BRPI0507985A - derivados de piperazina uréia para o tratamento de endometriose - Google Patents

derivados de piperazina uréia para o tratamento de endometriose

Info

Publication number
BRPI0507985A
BRPI0507985A BRPI0507985-3A BRPI0507985A BRPI0507985A BR PI0507985 A BRPI0507985 A BR PI0507985A BR PI0507985 A BRPI0507985 A BR PI0507985A BR PI0507985 A BRPI0507985 A BR PI0507985A
Authority
BR
Brazil
Prior art keywords
treatment
endometriosis
urea derivatives
piperazine urea
piperazine
Prior art date
Application number
BRPI0507985-3A
Other languages
English (en)
Inventor
Richard Horuk
Ulrike Kaufmann
Original Assignee
Schering Aktiengellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Aktiengellschaft filed Critical Schering Aktiengellschaft
Publication of BRPI0507985A publication Critical patent/BRPI0507985A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

DERIVADOS DE PIPERAZINA URéIA PARA O TRATAMENTO DE ENDOMETRIOSE. para a produção de um medicamento para o tratamento de endometriose no ser humano, onde o tratamento compreende administrar a uma mulher com necessidade tal tratamento uma quantidade terapeuticamente eficaz do referido composto.
BRPI0507985-3A 2004-02-24 2005-02-23 derivados de piperazina uréia para o tratamento de endometriose BRPI0507985A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04090065 2004-02-24
PCT/EP2005/002036 WO2005079769A2 (en) 2004-02-24 2005-02-23 Piperazine derivatives for the treatment of endometriosis

Publications (1)

Publication Number Publication Date
BRPI0507985A true BRPI0507985A (pt) 2007-05-08

Family

ID=34878280

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507985-3A BRPI0507985A (pt) 2004-02-24 2005-02-23 derivados de piperazina uréia para o tratamento de endometriose

Country Status (21)

Country Link
US (1) US20080119471A1 (pt)
EP (1) EP1727526A2 (pt)
JP (1) JP2007523126A (pt)
KR (1) KR20070033961A (pt)
CN (1) CN101090723A (pt)
AR (1) AR048068A1 (pt)
AU (1) AU2005215156A1 (pt)
BR (1) BRPI0507985A (pt)
CA (1) CA2556423A1 (pt)
CR (1) CR8584A (pt)
EA (1) EA200601514A1 (pt)
EC (1) ECSP066836A (pt)
GT (1) GT200500032A (pt)
IL (1) IL177406A0 (pt)
NO (1) NO20064298L (pt)
PA (1) PA8624501A1 (pt)
PE (1) PE20051129A1 (pt)
SV (1) SV2006002017A (pt)
TW (1) TW200539882A (pt)
WO (1) WO2005079769A2 (pt)
ZA (1) ZA200607970B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CL2007001829A1 (es) * 2006-06-23 2008-01-25 Smithkline Beecham Corp P-toluensulfonato de n-[4-cloro-2-hidroxi-3-(piperazina-1-sulfonil)fenil]-n-(2-cloro-3-fluorofenil)urea;procedimiento de preparacion;composicion farmaceutica;combinacion farmaceutica;y uso en el tratamiento de una enfermedad mediada por la quiimioquina il-8, tales como asma y epoc.
US8445674B2 (en) * 2009-10-21 2013-05-21 Hoffmann-La Roche Inc Heterocyclyl compounds
HUE040420T2 (hu) 2010-03-11 2019-03-28 Univ New York Amidvegyületek, mint RORyT modulátorok és felhasználásuk
PL3022202T3 (pl) 2013-07-18 2019-10-31 Novartis Ag Inhibitory autotaksyny zawierające heteroaromatyczny rdzeń pierścienia benzylowego - cyklicznego amidu

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6207665B1 (en) * 1997-06-12 2001-03-27 Schering Aktiengesellschaft Piperazine derivatives and their use as anti-inflammatory agents
CA2489560A1 (en) * 2002-06-27 2004-01-08 Schering Aktiengesellschaft Substituted quinoline ccr5 receptor antagonists

Also Published As

Publication number Publication date
EA200601514A1 (ru) 2007-02-27
ECSP066836A (es) 2006-11-24
SV2006002017A (es) 2006-05-09
NO20064298L (no) 2006-11-24
CA2556423A1 (en) 2005-09-01
WO2005079769A3 (en) 2007-01-04
GT200500032A (es) 2005-10-31
US20080119471A1 (en) 2008-05-22
JP2007523126A (ja) 2007-08-16
ZA200607970B (en) 2008-12-31
CR8584A (es) 2007-08-28
AR048068A1 (es) 2006-03-29
PA8624501A1 (es) 2006-07-03
TW200539882A (en) 2005-12-16
AU2005215156A1 (en) 2005-09-01
PE20051129A1 (es) 2006-02-16
IL177406A0 (en) 2006-12-10
KR20070033961A (ko) 2007-03-27
EP1727526A2 (en) 2006-12-06
CN101090723A (zh) 2007-12-19
WO2005079769A2 (en) 2005-09-01

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]