AR048068A1 - Piperazinas derivadas de urea para el tratamiento de endometriosis - Google Patents

Piperazinas derivadas de urea para el tratamiento de endometriosis

Info

Publication number
AR048068A1
AR048068A1 ARP050100664A ARP050100664A AR048068A1 AR 048068 A1 AR048068 A1 AR 048068A1 AR P050100664 A ARP050100664 A AR P050100664A AR P050100664 A ARP050100664 A AR P050100664A AR 048068 A1 AR048068 A1 AR 048068A1
Authority
AR
Argentina
Prior art keywords
treatment
piperazinas
endometriosis
urea
derived
Prior art date
Application number
ARP050100664A
Other languages
English (en)
Inventor
Ulrike Kaufman
Richard Horuk
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of AR048068A1 publication Critical patent/AR048068A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Uso de un compuesto de la siguiente formula (1a); para la produccion de un medicamento para el tratamiento de la endometrosis en seres humanos. El tratamiento comprende administrar a un humano de sexo femenino que necesita dicho tratamiento una cantidad eficaz de términos terapéuticos de dicho compuesto.
ARP050100664A 2004-02-24 2005-02-24 Piperazinas derivadas de urea para el tratamiento de endometriosis AR048068A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04090065 2004-02-24

Publications (1)

Publication Number Publication Date
AR048068A1 true AR048068A1 (es) 2006-03-29

Family

ID=34878280

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050100664A AR048068A1 (es) 2004-02-24 2005-02-24 Piperazinas derivadas de urea para el tratamiento de endometriosis

Country Status (21)

Country Link
US (1) US20080119471A1 (es)
EP (1) EP1727526A2 (es)
JP (1) JP2007523126A (es)
KR (1) KR20070033961A (es)
CN (1) CN101090723A (es)
AR (1) AR048068A1 (es)
AU (1) AU2005215156A1 (es)
BR (1) BRPI0507985A (es)
CA (1) CA2556423A1 (es)
CR (1) CR8584A (es)
EA (1) EA200601514A1 (es)
EC (1) ECSP066836A (es)
GT (1) GT200500032A (es)
IL (1) IL177406A0 (es)
NO (1) NO20064298L (es)
PA (1) PA8624501A1 (es)
PE (1) PE20051129A1 (es)
SV (1) SV2006002017A (es)
TW (1) TW200539882A (es)
WO (1) WO2005079769A2 (es)
ZA (1) ZA200607970B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CL2007001829A1 (es) * 2006-06-23 2008-01-25 Smithkline Beecham Corp P-toluensulfonato de n-[4-cloro-2-hidroxi-3-(piperazina-1-sulfonil)fenil]-n-(2-cloro-3-fluorofenil)urea;procedimiento de preparacion;composicion farmaceutica;combinacion farmaceutica;y uso en el tratamiento de una enfermedad mediada por la quiimioquina il-8, tales como asma y epoc.
US8445674B2 (en) * 2009-10-21 2013-05-21 Hoffmann-La Roche Inc Heterocyclyl compounds
HUE040420T2 (hu) 2010-03-11 2019-03-28 Univ New York Amidvegyületek, mint RORyT modulátorok és felhasználásuk
PL3022202T3 (pl) 2013-07-18 2019-10-31 Novartis Ag Inhibitory autotaksyny zawierające heteroaromatyczny rdzeń pierścienia benzylowego - cyklicznego amidu

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6207665B1 (en) * 1997-06-12 2001-03-27 Schering Aktiengesellschaft Piperazine derivatives and their use as anti-inflammatory agents
CA2489560A1 (en) * 2002-06-27 2004-01-08 Schering Aktiengesellschaft Substituted quinoline ccr5 receptor antagonists

Also Published As

Publication number Publication date
EA200601514A1 (ru) 2007-02-27
ECSP066836A (es) 2006-11-24
SV2006002017A (es) 2006-05-09
NO20064298L (no) 2006-11-24
CA2556423A1 (en) 2005-09-01
BRPI0507985A (pt) 2007-05-08
WO2005079769A3 (en) 2007-01-04
GT200500032A (es) 2005-10-31
US20080119471A1 (en) 2008-05-22
JP2007523126A (ja) 2007-08-16
ZA200607970B (en) 2008-12-31
CR8584A (es) 2007-08-28
PA8624501A1 (es) 2006-07-03
TW200539882A (en) 2005-12-16
AU2005215156A1 (en) 2005-09-01
PE20051129A1 (es) 2006-02-16
IL177406A0 (en) 2006-12-10
KR20070033961A (ko) 2007-03-27
EP1727526A2 (en) 2006-12-06
CN101090723A (zh) 2007-12-19
WO2005079769A2 (en) 2005-09-01

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