AR018935A1 - Compuesto derivado de la tienopiridina, proceso para producirlo, composicion farmaceutica que lo contiene, y su uso para elaborar dicha composicion - Google Patents

Compuesto derivado de la tienopiridina, proceso para producirlo, composicion farmaceutica que lo contiene, y su uso para elaborar dicha composicion

Info

Publication number
AR018935A1
AR018935A1 ARP990103031A ARP990103031A AR018935A1 AR 018935 A1 AR018935 A1 AR 018935A1 AR P990103031 A ARP990103031 A AR P990103031A AR P990103031 A ARP990103031 A AR P990103031A AR 018935 A1 AR018935 A1 AR 018935A1
Authority
AR
Argentina
Prior art keywords
substituted
compound derived
tienopiridine
prepare
produce
Prior art date
Application number
ARP990103031A
Other languages
English (en)
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of AR018935A1 publication Critical patent/AR018935A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un compuesto derivado de la tienopiridina de formula (I): caracterizado porque R1 representa a un grupo alquilo C1-7 que puede estar sustituido, un grupocicloalquilo C3-7 que puede estar sustituido, un grupo alcoxiamino C1-6 que puede estar sustituido o un hidroxiamino que puede estar sustituido; y R2representa a un grupo alquilo C1-7 que puede estar sustituido o un grupo fenilo que puede estar sustituido; cuando R1 es un grupo alquilo C1-7 no sustituido,entones R7 es un grupo alquilo C1-7 sustituido o un grupo fenilo sustituido o una sal del mismo. Poseen excelente actividad antagonismo de la hormonaliberadora de gonadotropina.
ARP990103031A 1998-06-26 1999-06-24 Compuesto derivado de la tienopiridina, proceso para producirlo, composicion farmaceutica que lo contiene, y su uso para elaborar dicha composicion AR018935A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP18126398 1998-06-26
JP33300498 1998-11-24

Publications (1)

Publication Number Publication Date
AR018935A1 true AR018935A1 (es) 2001-12-12

Family

ID=26500516

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP990103031A AR018935A1 (es) 1998-06-26 1999-06-24 Compuesto derivado de la tienopiridina, proceso para producirlo, composicion farmaceutica que lo contiene, y su uso para elaborar dicha composicion

Country Status (10)

Country Link
US (1) US6329388B2 (es)
JP (1) JP2000219691A (es)
KR (2) KR20010020155A (es)
CN (1) CN1306535A (es)
AR (1) AR018935A1 (es)
ID (1) ID26780A (es)
OA (1) OA11568A (es)
PL (1) PL345074A1 (es)
TR (1) TR200003784T2 (es)
TW (1) TW430665B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2407472A1 (en) * 2000-06-14 2002-10-23 Takeda Chemical Industries, Ltd. Sustained release compositions
WO2003064429A1 (fr) 2002-01-30 2003-08-07 Takeda Chemical Industries, Ltd. Thienopyrimidines, procedes de fabrication et d'utilisation correspondants
WO2003086464A1 (fr) * 2002-04-12 2003-10-23 Takeda Pharmaceutical Company Limited. Agents pour prevenir/traiter les bouffees de chaleur
CN101684123B (zh) * 2008-09-27 2013-12-11 四川大学 2-甲酰胺基噻吩并吡啶衍生物制备方法及医药用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW449600B (en) 1994-04-19 2001-08-11 Takeda Chemical Industries Ltd Condensed-ring thiophene derivatives, their production and use
JPH09169766A (ja) 1995-10-19 1997-06-30 Takeda Chem Ind Ltd チエノピリジン誘導体，その製造法および用途
ATE221534T1 (de) * 1995-12-08 2002-08-15 Takeda Chemical Industries Ltd Hemmer der prolaktinsynthese
WO1997041126A1 (en) 1996-04-26 1997-11-06 Takeda Chemical Industries, Ltd. Thienopyridine derivatives, their production and use

Also Published As

Publication number Publication date
JP2000219691A (ja) 2000-08-08
TW430665B (en) 2001-04-21
US6329388B2 (en) 2001-12-11
PL345074A1 (en) 2001-12-03
OA11568A (en) 2004-07-26
KR20010020155A (ko) 2001-03-15
KR20000012154A (ko) 2000-02-25
TR200003784T2 (tr) 2001-06-21
CN1306535A (zh) 2001-08-01
ID26780A (id) 2001-02-08
US20010001104A1 (en) 2001-05-10

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