AR019279A1 - Forma medicamentosa solida de estructura polifasica para la aplicacion oral que contiene gatifloxacina o sus sales o hidratos farmaceuticamente aplicables, y procedimiento para su preparacion. - Google Patents

Forma medicamentosa solida de estructura polifasica para la aplicacion oral que contiene gatifloxacina o sus sales o hidratos farmaceuticamente aplicables, y procedimiento para su preparacion.

Info

Publication number
AR019279A1
AR019279A1 ARP990102177A ARP990102177A AR019279A1 AR 019279 A1 AR019279 A1 AR 019279A1 AR P990102177 A ARP990102177 A AR P990102177A AR P990102177 A ARP990102177 A AR P990102177A AR 019279 A1 AR019279 A1 AR 019279A1
Authority
AR
Argentina
Prior art keywords
procedure
preparation
salts
pharmaceutically applicable
oral application
Prior art date
Application number
ARP990102177A
Other languages
English (en)
Inventor
Betzing Juergen Dr
Bartholomaeus Johannes Dr
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of AR019279A1 publication Critical patent/AR019279A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Forma medicamentosa solida de estructura polifásica para aplicacion oral, que consiste en gatifloxacina o sus sales o hidratos farmacéuticamente aplicables, y auxiliares elegidos del grupo que comprende cargas, aglutinantes, lubricantes, promotoresd e disgregacion o sus mezclas, que comprende una fase interior quecontiene la sustancia activa gatifloxacina o sus sales o hidratos farmacéuticamente aplicables, auxiliares elegidos del grupo que comprende aglutinantes,cargas, promotores dedisgregaci on o sus mezclas, y al menos una fase exterior que contiene como componente necesario al menos un promotor de disgregacion, yotros auxiliares elegidos del grupo que comprende al menos un lubricante, y eventualmente cargas y/oeventualmente aglutinant es. Procedimietno para lapreparacion de la forma medicamentosa solida.
ARP990102177A 1998-05-09 1999-05-07 Forma medicamentosa solida de estructura polifasica para la aplicacion oral que contiene gatifloxacina o sus sales o hidratos farmaceuticamente aplicables, y procedimiento para su preparacion. AR019279A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19820801A DE19820801A1 (de) 1998-05-09 1998-05-09 Orale Arzneiformen mit reproduzierbarer Wirkstofffreisetzung von Gatifloxacin oder pharmazeutisch verwendbaren Salzen oder Hydraten

Publications (1)

Publication Number Publication Date
AR019279A1 true AR019279A1 (es) 2002-02-13

Family

ID=7867223

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP990102177A AR019279A1 (es) 1998-05-09 1999-05-07 Forma medicamentosa solida de estructura polifasica para la aplicacion oral que contiene gatifloxacina o sus sales o hidratos farmaceuticamente aplicables, y procedimiento para su preparacion.

Country Status (28)

Country Link
US (1) US6291462B1 (es)
EP (1) EP1077703B1 (es)
JP (1) JP2002514600A (es)
KR (1) KR100587210B1 (es)
CN (1) CN1198615C (es)
AR (1) AR019279A1 (es)
AT (1) ATE235242T1 (es)
AU (1) AU753482B2 (es)
BR (1) BR9910350A (es)
CA (1) CA2325636A1 (es)
CO (1) CO5050341A1 (es)
DE (2) DE19820801A1 (es)
DK (1) DK1077703T3 (es)
ES (1) ES2195573T3 (es)
HK (1) HK1033281A1 (es)
HU (1) HUP0101597A3 (es)
IL (1) IL139512A0 (es)
MY (1) MY118569A (es)
NO (1) NO20005385L (es)
NZ (1) NZ507968A (es)
PE (1) PE20000480A1 (es)
PL (1) PL343936A1 (es)
PT (1) PT1077703E (es)
RU (1) RU2226394C2 (es)
SK (1) SK16772000A3 (es)
UA (1) UA60364C2 (es)
WO (1) WO1999058129A1 (es)
ZA (1) ZA200006440B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL148820A0 (en) * 1999-10-08 2002-09-12 Smithkline Beecham Corp Fab i inhibitors
US6413969B1 (en) * 2000-09-13 2002-07-02 Bristol-Myers Squibb Company Gatifloxacin pentahydrate
AU2002367773A1 (en) * 2001-04-06 2003-11-03 Affinium Pharmaceuticals, Inc. Fab i inhibitors
US6589955B2 (en) * 2001-06-20 2003-07-08 Bristol-Myers Squibb Company Pediatric formulation of gatifloxacin
US7790709B2 (en) 2002-12-06 2010-09-07 Affinium Pharmaceuticals, Inc. Heterocyclic compounds, methods of making them and their use in therapy
WO2004082586A2 (en) 2003-03-17 2004-09-30 Affinium Pharmaceuticals, Inc. Phamaceutical compositions comprising inhibitors of fab i and further antibiotics
US20050031683A1 (en) * 2003-08-04 2005-02-10 Ashish Kapoor Solid pharmaceutical composition
WO2005021000A1 (en) * 2003-08-28 2005-03-10 Ranbaxy Laboratories Limited Solid oral dosage forms of gatifloxacin
MY148773A (en) * 2004-03-17 2013-05-31 Novartis Ag Galenic formulations of organic compounds
PT1828167E (pt) * 2004-06-04 2014-10-08 Debiopharm Int Sa Derivados de acrilamida como agentes antibióticos
US20060247255A1 (en) * 2005-05-02 2006-11-02 Patel Satishkumar A Method for preparing a stable gatifloxacin composition
ES2358682T3 (es) * 2005-08-02 2011-05-12 Baxter International Inc. Recipientes de múltiples cámaras.
WO2007067416A2 (en) * 2005-12-05 2007-06-14 Affinium Pharmaceuticals, Inc. Heterocyclylacrylamide compounds as fabi inhibitors and antibacterial agents
EP2687533B1 (en) 2006-07-20 2017-07-19 Debiopharm International SA Acrylamide derivatives as FAB I inhibitors
CN100415212C (zh) * 2006-07-21 2008-09-03 哈药集团制药总厂 一种含乳酸卡德沙星的口服制剂
CA2563690C (en) * 2006-10-12 2014-10-07 Pharmascience Inc. Pharmaceutical compositions comprising intra- and extra- granular fractions
EP2125802A4 (en) 2007-02-16 2014-08-20 Debiopharm Int Sa SALTS, PRODRUGS AND POLYMORPHES OF FAB I INHIBITORS
RS58898B1 (sr) 2012-06-19 2019-08-30 Debiopharm Int Sa Prolek derivati (e)-n-metil-n-((3-metilbenzofuran-2-il)metil)-3-(7-okso-5,6,7,8-tetrahidro-1,8-naftiridin-3-il)akrilamida
LT3419628T (lt) 2016-02-26 2021-01-25 Debiopharm International Sa Medikamentas diabetinėms pėdų infekcijoms gydyti

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH089597B2 (ja) * 1986-01-21 1996-01-31 杏林製薬株式会社 選択毒性に優れた8‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法
PL169106B1 (pl) * 1991-01-30 1996-06-28 Wellcome Found Sposób wytwarzania dyspergowalnej w wodzie tabletki PL PL PL PL PL PL PL
GB9109862D0 (en) * 1991-05-08 1991-07-03 Beecham Lab Sa Pharmaceutical formulations
US5436253A (en) * 1993-09-08 1995-07-25 Daiichi Pharmaceutical Co., Ltd. Pyridonecarboxylic acid derivatives and mycotic infections
EP0797987B1 (en) * 1994-12-19 2003-10-15 Daiichi Pharmaceutical Co., Ltd. Sustained-release granular preparation and process for producing the same
US5945124A (en) * 1995-07-05 1999-08-31 Byk Gulden Chemische Fabrik Gmbh Oral pharmaceutical composition with delayed release of active ingredient for pantoprazole
US5837292A (en) * 1996-07-03 1998-11-17 Yamanouchi Europe B.V. Granulate for the preparation of fast-disintegrating and fast-dissolving compositions containing a high amount of drug

Also Published As

Publication number Publication date
SK16772000A3 (sk) 2001-05-10
CA2325636A1 (en) 1999-11-18
CN1300216A (zh) 2001-06-20
UA60364C2 (uk) 2003-10-15
HUP0101597A3 (en) 2003-01-28
RU2226394C2 (ru) 2004-04-10
KR100587210B1 (ko) 2006-06-08
AU753482B2 (en) 2002-10-17
DE59904737D1 (de) 2003-04-30
HK1033281A1 (en) 2001-08-24
MY118569A (en) 2004-12-31
PT1077703E (pt) 2003-08-29
PL343936A1 (en) 2001-09-10
EP1077703B1 (de) 2003-03-26
IL139512A0 (en) 2001-11-25
JP2002514600A (ja) 2002-05-21
DE19820801A1 (de) 1999-11-25
HUP0101597A2 (hu) 2001-11-28
CN1198615C (zh) 2005-04-27
ZA200006440B (en) 2002-02-08
KR20010043408A (ko) 2001-05-25
BR9910350A (pt) 2001-09-25
DK1077703T3 (da) 2003-06-23
AU4035299A (en) 1999-11-29
NO20005385D0 (no) 2000-10-26
NZ507968A (en) 2002-12-20
US6291462B1 (en) 2001-09-18
PE20000480A1 (es) 2000-05-20
NO20005385L (no) 2000-10-26
ES2195573T3 (es) 2003-12-01
EP1077703A1 (de) 2001-02-28
WO1999058129A1 (de) 1999-11-18
ATE235242T1 (de) 2003-04-15
CO5050341A1 (es) 2001-06-27

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