AR039428A1 - Sal de perindopril y composiciones farmaceuticas que las contienen - Google Patents

Sal de perindopril y composiciones farmaceuticas que las contienen

Info

Publication number
AR039428A1
AR039428A1 ARP030101332A ARP030101332A AR039428A1 AR 039428 A1 AR039428 A1 AR 039428A1 AR P030101332 A ARP030101332 A AR P030101332A AR P030101332 A ARP030101332 A AR P030101332A AR 039428 A1 AR039428 A1 AR 039428A1
Authority
AR
Argentina
Prior art keywords
salt
perindoprile
pharmaceutical compositions
compositions containing
carbonyloxybutylamino
Prior art date
Application number
ARP030101332A
Other languages
English (en)
Inventor
Gerard Damien
Francois Lefoulon
Bernard Marchand
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8871521&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR039428(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Servier Lab filed Critical Servier Lab
Publication of AR039428A1 publication Critical patent/AR039428A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Abstract

Una sal de perindopril (ácido(2S)-2-((1S)-carbetoxibutilamino)-1-oxopropil-(2S, 3aS, 7aS) perhidroindol carboxílico) inhibidor de la enzima de conversión de la angiotensina I (ICE "CEI"), útil en el tratamiento de la hipertensión arterial y de la insuficiencia cardíaca.
ARP030101332A 2002-04-18 2003-04-16 Sal de perindopril y composiciones farmaceuticas que las contienen AR039428A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0204847A FR2838648B1 (fr) 2002-04-18 2002-04-18 Nouveau sel de perindopril et les compositions pharmaceutiques qui le contiennent

Publications (1)

Publication Number Publication Date
AR039428A1 true AR039428A1 (es) 2005-02-16

Family

ID=8871521

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP030101332A AR039428A1 (es) 2002-04-18 2003-04-16 Sal de perindopril y composiciones farmaceuticas que las contienen

Country Status (38)

Country Link
US (1) US6696481B2 (es)
EP (1) EP1354873B1 (es)
JP (1) JP3737488B2 (es)
KR (1) KR100542468B1 (es)
CN (1) CN1211365C (es)
AP (1) AP1787A (es)
AR (1) AR039428A1 (es)
AT (1) ATE271036T1 (es)
AU (2) AU2003222921A1 (es)
BR (1) BR0300709A (es)
CA (1) CA2423825C (es)
CR (1) CR7576A (es)
DE (1) DE60300011T2 (es)
DK (1) DK1354873T3 (es)
EA (1) EA005676B1 (es)
EC (1) ECSP045441A (es)
ES (1) ES2224092T3 (es)
FR (1) FR2838648B1 (es)
GE (1) GEP20074211B (es)
HK (1) HK1057367A1 (es)
HR (1) HRP20041079B1 (es)
IL (1) IL164424A (es)
IS (1) IS2842B (es)
MA (1) MA27115A1 (es)
ME (1) ME00454B (es)
MX (1) MXPA03002346A (es)
NO (1) NO324323B1 (es)
NZ (1) NZ524478A (es)
OA (1) OA12806A (es)
PL (1) PL359321A1 (es)
PT (1) PT1354873E (es)
RS (1) RS51694B (es)
SI (1) SI1354873T1 (es)
TN (1) TNSN04206A1 (es)
TR (1) TR200401793T4 (es)
UA (1) UA79463C2 (es)
WO (1) WO2003087050A2 (es)
ZA (1) ZA200301395B (es)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2395195A (en) * 2002-11-18 2004-05-19 Cipla Ltd Preparation of perindopril from carboxy-protected precursor, & perindopril monohydrates for use as angiotensin converting enzyme (ACE) inhibitors
LT1729739T (lt) * 2004-03-29 2016-11-10 Les Laboratoires Servier Kietos farmacinės kompozicijos gamybos būdas
SI21800A (sl) 2004-05-14 2005-12-31 Krka, Tovarna Zdravil, D.D., Novo Mesto Nov postopek sinteze perindoprila
DK1679072T5 (da) * 2005-01-06 2009-04-20 Ipca Lab Ltd Fremgangsmåde til syntese af (2S,3aS,7aS)-1-(S)-alanyl-octahydro-1H-indol-2-carboxylsyrederivater og anvendelse i syntesen af perindopril
EA012420B1 (ru) * 2005-03-14 2009-10-30 Ле Лаборатуар Сервье Улучшенный способ очистки периндоприла
FR2894825B1 (fr) * 2005-12-21 2010-12-03 Servier Lab Nouvelle association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion et les compositions pharmaceutiques qui la contiennent
FR2897865B1 (fr) * 2006-02-28 2008-04-18 Servier Lab Forme cristalline beta du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2897866B1 (fr) * 2006-02-28 2008-04-18 Servier Lab Forme cristalline alpha du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
GB0624090D0 (en) * 2006-12-01 2007-01-10 Selamine Ltd Ramipril amine salts
GB0624087D0 (en) * 2006-12-01 2007-01-10 Selamine Ltd Ramipril combination salt
GB0624084D0 (en) * 2006-12-01 2007-01-10 Selamine Ltd Ramipril amino acid salts
SI22542A (sl) * 2007-06-04 2008-12-31 Diagen D.O.O. Stabilna formulacija amorfnih soli perindoprila, postopek za njeno pripravo v industrijskem merilu in njena uporaba za zdravljenje hipertenzije
WO2009157018A2 (en) * 2008-06-24 2009-12-30 Matrix Laboratories Ltd Novel polymorphic forms of perindopril (l)-arginine and process for the preparation thereof
AU2009212902A1 (en) * 2008-09-03 2010-03-18 Apotex Pharmachem Inc. Amorphous form of an L-arginine salt of perindopril and processes of preparation thereof
CN101766598A (zh) * 2008-12-31 2010-07-07 东英（江苏）药业有限公司 含有培哚普利的药物组合物
GB0910692D0 (en) 2009-06-20 2009-08-05 Teva Pharma Compound
SI23149A (sl) 2009-09-21 2011-03-31 Silverstone Pharma Nove benzatinske soli ACE inhibitorjev, postopek za njihovo pripravo in njihova uporaba za zdravljenje kardiovaskularnih bolezni
FR2961105B1 (fr) * 2010-06-15 2013-02-08 Servier Lab Utilisation de l'association d'un inhibiteur du courant if sinusal et d'un inhibiteur de l'enzyme de conversion de l'angiotensine pour le traitement de l'insuffisance cardiaque
FR2985511B1 (fr) * 2012-01-05 2014-01-03 Servier Lab Forme cristalline delta du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent
FR2985512B1 (fr) * 2012-01-05 2014-06-20 Servier Lab Procede de preparation du sel de l-arginine du perindopril
CN103172696B (zh) * 2012-12-19 2014-12-17 宁波美诺华药业股份有限公司 一种γ晶型的培哚普利精氨酸盐的制备方法
FR3040303B1 (fr) * 2015-08-27 2019-04-05 Les Laboratoires Servier Suivi Par Sabine Goudeau-Wenger Composition pharmaceutique comprenant un inhibiteur de la hmg-coa reductase et un inhibiteur eca
FR3050380B1 (fr) 2016-04-20 2020-07-10 Les Laboratoires Servier Composition pharmaceutique comprenant un betabloquant, un inhibiteur de l'enzyme de conversion et un antihypertenseur ou un ains.
EP3842035A1 (en) 2019-12-23 2021-06-30 KRKA, d.d., Novo mesto Composition for the preparation of perindopril arginine granules, a method for their preparation and pharmaceutical composition comprising the granules
SI26268A (sl) 2021-11-18 2023-05-31 Zupet Rok Postopek za pripravo hidratirane oblike perindopril l-arginina

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2503155A2 (fr) * 1980-10-02 1982-10-08 Science Union & Cie Nouveaux imino diacides substitues, leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme
FR2811320B1 (fr) * 2000-07-06 2002-08-23 Adir Nouvelle forme cristalline alpha du sel de tert-butylamine du perindopril, son procede de preparation et les compositions pharmaceutiques qui la contiennent

Also Published As

Publication number Publication date
TR200401793T4 (tr) 2004-08-23
CR7576A (es) 2008-08-21
ZA200301395B (en) 2003-09-02
AP2004003154A0 (en) 2004-12-31
NO324323B1 (no) 2007-09-24
MXPA03002346A (es) 2005-08-26
IL164424A0 (en) 2005-12-18
OA12806A (en) 2006-07-11
SI1354873T1 (en) 2004-12-31
HK1057367A1 (en) 2004-04-02
JP3737488B2 (ja) 2006-01-18
CA2423825C (fr) 2006-02-21
EP1354873B1 (fr) 2004-07-14
DE60300011D1 (de) 2004-08-19
EP1354873A1 (fr) 2003-10-22
JP2003321493A (ja) 2003-11-11
FR2838648A1 (fr) 2003-10-24
EA005676B1 (ru) 2005-04-28
KR20030082902A (ko) 2003-10-23
PL359321A1 (en) 2003-10-20
HRP20041079B1 (hr) 2013-04-30
GEP20074211B (en) 2007-10-10
NO20030849D0 (no) 2003-02-24
DK1354873T3 (da) 2004-11-01
IS2842B (is) 2013-08-15
ATE271036T1 (de) 2004-07-15
US6696481B2 (en) 2004-02-24
UA79463C2 (en) 2007-06-25
TNSN04206A1 (en) 2007-03-12
RS90904A (en) 2007-02-05
AU2003200700A1 (en) 2003-11-06
KR100542468B1 (ko) 2006-01-11
ES2224092T3 (es) 2005-03-01
ME00454B (me) 2011-10-10
HRP20041079A2 (en) 2004-12-31
CN1451656A (zh) 2003-10-29
IL164424A (en) 2010-12-30
NZ524478A (en) 2004-05-28
CA2423825A1 (fr) 2003-10-18
US20030199568A1 (en) 2003-10-23
AU2003222921A1 (en) 2003-10-27
EA200300334A1 (ru) 2003-12-25
FR2838648B1 (fr) 2004-05-21
WO2003087050A3 (fr) 2004-03-25
AU2003222921A8 (en) 2003-10-27
IS7516A (is) 2004-10-27
RS51694B (en) 2011-10-31
AP1787A (en) 2007-10-04
NO20030849L (no) 2003-10-20
BR0300709A (pt) 2004-09-08
PT1354873E (pt) 2004-10-29
AU2003200700C1 (en) 2015-04-23
WO2003087050A2 (fr) 2003-10-23
CN1211365C (zh) 2005-07-20
AU2003200700B2 (en) 2005-01-20
MA27115A1 (fr) 2004-12-20
ECSP045441A (es) 2005-03-10
DE60300011T2 (de) 2005-03-17

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Legal Events

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