AR032695A1 - Composicion farmaceutica - Google Patents

Composicion farmaceutica

Info

Publication number
AR032695A1
AR032695A1 ARP020100516A ARP020100516A AR032695A1 AR 032695 A1 AR032695 A1 AR 032695A1 AR P020100516 A ARP020100516 A AR P020100516A AR P020100516 A ARP020100516 A AR P020100516A AR 032695 A1 AR032695 A1 AR 032695A1
Authority
AR
Argentina
Prior art keywords
pharmaceutical composition
thieno
benzylamino
pyrimidin
benzo
Prior art date
Application number
ARP020100516A
Other languages
English (en)
Inventor
Schreder Sven Dr
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of AR032695A1 publication Critical patent/AR032695A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Organic Chemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Composicion farmacéutica de elevada biodisponibilidad para la administracion oral de ácido 4-[4-(3-cloro-4-metoxi-bencilamino)-benzo [4,5] tieno [2,3-d]pirimidin-2-il]-ciclohexancarboxílico y/o ácido 4-[4-(3-cloro-4hidroxi-bencilamino)-benzo[4,5]tieno[2,3]-dpirimidin-2-il]-ciclohexancarboxílico o de sus sales aptas para uso farmacéutico, con un procedimiento para preparar la composicion farmacéutica y con su uso.
ARP020100516A 2001-02-16 2002-02-15 Composicion farmaceutica AR032695A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10107261A DE10107261B4 (de) 2001-02-16 2001-02-16 Pharmazeutische Zusammensetzung

Publications (1)

Publication Number Publication Date
AR032695A1 true AR032695A1 (es) 2003-11-19

Family

ID=7674278

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020100516A AR032695A1 (es) 2001-02-16 2002-02-15 Composicion farmaceutica

Country Status (21)

Country Link
US (1) US20040082600A1 (es)
EP (1) EP1385521A2 (es)
JP (1) JP2004519489A (es)
KR (1) KR20030074822A (es)
CN (1) CN1649592A (es)
AR (1) AR032695A1 (es)
BR (1) BR0207271A (es)
CA (1) CA2438401A1 (es)
CZ (1) CZ20032423A3 (es)
DE (1) DE10107261B4 (es)
EC (1) ECSP034769A (es)
EE (1) EE200300378A (es)
HU (1) HUP0303141A3 (es)
IL (1) IL157411A0 (es)
MX (1) MXPA03007318A (es)
PE (1) PE20021039A1 (es)
PL (1) PL364467A1 (es)
RU (1) RU2003127393A (es)
SK (1) SK11352003A3 (es)
WO (1) WO2002072100A2 (es)
ZA (1) ZA200307216B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101065115A (zh) * 2004-11-24 2007-10-31 默克公司 取代酰胺的液体和半固体口服药物制剂
WO2013109354A2 (en) * 2011-12-07 2013-07-25 Texas Southern University Etravirine formulations and uses thereof
JP6943384B2 (ja) * 2017-03-01 2021-09-29 ヱスビー食品株式会社 食品の食感劣化防止用ソフトカプセル、並びに、該食感劣化防止用ソフトカプセル及び食用油を含有する食品

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0517412A1 (en) * 1991-06-03 1992-12-09 MERCK SHARP & DOHME LTD. Pharmaceutical formulations of a benzodiazepine
DE19819023A1 (de) * 1998-04-29 1999-11-04 Merck Patent Gmbh Thienopyrimidine
DE19928146A1 (de) * 1999-06-19 2000-12-21 Merck Patent Gmbh Thienopyrimidine
EP1255565A1 (de) * 2000-01-13 2002-11-13 MERCK PATENT GmbH Pharmazeutische zubereitungen enthaltend 2-pyrrolidon als lösungsvermittler
DE10001021A1 (de) * 2000-01-13 2001-07-19 Merck Patent Gmbh Pharmazeutische Zubereitung

Also Published As

Publication number Publication date
PE20021039A1 (es) 2002-11-14
US20040082600A1 (en) 2004-04-29
HUP0303141A2 (hu) 2003-12-29
EE200300378A (et) 2003-10-15
WO2002072100A2 (en) 2002-09-19
MXPA03007318A (es) 2003-12-04
SK11352003A3 (sk) 2003-12-02
DE10107261A1 (de) 2002-09-12
CA2438401A1 (en) 2002-09-19
DE10107261B4 (de) 2005-03-10
JP2004519489A (ja) 2004-07-02
EP1385521A2 (en) 2004-02-04
WO2002072100A3 (en) 2003-11-06
CN1649592A (zh) 2005-08-03
BR0207271A (pt) 2004-03-23
ECSP034769A (es) 2003-12-24
HUP0303141A3 (en) 2006-05-29
ZA200307216B (en) 2005-01-13
IL157411A0 (en) 2004-03-28
PL364467A1 (en) 2004-12-13
RU2003127393A (ru) 2005-01-20
KR20030074822A (ko) 2003-09-19
CZ20032423A3 (en) 2004-07-14

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal