AP3546A - Amides of 2-amino-4-arylthiazole compounds and their salts - Google Patents
Amides of 2-amino-4-arylthiazole compounds and their saltsInfo
- Publication number
- AP3546A AP3546A AP2014008076A AP2014008076A AP3546A AP 3546 A AP3546 A AP 3546A AP 2014008076 A AP2014008076 A AP 2014008076A AP 2014008076 A AP2014008076 A AP 2014008076A AP 3546 A AP3546 A AP 3546A
- Authority
- AP
- ARIPO
- Prior art keywords
- amides
- salts
- amino
- arylthiazole compounds
- arylthiazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
- C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T428/00—Stock material or miscellaneous articles
- Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
- Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1687MU2012 | 2012-06-08 | ||
US201261665282P | 2012-06-27 | 2012-06-27 | |
IN3519MU2012 | 2012-12-13 | ||
US201261748016P | 2012-12-31 | 2012-12-31 | |
PCT/IB2013/054703 WO2013183035A2 (en) | 2012-06-08 | 2013-06-08 | Amides of 2-amino-4-arylthiazole compounds and their salts |
Publications (2)
Publication Number | Publication Date |
---|---|
AP2014008076A0 AP2014008076A0 (en) | 2014-11-30 |
AP3546A true AP3546A (en) | 2016-01-14 |
Family
ID=54193746
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2014008076A AP3546A (en) | 2012-06-08 | 2013-06-08 | Amides of 2-amino-4-arylthiazole compounds and their salts |
Country Status (22)
Country | Link |
---|---|
US (1) | US9458173B2 (es) |
EP (1) | EP2858999B1 (es) |
JP (1) | JP5989900B2 (es) |
KR (1) | KR20150015488A (es) |
CN (1) | CN104350058A (es) |
AP (1) | AP3546A (es) |
AU (1) | AU2013273118B2 (es) |
BR (1) | BR112014029155A2 (es) |
CA (1) | CA2873570C (es) |
CL (1) | CL2014003317A1 (es) |
EA (1) | EA031334B1 (es) |
HK (1) | HK1207643A1 (es) |
IL (1) | IL236084A0 (es) |
IN (1) | IN2014MN02467A (es) |
MX (1) | MX354014B (es) |
MY (1) | MY165622A (es) |
NZ (1) | NZ701721A (es) |
PE (1) | PE20142306A1 (es) |
PH (1) | PH12014502685A1 (es) |
SG (1) | SG11201408093PA (es) |
WO (1) | WO2013183035A2 (es) |
ZA (1) | ZA201500082B (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR091279A1 (es) | 2012-06-08 | 2015-01-21 | Gilead Sciences Inc | Inhibidores macrociclicos de virus flaviviridae |
BR112014030630A2 (pt) | 2012-06-08 | 2017-06-27 | Gilead Sciences Inc | inibidores macrocíclicos de vírus flaviviridae |
BR112015030341A2 (pt) * | 2013-06-20 | 2017-07-25 | Glenmark Pharmaceuticals Sa | formulações de nanoparticulado e processo para prepará-las, composição farmacêutica e uso de composto ou seu sal farmaceuticamente aceitável e estabilizante de superfície |
WO2016023832A1 (en) * | 2014-08-11 | 2016-02-18 | Hydra Biosciences, Inc. | Thieno- and furo[2,3-d]pyrimidine-2,4[1h,3h]-dione derivatives as trpc5 modulators for the treatment of neuropsychiatric disorders |
US20190175599A1 (en) * | 2014-09-16 | 2019-06-13 | Glemark Pharmaceuticals S.A. | Trpa1 antagonist for the treatment of pain associated to diabetic neuropathic pain |
TW202321229A (zh) | 2021-08-18 | 2023-06-01 | 美商富曼西公司 | 殺真菌的取代的雜環化合物 |
CN114671875A (zh) * | 2022-04-27 | 2022-06-28 | 成都施贝康生物医药科技有限公司 | 新型二氢嘧啶类化合物、异构体或盐及其制备方法和用途 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010109334A2 (en) * | 2009-03-23 | 2010-09-30 | Glenmark Pharmaceuticals, S.A. | Thienopyrimidinedione derivatives as trpa1 modulators |
Family Cites Families (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2248231A1 (de) | 1972-10-02 | 1974-04-11 | Basf Ag | 3-aminoisothiazolo eckige klammer auf 3,4-d eckige klammer zu pyrimidine |
SE9701398D0 (sv) | 1997-04-15 | 1997-04-15 | Astra Pharma Prod | Novel compounds |
ES2193839B1 (es) * | 2001-06-22 | 2005-02-16 | Almirall Prodesfarma, S.A. | Nuevos derivados de 6-fenildihidropirrolpirimidindiona. |
AU2003253165A1 (en) | 2002-08-13 | 2004-02-25 | Warner-Lambert Company Llc | Pyrimidine fused bicyclic metalloproteinase inhibitors |
US6890923B2 (en) | 2002-12-16 | 2005-05-10 | Astrazeneca Ab | Compounds |
WO2004055054A1 (en) | 2002-12-18 | 2004-07-01 | Novartis Ag | Anktm1, a cold-activated trp-like channel expressed in nociceptive neurons |
EP1657238A4 (en) | 2003-08-22 | 2008-12-03 | Takeda Pharmaceutical | MERGED PYRIMIDINE DERIVATIVE AND USE THEREOF |
US20070099940A1 (en) | 2004-02-11 | 2007-05-03 | Spearing Paul K | Pth agonists |
WO2005089206A2 (en) | 2004-03-13 | 2005-09-29 | Irm Llc | Modulators of ion channel trpa1 |
JPWO2006083005A1 (ja) | 2005-02-03 | 2008-06-26 | 武田薬品工業株式会社 | 縮合ピリミジン誘導体およびその用途 |
AU2006278592A1 (en) | 2005-08-04 | 2007-02-15 | Apogee Biotechnology Corporation | Sphingosine kinase inhibitors and methods of their use |
US20070105920A1 (en) | 2005-11-08 | 2007-05-10 | Akzo Nobel N.V. | 2-(Benzimidazol-1-Yl)-N-(4-phenylthiazol-2-yl) acetamide derivatives |
CA2634152A1 (en) | 2005-12-22 | 2007-06-28 | Hydra Biosciences, Inc. | Trpa1 inhibitors for treating pain |
TW200800997A (en) | 2006-03-22 | 2008-01-01 | Astrazeneca Ab | Chemical compounds |
CN101454318A (zh) * | 2006-03-22 | 2009-06-10 | 阿斯利康(瑞典)有限公司 | 吡啶并嘧啶衍生物及其作为pde4抑制剂的用途 |
JP2011201776A (ja) | 2008-07-23 | 2011-10-13 | Mochida Pharmaceut Co Ltd | ヘテロシクリデン−n−(3,4−ジヒドロ−2(1h)−キナゾリノン−5−イル)アセトアミド誘導体 |
AR065081A1 (es) | 2007-01-29 | 2009-05-13 | Xenon Pharmaceuticals Inc | Compuestos de quinazolinona y pirimidona fusionados y composicion farmaceutica |
WO2009002933A1 (en) * | 2007-06-22 | 2008-12-31 | Hydra Biosciences, Inc. | Methods and compositions for treating disorders |
WO2010004390A1 (en) * | 2008-06-17 | 2010-01-14 | Glenmark Pharmaceuticals, S.A. | Quinazoline dione derivatives as trpa1 modulators |
WO2009158719A2 (en) | 2008-06-27 | 2009-12-30 | Hydra Biosciences, Inc. | Methods and compositions for treating disorders |
KR20120001746A (ko) | 2009-03-23 | 2012-01-04 | 그렌마크 파머수티칼스 에스. 아. | Trpa1 조절자로서 이소티아졸로-피리미딘디온 유도체 |
US8623880B2 (en) | 2009-03-23 | 2014-01-07 | Glenmark Pharmaceuticals S.A. | Fused pyrimidine-dione derivatives as TRPA1 modulators |
KR20110132575A (ko) | 2009-03-23 | 2011-12-08 | 그렌마크 파머수티칼스 에스. 아. | Trpa1 조절자로서 융합된 피리미딘디온 유도체 |
MY159059A (en) | 2010-12-20 | 2016-12-15 | Glenmark Pharmaceuticals Sa | 2-amino-4-arylthiazole compounds as trpa1 antagonists |
-
2013
- 2013-06-08 EP EP13742279.6A patent/EP2858999B1/en active Active
- 2013-06-08 CN CN201380030184.XA patent/CN104350058A/zh active Pending
- 2013-06-08 AP AP2014008076A patent/AP3546A/xx active
- 2013-06-08 NZ NZ701721A patent/NZ701721A/en not_active IP Right Cessation
- 2013-06-08 US US14/402,608 patent/US9458173B2/en active Active
- 2013-06-08 CA CA2873570A patent/CA2873570C/en active Active
- 2013-06-08 PE PE2014002226A patent/PE20142306A1/es not_active Application Discontinuation
- 2013-06-08 EA EA201492054A patent/EA031334B1/ru unknown
- 2013-06-08 AU AU2013273118A patent/AU2013273118B2/en not_active Ceased
- 2013-06-08 MY MYPI2014003389A patent/MY165622A/en unknown
- 2013-06-08 WO PCT/IB2013/054703 patent/WO2013183035A2/en active Application Filing
- 2013-06-08 IN IN2467MUN2014 patent/IN2014MN02467A/en unknown
- 2013-06-08 KR KR1020147033855A patent/KR20150015488A/ko active IP Right Grant
- 2013-06-08 JP JP2015515642A patent/JP5989900B2/ja not_active Expired - Fee Related
- 2013-06-08 BR BR112014029155A patent/BR112014029155A2/pt not_active Application Discontinuation
- 2013-06-08 SG SG11201408093PA patent/SG11201408093PA/en unknown
- 2013-06-08 MX MX2014014482A patent/MX354014B/es active IP Right Grant
-
2014
- 2014-12-02 PH PH12014502685A patent/PH12014502685A1/en unknown
- 2014-12-04 IL IL236084A patent/IL236084A0/en unknown
- 2014-12-04 CL CL2014003317A patent/CL2014003317A1/es unknown
-
2015
- 2015-01-07 ZA ZA2015/00082A patent/ZA201500082B/en unknown
- 2015-08-27 HK HK15108333.2A patent/HK1207643A1/xx unknown
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010109334A2 (en) * | 2009-03-23 | 2010-09-30 | Glenmark Pharmaceuticals, S.A. | Thienopyrimidinedione derivatives as trpa1 modulators |
WO2010109329A1 (en) * | 2009-03-23 | 2010-09-30 | Glenmark Pharmaceuticals, S.A. | Furopyrimidinedione derivatives as trpa1 modulators |
Also Published As
Publication number | Publication date |
---|---|
WO2013183035A3 (en) | 2014-02-27 |
PH12014502685B1 (en) | 2015-01-26 |
US20150111038A1 (en) | 2015-04-23 |
BR112014029155A2 (pt) | 2017-06-27 |
EA031334B1 (ru) | 2018-12-28 |
AP2014008076A0 (en) | 2014-11-30 |
IL236084A0 (en) | 2015-02-01 |
EP2858999A2 (en) | 2015-04-15 |
EP2858999B1 (en) | 2017-05-10 |
CN104350058A (zh) | 2015-02-11 |
NZ701721A (en) | 2016-03-31 |
JP2015520183A (ja) | 2015-07-16 |
WO2013183035A2 (en) | 2013-12-12 |
MX2014014482A (es) | 2015-06-05 |
JP5989900B2 (ja) | 2016-09-07 |
AU2013273118A1 (en) | 2014-11-27 |
CL2014003317A1 (es) | 2015-02-13 |
PE20142306A1 (es) | 2015-01-16 |
MX354014B (es) | 2018-02-08 |
AU2013273118B2 (en) | 2015-11-05 |
US9458173B2 (en) | 2016-10-04 |
PH12014502685A1 (en) | 2015-01-26 |
MY165622A (en) | 2018-04-18 |
CA2873570A1 (en) | 2013-12-12 |
IN2014MN02467A (es) | 2015-07-10 |
SG11201408093PA (en) | 2015-01-29 |
EA201492054A1 (ru) | 2016-08-31 |
ZA201500082B (en) | 2015-12-23 |
KR20150015488A (ko) | 2015-02-10 |
HK1207643A1 (en) | 2016-02-05 |
CA2873570C (en) | 2016-11-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
HRP20181628T1 (hr) | Spojevi i postupci za njihovu upotrebu | |
HK1208439A1 (en) | 5-azaindazole compounds and methods of use 5- | |
ZA201502503B (en) | Hppd variants and methods of use | |
HUE044300T2 (hu) | 3-amino-cikloalkil-vegyületek, mint ROR-GAMMA-T inhibitorok és alkalmazásuk | |
EP2938341A4 (en) | Heterocyclic compounds and methods for the use thereof | |
ZA201406082B (en) | Use of ccr3-inhibitors | |
HK1207643A1 (en) | Amides of 2-amino-4-arylthiazole compounds and their salts 2--4- | |
AP3611A (en) | Heterocyclic compounds and their uses | |
EP2938607A4 (en) | CRYSTALLINE SALTS AND FORMS | |
EP2881113A4 (en) | NEW APPLICATION OF POGOSTONE | |
EP2935227A4 (en) | DIAZOLAMIDE | |
HK1210168A1 (en) | Amine salt and crystals thereof |