ZA817187B - Medicament based on 2-amino-6-trifluoromethoxy-benzothiazole - Google Patents

Medicament based on 2-amino-6-trifluoromethoxy-benzothiazole

Info

Publication number
ZA817187B
ZA817187B ZA817187A ZA817187A ZA817187B ZA 817187 B ZA817187 B ZA 817187B ZA 817187 A ZA817187 A ZA 817187A ZA 817187 A ZA817187 A ZA 817187A ZA 817187 B ZA817187 B ZA 817187B
Authority
ZA
South Africa
Prior art keywords
benzothiazole
trifluoromethoxy
amino
medicament based
medicament
Prior art date
Application number
ZA817187A
Other languages
English (en)
Inventor
Jacques Mizoule
Original Assignee
Pharmindustrie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmindustrie filed Critical Pharmindustrie
Publication of ZA817187B publication Critical patent/ZA817187B/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82—Nitrogen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicinal Preparation (AREA)
ZA817187A 1980-10-17 1981-10-16 Medicament based on 2-amino-6-trifluoromethoxy-benzothiazole ZA817187B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8022218A FR2492258A1 (fr) 1980-10-17 1980-10-17 Nouveau medicament a base d'amino-2 trifluoromethoxy-6 benzothiazole

Publications (1)

Publication Number Publication Date
ZA817187B true ZA817187B (en) 1982-09-29

Family

ID=9247013

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA817187A ZA817187B (en) 1980-10-17 1981-10-16 Medicament based on 2-amino-6-trifluoromethoxy-benzothiazole

Country Status (16)

Country Link
US (1) US4370338A (xx)
EP (1) EP0050551B1 (xx)
JP (1) JPS5795910A (xx)
AR (1) AR227069A1 (xx)
AU (1) AU545437B2 (xx)
CA (1) CA1166159A (xx)
DE (1) DE3163230D1 (xx)
DK (1) DK444281A (xx)
FR (1) FR2492258A1 (xx)
GR (1) GR75804B (xx)
HU (1) HU184893B (xx)
IL (1) IL63880A0 (xx)
MA (1) MA19364A1 (xx)
NO (1) NO813492L (xx)
PT (1) PT73828B (xx)
ZA (1) ZA817187B (xx)

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FR2640624B1 (fr) * 1988-12-15 1994-08-12 Rhone Poulenc Sante Medicaments a base de derives de la benzothiazolamine-2, nouveaux derives et leur preparation
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FR2649705B2 (fr) * 1989-07-13 1994-09-23 Rhone Poulenc Sante Medicaments a base de derives de la benzothiazolamine-2, nouveaux derives et leur preparation
ES2043070T3 (es) * 1988-12-15 1993-12-16 Rhone Poulenc Sante Procedimiento para la preparacion de derivados de la benzotiazolamina-2.
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FR2649703B1 (fr) * 1989-07-13 1991-11-22 Rhone Poulenc Sante Derives d'imino-2 polyfluoroalcoxy-6 benzothiazole, leurs procedes de preparation et les medicaments les contenant
US5260297A (en) * 1989-07-13 1993-11-09 Rhone Poulenc Rorer, S.A. 2-imino-3-alkylbenzothiazoline derivatives bearing a heterocyclic substituent on the alkyl group, their preparation and medicinal products containing them.
FR2649702B1 (fr) * 1989-07-13 1991-11-22 Rhone Poulenc Sante Derives d'alkylimino-2 benzothiazoline, leurs procedes de preparation et les medicaments les contenant
FR2661910B1 (fr) * 1990-05-11 1992-08-21 Rhone Poulenc Sante Derives d'imino-2 heterocyclylalkyl-3 benzothiazoline, leur preparation et les medicaments les contenant.
ATE102612T1 (de) * 1989-07-13 1994-03-15 Rhone Poulenc Sante 2-imino-3 heterocyclylamino-benzothiazoline, ihre herstellung und sie enthaltende arzneimittel.
FR2649704B1 (fr) * 1989-07-13 1991-11-22 Rhone Poulenc Sante Derives d'imino-2 ethyl-3 benzothiazoline, leurs procedes de preparation et les medicaments les contenant
FR2662160B1 (fr) * 1990-05-18 1992-07-24 Rhone Poulenc Sante Derives d'alkylthio-3 propyl-3 benzothiazoline leur preparation et les medicaments les contenant.
FR2663030A1 (fr) * 1990-06-05 1991-12-13 Rhone Poulenc Sante Derives selenies de benzothiazoline leur preparation et les medicaments les contenant.
FR2662694A1 (fr) * 1990-06-05 1991-12-06 Rhone Poulenc Sante Derives du benzoselenazole, leur preparation et les medicaments les contenant.
FR2662695A1 (fr) * 1990-06-05 1991-12-06 Rhone Poulenc Sante Amino-2 polyfluoroalcoxy-6 benzoselenazoles, leur preparation et les medicaments les contenant.
FR2663029B1 (fr) * 1990-06-07 1992-07-31 Rhone Poulenc Sante Derives de benzothiazole, leur preparation et les medicaments les contenant.
FR2688138B1 (fr) * 1992-03-06 1995-05-05 Rhone Poulenc Rorer Sa Application de l'amino-2 trifluoromethoxy-6 benzothiazole pour obtenir un medicament destine au traitement de la sclerose laterale amyotrophique.
FR2699077B1 (fr) * 1992-12-16 1995-01-13 Rhone Poulenc Rorer Sa Application d'anticonvulsivants dans le traitement de lésions neurologiques liées à des traumatismes.
FR2700116B1 (fr) * 1993-01-07 1995-02-03 Rhone Poulenc Rorer Sa Application d'anticonvulsivants comme radioprotecteurs.
FR2700117B1 (fr) * 1993-01-07 1995-02-03 Rhone Poulenc Rorer Sa Application d'anticonvulsivants dans le traitement de la maladie de Parkinson et des syndromes parkinsoniens.
FR2702148B1 (fr) * 1993-03-05 1995-04-07 Rhone Poulenc Rorer Sa Application d'anticonvulsivants dans le traitement du neuro-sida.
FR2726271B1 (fr) * 1994-10-26 1996-12-06 Rhone Poulenc Rorer Sa Derives de 6-polyfluoroalcoxy-2-aminobenzothiazole
FR2786101B1 (fr) 1998-11-24 2002-07-05 Aventis Laboratoire Utilisation de la nicergoline dans le traitement de la spasticite
FR2787028B1 (fr) 1998-12-15 2002-10-18 Aventis Pharma Sa Utilisation du riluzole dans le traitement des traumatismes acoustiques
CA2361924A1 (en) * 1999-01-12 2000-07-20 Izumi Kamo Compositions for treating frequent urination and urinary incontinence
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CA2430298A1 (en) * 2000-11-30 2002-06-06 Banavara Lakshman Mylari Combination of gaba agonists and sorbitol dehydrogenase inhibitors
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EP1633400A2 (en) * 2003-05-16 2006-03-15 Pfizer Products Inc. Therapeutic combinations of atypical antipsychotics with gaba modulators, anticonvulsants or benzodiazapines
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EP1874353A1 (en) * 2005-04-05 2008-01-09 Yale University Glutamate modulating agents in the treatment of mental disorders
US9629817B2 (en) 2005-08-25 2017-04-25 Steven Michael Weiss Reducing myocardial damage and the incidence of arrhythmia arising from loss, reduction or interruption in coronary blood flow
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US3876653A (en) * 1973-03-26 1975-04-08 Kyowa Hakko Kogyo Kk Benzothiazole derivatives

Also Published As

Publication number Publication date
CA1166159A (fr) 1984-04-24
GR75804B (xx) 1984-08-02
NO813492L (no) 1982-04-19
DE3163230D1 (en) 1984-05-24
HU184893B (en) 1984-10-29
JPS5795910A (en) 1982-06-15
DK444281A (da) 1982-04-18
AU7654581A (en) 1982-04-22
PT73828B (fr) 1983-01-17
AU545437B2 (en) 1985-07-11
EP0050551A1 (fr) 1982-04-28
IL63880A0 (en) 1981-12-31
EP0050551B1 (fr) 1984-04-18
US4370338A (en) 1983-01-25
AR227069A1 (es) 1982-09-15
JPH0148884B2 (xx) 1989-10-20
PT73828A (fr) 1981-11-01
FR2492258A1 (fr) 1982-04-23
FR2492258B1 (xx) 1982-11-26
MA19364A1 (fr) 1982-07-01

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