AR044473A1 - Derivados de isoindolinona, su uso como insecticidas y procedimientos de preparacion - Google Patents
Derivados de isoindolinona, su uso como insecticidas y procedimientos de preparacionInfo
- Publication number
- AR044473A1 AR044473A1 ARP040101902A ARP040101902A AR044473A1 AR 044473 A1 AR044473 A1 AR 044473A1 AR P040101902 A ARP040101902 A AR P040101902A AR P040101902 A ARP040101902 A AR P040101902A AR 044473 A1 AR044473 A1 AR 044473A1
- Authority
- AR
- Argentina
- Prior art keywords
- case
- alkyl
- formula
- group
- together form
- Prior art date
Links
- PXZQEOJJUGGUIB-UHFFFAOYSA-N isoindolin-1-one Chemical class C1=CC=C2C(=O)NCC2=C1 PXZQEOJJUGGUIB-UHFFFAOYSA-N 0.000 title abstract 3
- 239000002917 insecticide Substances 0.000 title abstract 2
- 238000000034 method Methods 0.000 title 1
- -1 3-trifluoromethylanilino Chemical group 0.000 abstract 11
- 125000000217 alkyl group Chemical group 0.000 abstract 10
- 125000001188 haloalkyl group Chemical group 0.000 abstract 6
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 4
- 125000004414 alkyl thio group Chemical group 0.000 abstract 4
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 4
- 229910052736 halogen Inorganic materials 0.000 abstract 4
- 150000002367 halogens Chemical group 0.000 abstract 4
- 125000002490 anilino group Chemical group [H]N(*)C1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 abstract 3
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 2
- 125000005278 alkyl sulfonyloxy group Chemical group 0.000 abstract 2
- 229910052801 chlorine Inorganic materials 0.000 abstract 2
- 239000000460 chlorine Substances 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 125000004108 n-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 125000001664 diethylamino group Chemical group [H]C([H])([H])C([H])([H])N(*)C([H])([H])C([H])([H])[H] 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000001972 isopentyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000006318 tert-butyl amino group Chemical group [H]N(*)C(C([H])([H])[H])(C([H])([H])[H])C([H])([H])[H] 0.000 abstract 1
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/50—Iso-indoles; Hydrogenated iso-indoles with oxygen and nitrogen atoms in positions 1 and 3
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
- A01N43/38—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Indole Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Reivindicación 1: Uso de derivados de isoindolinona de fórmula (1) en donde a) A1 representa H, y A2 representa uno de los siguiente grupos de fórmula (2) o b) A1 y A2 forman juntos =N-R2 o un grupo de fórmula (3), y A3 representa -R2 o el grupo de fórmula (4); R1 representa halógeno, alquilo, alcoxi, alquiltio, alquilsulfonilo, alquilsulfoniloxi, haloalquilo, haloalcoxi o nitro, m representa 0, 1, 2, 3 ó 4, en donde R1 puede ser idéntico o diferente en el caso de que m represente un entero de 2 o más, R2 representa alquilo que está opcionalmente sustituido con alquiltio, alquilsulfinilo o alquilsulfonilo, R3 representa H o alquilo, R4 representa halógeno, alquilo, haloalquilo que está opcionalmente sustituido con hidroxi, haloalcoxi o fenilo que está opcionalmente sustituido con haloalquilo, n representa 0, 1, 2, 3 o 4, en donde R4 puede ser idéntico o diferente en el caso de que m represente un entero de 2 o más, como insecticidas. Reivindicación 2: Derivados de isoindolinona de fórmula (5) en donde a) A11 representa H, y A12 representa uno de los siguientes grupos de fórmula (6) o b) A11 y A12 forman juntos =N-R12 o un grupo de fórmula (7) y A13 representa -R12 o el grupo de fórmula (8); R11 representa halógeno, alquilo, alcoxi, alquiltio, alquilsulfonilo, alquilsulfoniloxi, haloalquilo, haloalcoxi o nitro, p representa 0, 1, 2, 3, o 4, en donde R11 puede ser idéntico o diferente en el caso de que p represente un entero de 2 o más, R12 representa alquilo que está opcionalmente sustituido con alquiltio, alquilsulfinilo o alquilsulfonilo, R13 representa H o alquilo, R14 representa halógeno, alquilo, haloalquilo que está opcionalmente sustituido con hidroxi, haloalcoxi o fenilo que está opcionalmente sustituido con haloalquilo, q representa 0, 1, 2, 3 o 4, en donde R14 puede ser idéntico o diferente en el caso de que m represente un entero de 2 o más, con la excepción de los siguientes casos (E-1)-(E-11); (E-1) el caso en donde A11 representa H, A12 representa anilino, A13 representa terc-butilo, y p representa 0, (E-2) el caso en donde A11 representa H, A12 representa 2-flúor-4-metilanilino o 3-trifluorometilanilino, A13 representa n-butilo o 3-metilbutilo, (E-3) el caso en donde A11 representa H, A12 representa el grupo -NH-R12, A13 representa -R12, R12 en los grupos antes mencionados representa al mismo tiempo etilo, isopropilo, n-butilo, 1-metil-n-hexilo o n-dodecilo, y p representa 0, (E-4) el caso en donde A11 representa H, A12 representa terc-butilamino o dietilamino, A13 representa metilo, y p representa 0; (E-5) el caso en donde A11 representa un átomo de H, A12 representa anilino o 2-metilanilino, A13 representa fenilo, y p representa 0, (E-6) el caso en donde A11 y A12 forman juntos metilimino o etilimino, A13 representa 2,6-di(isopropil)fenilo, y p representa 0, (E-7) el caso en donde A11 y A12 forman juntos el grupo =N-alquilo, A13 representa 2,6-dietilfenilo, y p representa 0 o p representa 1 y R11 representa alquilo inferior, (E-8) el caso en donde A11 y A12 forman juntos fenilimino, A13 representa metilo o n-propilo, y p representa 0, (E-9) el caso en donde A11 y A12 juntos representan el grupo =N-R12, A13 representa -R12, R12 en los grupos mencionados representa al mismo tiempo alquilo C1-5, y p representa 0; (E-10) el caso en donde A11 y A12 forman juntos 4-metilanilino, A13 representa anilino o 4-metilanilino, y p representa 0; (E-11) el caso en donde A11 y A12 forman juntos el grupo de fórmula (7), A13 representa el grupo de fórmula (8), R14 en los grupos antes mencionados cada uno representa independientemente metilo o cloro, q representa 0 o 1; y p representa 1 y R11 representa Cl o Br.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2003162176A JP2004359633A (ja) | 2003-06-06 | 2003-06-06 | イソインドリノン誘導体の殺虫剤としての利用 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR044473A1 true AR044473A1 (es) | 2005-09-14 |
Family
ID=33549179
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP040101902A AR044473A1 (es) | 2003-06-06 | 2004-06-03 | Derivados de isoindolinona, su uso como insecticidas y procedimientos de preparacion |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20070031514A1 (es) |
| EP (1) | EP1635639A1 (es) |
| JP (2) | JP2004359633A (es) |
| KR (1) | KR20060031612A (es) |
| CN (1) | CN1802091A (es) |
| AR (1) | AR044473A1 (es) |
| AU (1) | AU2004246765A1 (es) |
| BR (1) | BRPI0411209A (es) |
| MX (1) | MXPA05012987A (es) |
| TW (1) | TW200503619A (es) |
| WO (1) | WO2004110149A1 (es) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5554319B2 (ja) | 2008-04-01 | 2014-07-23 | アボット ゲーエムベーハー ウント カンパニー カーゲー | テトラヒドロイソキノリン類、それを含む医薬組成物および治療におけるそれの使用 |
| AR075442A1 (es) | 2009-02-16 | 2011-03-30 | Abbott Gmbh & Co Kg | Derivados de aminotetralina, composiciones farmaceuticas que las contienen y sus usos en terapia |
| US8846743B2 (en) | 2010-08-13 | 2014-09-30 | Abbott Laboratories | Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US9051280B2 (en) | 2010-08-13 | 2015-06-09 | AbbVie Deutschland GmbH & Co. KG | Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US8883839B2 (en) | 2010-08-13 | 2014-11-11 | Abbott Laboratories | Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US8877794B2 (en) | 2010-08-13 | 2014-11-04 | Abbott Laboratories | Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US9045459B2 (en) | 2010-08-13 | 2015-06-02 | AbbVie Deutschland GmbH & Co. KG | Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US9309200B2 (en) | 2011-05-12 | 2016-04-12 | AbbVie Deutschland GmbH & Co. KG | Benzazepine derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US8853196B2 (en) | 2011-08-05 | 2014-10-07 | AbbVie Deutschland GmbH & Co. KG | Aminochromane, aminothiochromane and amino-1,2,3,4-tetrahydroquinoline derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US8846741B2 (en) | 2011-11-18 | 2014-09-30 | Abbvie Inc. | N-substituted aminobenzocycloheptene, aminotetraline, aminoindane and phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US9365512B2 (en) * | 2012-02-13 | 2016-06-14 | AbbVie Deutschland GmbH & Co. KG | Isoindoline derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US9650334B2 (en) | 2013-03-15 | 2017-05-16 | Abbvie Inc. | Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy |
| US9656955B2 (en) | 2013-03-15 | 2017-05-23 | Abbvie Inc. | Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy |
| KR20160062165A (ko) | 2013-10-17 | 2016-06-01 | 아비에 도이치란트 게엠베하 운트 콤파니 카게 | 아미노테트랄린 및 아미노인단 유도체, 이들을 포함하는 약제학적 조성물, 및 치료에서 이들의 용도 |
| WO2015055770A1 (en) | 2013-10-17 | 2015-04-23 | AbbVie Deutschland GmbH & Co. KG | Aminochromane, aminothiochromane and amino-1,2,3,4-tetrahydroquinoline derivatives, pharmaceutical compositions containing them, and their use in therapy |
| JP2018197192A (ja) * | 2015-10-13 | 2018-12-13 | 石原産業株式会社 | チエノピロール系化合物又はその塩を有効成分として含有する有害生物防除剤 |
| CN117158429A (zh) * | 2022-05-27 | 2023-12-05 | 农心作物科技股份有限公司 | 一种增效杀螨组合物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1055094A (en) * | 1965-02-23 | 1967-01-11 | Shell Int Research | Novel phosphorus-containing esters |
| US4164406A (en) * | 1975-07-11 | 1979-08-14 | Monsanto Company | Phosphinylphthalimidines and their use as plant growth regulants |
| JPS53144570A (en) * | 1977-05-18 | 1978-12-15 | Sankyo Co Ltd | 1-osoindolinone derivatives and agriculture and horticulture containing the same as active constituents |
| US6362369B2 (en) * | 1997-11-25 | 2002-03-26 | Nihon Nohyaku Co., Ltd. | Phthalic acid diamide derivatives fluorine-containing aniline compounds as starting material, agricultural and horticultural insecticides, and a method for application of the insecticides |
| EP1216988A4 (en) * | 1999-09-28 | 2005-04-20 | Nihon Nohyaku Co Ltd | THIOALKYLAMINE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
-
2003
- 2003-06-06 JP JP2003162176A patent/JP2004359633A/ja active Pending
-
2004
- 2004-05-25 WO PCT/EP2004/005600 patent/WO2004110149A1/en active Application Filing
- 2004-05-25 AU AU2004246765A patent/AU2004246765A1/en not_active Abandoned
- 2004-05-25 US US10/558,459 patent/US20070031514A1/en not_active Abandoned
- 2004-05-25 JP JP2006508198A patent/JP2006527172A/ja not_active Withdrawn
- 2004-05-25 KR KR1020057023082A patent/KR20060031612A/ko not_active Application Discontinuation
- 2004-05-25 EP EP04739332A patent/EP1635639A1/en not_active Withdrawn
- 2004-05-25 CN CNA2004800157750A patent/CN1802091A/zh active Pending
- 2004-05-25 MX MXPA05012987A patent/MXPA05012987A/es unknown
- 2004-05-25 BR BRPI0411209-1A patent/BRPI0411209A/pt not_active IP Right Cessation
- 2004-06-03 AR ARP040101902A patent/AR044473A1/es not_active Application Discontinuation
- 2004-06-04 TW TW093116042A patent/TW200503619A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1802091A (zh) | 2006-07-12 |
| KR20060031612A (ko) | 2006-04-12 |
| AU2004246765A1 (en) | 2004-12-23 |
| WO2004110149A1 (en) | 2004-12-23 |
| TW200503619A (en) | 2005-02-01 |
| EP1635639A1 (en) | 2006-03-22 |
| MXPA05012987A (es) | 2006-03-16 |
| BRPI0411209A (pt) | 2006-07-18 |
| JP2006527172A (ja) | 2006-11-30 |
| US20070031514A1 (en) | 2007-02-08 |
| JP2004359633A (ja) | 2004-12-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |