AR026731A1 - Procedimiento para fabricar tienopirimidinas - Google Patents

Procedimiento para fabricar tienopirimidinas

Info

Publication number
AR026731A1
AR026731A1 ARP000106452A ARP000106452A AR026731A1 AR 026731 A1 AR026731 A1 AR 026731A1 AR P000106452 A ARP000106452 A AR P000106452A AR P000106452 A ARP000106452 A AR P000106452A AR 026731 A1 AR026731 A1 AR 026731A1
Authority
AR
Argentina
Prior art keywords
tienopirimidines
procedure
manufacturing
formula
acid
Prior art date
Application number
ARP000106452A
Other languages
English (en)
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of AR026731A1 publication Critical patent/AR026731A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings

Abstract

Un procedimiento para obtener compuestos de la Formula (1) por el cual, un éster del ácido 2-aminobenzotiofen-3-carboxílico de la Formula (2) se transformacon un nitrilo de la Formula N:::C-R1 en un solvente en solucion o suspension, en presencia de un ácido.
ARP000106452A 1999-12-07 2000-12-06 Procedimiento para fabricar tienopirimidinas AR026731A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19958926A DE19958926A1 (de) 1999-12-07 1999-12-07 Verfahren zur Herstellung von Thienopyrimidinen

Publications (1)

Publication Number Publication Date
AR026731A1 true AR026731A1 (es) 2003-02-26

Family

ID=7931692

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000106452A AR026731A1 (es) 1999-12-07 2000-12-06 Procedimiento para fabricar tienopirimidinas

Country Status (19)

Country Link
US (1) US6689885B2 (es)
EP (1) EP1244675A1 (es)
JP (1) JP2003516406A (es)
KR (1) KR20020053888A (es)
CN (1) CN1407988A (es)
AR (1) AR026731A1 (es)
AU (1) AU2006401A (es)
BR (1) BR0016170A (es)
CA (1) CA2392692A1 (es)
CZ (1) CZ20021847A3 (es)
DE (1) DE19958926A1 (es)
HU (1) HUP0203754A2 (es)
MX (1) MXPA02005084A (es)
NO (1) NO20022671L (es)
PL (1) PL355153A1 (es)
RU (1) RU2002118333A (es)
SK (1) SK7542002A3 (es)
WO (1) WO2001042248A1 (es)
ZA (1) ZA200203794B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7274295B2 (en) * 2002-10-30 2007-09-25 At&T Bls Intellectual Property, Inc. Instantaneous mobile access to all pertinent life events

Also Published As

Publication number Publication date
CN1407988A (zh) 2003-04-02
RU2002118333A (ru) 2003-12-20
MXPA02005084A (es) 2004-08-23
BR0016170A (pt) 2002-08-20
AU2006401A (en) 2001-06-18
US6689885B2 (en) 2004-02-10
KR20020053888A (ko) 2002-07-05
NO20022671D0 (no) 2002-06-06
WO2001042248A1 (de) 2001-06-14
PL355153A1 (en) 2004-04-05
CZ20021847A3 (cs) 2002-10-16
JP2003516406A (ja) 2003-05-13
DE19958926A1 (de) 2001-06-13
US20030096994A1 (en) 2003-05-22
HUP0203754A2 (hu) 2003-03-28
CA2392692A1 (en) 2001-06-14
EP1244675A1 (de) 2002-10-02
SK7542002A3 (en) 2002-12-03
ZA200203794B (en) 2003-11-26
NO20022671L (no) 2002-06-06

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Legal Events

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