A AR052054A1 (es) 2004-12-16 2005-12-16 Procesos para la preparacion de derivados del acido 3-fenil-2-arilalquilpropionico

Country Status (17)

Country Link
US (1) US7803586B2 (es)
EP (1) EP1828394A2 (es)
JP (1) JP2008523797A (es)
KR (1) KR20070094908A (es)
CN (1) CN101080495A (es)
AR (1) AR052054A1 (es)
AU (1) AU2005315454A1 (es)
BR (1) BRPI0518948A2 (es)
CA (1) CA2588591A1 (es)
GB (1) GB0427524D0 (es)
IL (1) IL183524A0 (es)
MX (1) MX2007007219A (es)
NO (1) NO20072633L (es)
SA (1) SA05260405A (es)
TW (1) TW200636071A (es)
UY (1) UY29271A1 (es)
WO (1) WO2006064213A2 (es)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001011072A1 (en) 1999-08-05 2001-02-15 Novo Nordisk A/S Process for the preparation of substituted 3-phenyl-propanoic acid esters and substituted 3-phenyl-propanoic acids
JP2003506065A (ja) * 1999-08-05 2003-02-18 ノボ ノルディスク アクティーゼルスカブ 置換された3−フェニル−プロパン酸エステル及び置換された3−フェニル−プロパン酸の調製の方法
SE0104333D0 (sv) * 2001-12-19 2001-12-19 Astrazeneca Ab Therapeutic agents
GB0314130D0 (en) 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
GB0314075D0 (en) 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
GB0314131D0 (en) 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
GB0314260D0 (en) 2003-06-19 2003-07-23 Astrazeneca Ab Therapeutic agents

Also Published As

Publication number Publication date
WO2006064213A2 (en) 2006-06-22
TW200636071A (en) 2006-10-16
AU2005315454A1 (en) 2006-06-22
EP1828394A2 (en) 2007-09-05
IL183524A0 (en) 2007-09-20
WO2006064213A3 (en) 2006-08-24
UY29271A1 (es) 2006-07-31
CN101080495A (zh) 2007-11-28
SA05260405A (ar) 2005-12-03
NO20072633L (no) 2007-06-21
BRPI0518948A2 (pt) 2008-12-16
US7803586B2 (en) 2010-09-28
US20080115247A1 (en) 2008-05-15
GB0427524D0 (en) 2005-01-19
MX2007007219A (es) 2007-08-14
CA2588591A1 (en) 2006-06-22
JP2008523797A (ja) 2008-07-10
KR20070094908A (ko) 2007-09-27

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal