NO20022671L - Fremgangsmåte for fremstilling av tienopyrimidiner - Google Patents

Fremgangsmåte for fremstilling av tienopyrimidiner

Info

Publication number
NO20022671L
NO20022671L NO20022671A NO20022671A NO20022671L NO 20022671 L NO20022671 L NO 20022671L NO 20022671 A NO20022671 A NO 20022671A NO 20022671 A NO20022671 A NO 20022671A NO 20022671 L NO20022671 L NO 20022671L
Authority
NO
Norway
Prior art keywords
preparation
formula
thienopyrimidines
aminobenzothiophene
nitrile
Prior art date
Application number
NO20022671A
Other languages
English (en)
Other versions
NO20022671D0 (no
Inventor
Horst Juraszyk
Peter Wendel
Markus Woissyk
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of NO20022671D0 publication Critical patent/NO20022671D0/no
Publication of NO20022671L publication Critical patent/NO20022671L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Oppfinnelsen vedrører en fremgangsmåte for fremstilling av forbindelser med formel (I). En 2-aminobenzotiofen-3-karboksylsyreester med formel (II)omsettes med et nitril med formel (III). i oppløsning eller suspensjon i et oppløsningsmiddel i nærvær av en syre.
NO20022671A 1999-12-07 2002-06-06 Fremgangsmåte for fremstilling av tienopyrimidiner NO20022671L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19958926A DE19958926A1 (de) 1999-12-07 1999-12-07 Verfahren zur Herstellung von Thienopyrimidinen
PCT/EP2000/012351 WO2001042248A1 (de) 1999-12-07 2000-12-07 Verfahren zur herstellung von thienopyrimidinen

Publications (2)

Publication Number Publication Date
NO20022671D0 NO20022671D0 (no) 2002-06-06
NO20022671L true NO20022671L (no) 2002-06-06

Family

ID=7931692

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20022671A NO20022671L (no) 1999-12-07 2002-06-06 Fremgangsmåte for fremstilling av tienopyrimidiner

Country Status (19)

Country Link
US (1) US6689885B2 (no)
EP (1) EP1244675A1 (no)
JP (1) JP2003516406A (no)
KR (1) KR20020053888A (no)
CN (1) CN1407988A (no)
AR (1) AR026731A1 (no)
AU (1) AU2006401A (no)
BR (1) BR0016170A (no)
CA (1) CA2392692A1 (no)
CZ (1) CZ20021847A3 (no)
DE (1) DE19958926A1 (no)
HU (1) HUP0203754A2 (no)
MX (1) MXPA02005084A (no)
NO (1) NO20022671L (no)
PL (1) PL355153A1 (no)
RU (1) RU2002118333A (no)
SK (1) SK7542002A3 (no)
WO (1) WO2001042248A1 (no)
ZA (1) ZA200203794B (no)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7274295B2 (en) * 2002-10-30 2007-09-25 At&T Bls Intellectual Property, Inc. Instantaneous mobile access to all pertinent life events

Also Published As

Publication number Publication date
US20030096994A1 (en) 2003-05-22
MXPA02005084A (es) 2004-08-23
US6689885B2 (en) 2004-02-10
NO20022671D0 (no) 2002-06-06
PL355153A1 (en) 2004-04-05
DE19958926A1 (de) 2001-06-13
EP1244675A1 (de) 2002-10-02
HUP0203754A2 (hu) 2003-03-28
RU2002118333A (ru) 2003-12-20
AR026731A1 (es) 2003-02-26
KR20020053888A (ko) 2002-07-05
BR0016170A (pt) 2002-08-20
AU2006401A (en) 2001-06-18
CZ20021847A3 (cs) 2002-10-16
CA2392692A1 (en) 2001-06-14
JP2003516406A (ja) 2003-05-13
ZA200203794B (en) 2003-11-26
SK7542002A3 (en) 2002-12-03
CN1407988A (zh) 2003-04-02
WO2001042248A1 (de) 2001-06-14

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application