AR041069A1 - Composicion de tolterodina liquida oral - Google Patents

Composicion de tolterodina liquida oral

Info

Publication number
AR041069A1
AR041069A1 ARP030103101A ARP030103101A AR041069A1 AR 041069 A1 AR041069 A1 AR 041069A1 AR P030103101 A ARP030103101 A AR P030103101A AR P030103101 A ARP030103101 A AR P030103101A AR 041069 A1 AR041069 A1 AR 041069A1
Authority
AR
Argentina
Prior art keywords
composition
concentration
tolterodine
therapeutically effective
agent
Prior art date
Application number
ARP030103101A
Other languages
English (en)
Inventor
Joseph Reo
Kathryn Kienle
Jennifer Fredrickson
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of AR041069A1 publication Critical patent/AR041069A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Composición farmacéutica en forma de un líquido administrable por vía oral comprende agua que tiene disuelta una sal soluble en agua farmacéuticamente aceptable de un compuesto relacionado con la tolterodina a una concentración terapéuticamente eficaz de la composición. La composición tiene un pH de aproximadamente 2 a aproximadamente 6 y comprende adicionalmente un agente edulcorante y un agente antimacrobiano a una concentración que es antimicrobianamente eficaz al pH de la composición. La composición es útil para tratar un trastorno mediado por receptores muscarínicos, más particularmente vejiga hiperactiva, en un paciente, mediante administración por vía oral al mismo de una cantidad terapéuticamente eficaz de la composición. Reivindicación 1: Una composición farmacéutica en forma de un líquido administrable por vía oral, caracterizada porque comprende la composición agua que tiene disuelta una sal soluble en agua farmacéuticamente aceptable de un compuesto relacionado con la tolterodina a una concentración terapéuticamente eficaz en la composición; donde la composición tiene un pH de aproximadamente 2 aproximadamente 6, preferiblemente de aproximadamente 3 aproximadamente 5 y más preferiblemente de aproximadamente 3,5 a aproximadamente 4,5, y comprende adicionalmente un agente edulcorante y un agente antimicrobiano a una concentración que es antimicrobianamente eficaz al pH de la composición.
ARP030103101A 2002-08-28 2003-08-27 Composicion de tolterodina liquida oral AR041069A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US40642902P 2002-08-28 2002-08-28

Publications (1)

Publication Number Publication Date
AR041069A1 true AR041069A1 (es) 2005-04-27

Family

ID=31978300

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP030103101A AR041069A1 (es) 2002-08-28 2003-08-27 Composicion de tolterodina liquida oral

Country Status (10)

Country Link
US (1) US7101888B2 (es)
EP (1) EP1536780A1 (es)
JP (1) JP2006500381A (es)
AR (1) AR041069A1 (es)
AU (1) AU2003265680A1 (es)
BR (1) BR0313714A (es)
CA (1) CA2496806A1 (es)
MX (1) MXPA05002302A (es)
TW (1) TW200413027A (es)
WO (1) WO2004019925A1 (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20080066997A (ko) 2005-11-10 2008-07-17 바스프 에스이 유해 진균 방제용 트리티코나졸을 위한 완화제로서의피라클로스트로빈의 용도
CZ298448B6 (cs) * 2006-08-09 2007-10-03 Zentiva, A. S. Farmaceutická kompozice s obsahem tolterodinu
US8871275B2 (en) 2007-08-08 2014-10-28 Inventia Healthcare Private Limited Extended release compositions comprising tolterodine
US20090214665A1 (en) * 2008-02-26 2009-08-27 Lai Felix S Controlled Release Muscarinic Receptor Antagonist Formulation
CN102238954A (zh) 2008-11-04 2011-11-09 肯塔基大学研究基金会 基于d-塔格糖的组合物以及用于预防和治疗动脉粥样硬化、代谢综合征及其症状的方法
EP2386289A1 (en) * 2010-04-29 2011-11-16 Ipsen Pharma S.A.S. Clay compositions
DE102012202193A1 (de) 2012-02-14 2013-08-14 Evonik Degussa Gmbh pH-eingestelltes Süßungsmittel
US8568747B1 (en) 2012-10-05 2013-10-29 Silvergate Pharmaceuticals, Inc. Enalapril compositions
US9463183B1 (en) 2015-10-30 2016-10-11 Silvergate Pharmaceuticals, Inc. Lisinopril formulations
US9669008B1 (en) 2016-03-18 2017-06-06 Silvergate Pharmaceuticals, Inc. Enalapril formulations
GR1009534B (el) * 2017-11-21 2019-05-31 Laboserve Φαρμακευτικη Βιομηχανια Α.Ε. Ποσιμα φαρμακευτικα διαλυματα που περιλαμβανουν υδροχλωρικη οξυβουτυνινη
CN111925294A (zh) * 2020-07-06 2020-11-13 济南大学 一种托特罗定帕莫酸盐及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20000057548A (ko) * 1996-12-13 2000-09-25 알프레드 엘. 미첼슨 광학적 전송물질 및 결합재
SE9803871D0 (sv) * 1998-11-11 1998-11-11 Pharmacia & Upjohn Ab Therapeutic method and formulation
US20030060513A1 (en) * 2001-09-27 2003-03-27 Arneric Stephen P. Pharmaceutical composition
US7005449B2 (en) * 2002-04-23 2006-02-28 Pharmacia & Upjohn Company Tolterodine salts

Also Published As

Publication number Publication date
US20050032905A1 (en) 2005-02-10
JP2006500381A (ja) 2006-01-05
WO2004019925A1 (en) 2004-03-11
EP1536780A1 (en) 2005-06-08
BR0313714A (pt) 2005-06-28
AU2003265680A1 (en) 2004-03-19
US7101888B2 (en) 2006-09-05
CA2496806A1 (en) 2004-03-11
TW200413027A (en) 2004-08-01
MXPA05002302A (es) 2005-06-08

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal